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1 |
Material Type: Artigo
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Synthesis and antileishmanial evaluation of 1-aryl-4-(4,5-dihydro-1H-imidazol-2-yl)-1H-pyrazole derivativesdos Santos, Maurício S ; Oliveira, Mariana L.V ; Bernardino, Alice M.R ; de Léo, Rosa M ; Amaral, Veronica F ; de Carvalho, Flavia T ; Leon, Leonor L ; Canto-Cavalheiro, Marilene MBioorganic & medicinal chemistry letters, 2011-12, Vol.21 (24), p.7451-7454 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Discovery of new Gram-negative antivirulence drugs: Structure and properties of novel E. coli WaaC inhibitorsMoreau, F. ; Desroy, N. ; Genevard, J.M. ; Vongsouthi, V. ; Gerusz, V. ; Le Fralliec, G. ; Oliveira, C. ; Floquet, S. ; Denis, A. ; Escaich, S. ; Wolf, K. ; Busemann, M. ; Aschenbrenner, A.Bioorganic & medicinal chemistry, 2008-07, Vol.18 (14), p.4022-4026 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Oxoquinoline acyclonucleoside phosphonate analogues as a new class of specific inhibitors of human immunodeficiency virus type 1Faro, Letícia V. ; de Almeida, Jéssica M. ; Cirne-Santos, Cláudio C. ; Giongo, Viveca A. ; Castello-Branco, Luís R. ; Oliveira, Ingrid de B. ; Barbosa, Juliana E.F. ; Cunha, Anna C. ; Ferreira, Vítor F. ; de Souza, Marcos C. ; Paixão, Izabel C.N.P. ; de Souza, Maria Cecília B.V.Bioorganic & medicinal chemistry letters, 2012-08, Vol.22 (15), p.5055-5058 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Discovery of thiadiazoles as a novel structural class of potent and selective PDE7 inhibitors. Part 1: Design, synthesis and structure–activity relationship studiesVergne, Fabrice ; Bernardelli, Patrick ; Lorthiois, Edwige ; Pham, Nga ; Proust, Emmanuelle ; Oliveira, Chrystelle ; Mafroud, Abdel-Kader ; Royer, Frederique ; Wrigglesworth, Roger ; Schellhaas, Jennifer ; Barvian, Mark ; Moreau, François ; Idrissi, Moulay ; Tertre, Anita ; Bertin, Bernadette ; Coupe, Magali ; Berna, Patrick ; Soulard, PatriciaBioorganic & medicinal chemistry letters, 2004-09, Vol.14 (18), p.4607-4613 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Trypanocidal activity and redox potential of heterocyclic- and 2-hydroxy-naphthoquinonesGoulart, Marília O.F. ; Zani, Carlos L. ; Tonholo, Josealdo ; Freitas, Luciano R. ; de Abreu, Fabiane C. ; Oliveira, Alaíde B. ; Raslan, Délio S. ; Starling, Sérgia ; Chiari, EglerBioorganic & medicinal chemistry letters, 1997-08, Vol.7 (15), p.2043-2048 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Discovery of thiadiazoles as a novel structural class of potent and selective PDE7 inhibitors. Part 2: Metabolism-directed optimization studies towards orally bioavailable derivativesVergne, Fabrice ; Bernardelli, Patrick ; Lorthiois, Edwige ; Pham, Nga ; Proust, Emmanuelle ; Oliveira, Chrystelle ; Mafroud, Abdel-Kader ; Ducrot, Pierre ; Wrigglesworth, Roger ; Berlioz-Seux, Françoise ; Coleon, Francis ; Chevalier, Eric ; Moreau, François ; Idrissi, Moulay ; Tertre, Anita ; Descours, Arnaud ; Berna, Patrick ; Li, MeiBioorganic & medicinal chemistry letters, 2004-09, Vol.14 (18), p.4615-4621 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 1Lorthiois, Edwige ; Bernardelli, Patrick ; Vergne, Fabrice ; Oliveira, Chrystelle ; Mafroud, Abdel-Kader ; Proust, Emmanuelle ; Heuze, Lamia ; Moreau, François ; Idrissi, Moulay ; Tertre, Anita ; Bertin, Bernadette ; Coupe, Magali ; Wrigglesworth, Roger ; Descours, Arnaud ; Soulard, Patricia ; Berna, PatrickBioorganic & medicinal chemistry letters, 2004-09, Vol.14 (18), p.4623-4626 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
8 |
Material Type: Artigo
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Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 2: Optimization of 5,8-disubstituted derivativesBernardelli, Patrick ; Lorthiois, Edwige ; Vergne, Fabrice ; Oliveira, Chrystelle ; Mafroud, Abdel-Kader ; Proust, Emmanuelle ; Pham, Nga ; Ducrot, Pierre ; Moreau, François ; Idrissi, Moulay ; Tertre, Anita ; Bertin, Bernadette ; Coupe, Magali ; Chevalier, Eric ; Descours, Arnaud ; Berlioz-Seux, Françoise ; Berna, Patrick ; Li, MeiBioorganic & medicinal chemistry letters, 2004-09, Vol.14 (18), p.4627-4631 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |