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Refinado por: Nome da Publicação: Journal Of Medicinal Chemistry remover
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1
Novel Tricyclic-α-alkyloxyphenylpropionic Acids:  Dual PPARα/γ Agonists with Hypolipidemic and Antidiabetic Activity
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Artigo
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Novel Tricyclic-α-alkyloxyphenylpropionic Acids:  Dual PPARα/γ Agonists with Hypolipidemic and Antidiabetic Activity

Sauerberg, Per ; Pettersson, Ingrid ; Jeppesen, Lone ; Bury, Paul S ; Mogensen, John P ; Wassermann, Karsten ; Brand, Christian L ; Sturis, Jeppe ; Wöldike, Helle F ; Fleckner, Jan ; Andersen, Anne-Sofie T ; Mortensen, Steen B ; Svensson, L. Anders ; Rasmussen, Hanne B ; Lehmann, Søren V ; Polivka, Zdenek ; Sindelar, Karel ; Panajotova, Vladimira ; Ynddal, Lars ; Wulff, Erik M

Journal of medicinal chemistry, 2002-02, Vol.45 (4), p.789-804 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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2
Identification and Synthesis of a Novel Selective Partial PPARδ Agonist with Full Efficacy on Lipid Metabolism In Vitro and In Vivo
Material Type:
Artigo
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Identification and Synthesis of a Novel Selective Partial PPARδ Agonist with Full Efficacy on Lipid Metabolism In Vitro and In Vivo

Sauerberg, Per ; Olsen, Grith S ; Jeppesen, Lone ; Mogensen, John P ; Pettersson, Ingrid ; Jeppesen, Claus B ; Daugaard, Jens R ; Galsgaard, Elisabeth D ; Ynddal, Lars ; Fleckner, Jan ; Panajotova, Vladimira ; Polivka, Zdenek ; Pihera, Pavel ; Havranek, Miroslav ; Wulff, Erik M

Journal of medicinal chemistry, 2007-04, Vol.50 (7), p.1495-1503 [Periódico revisado por pares]

Washington, DC: American Chemical Society

Texto completo disponível

3
6-Chloro-3-alkylamino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide Derivatives Potently and Selectively Activate ATP Sensitive Potassium Channels of Pancreatic β-Cells
Material Type:
Artigo
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6-Chloro-3-alkylamino-4H-thieno[3,2-e]-1,2,4-thiadiazine 1,1-Dioxide Derivatives Potently and Selectively Activate ATP Sensitive Potassium Channels of Pancreatic β-Cells

Nielsen, Flemming E ; Bodvarsdottir, Thora B ; Worsaae, Anne ; MacKay, Peter ; Stidsen, Carsten E ; Boonen, Harrie C. M ; Pridal, Lone ; Arkhammar, Per O. G ; Wahl, Philip ; Ynddal, Lars ; Junager, Finn ; Dragsted, Nils ; Tagmose, Tina M ; Mogensen, John P ; Koch, Anette ; Treppendahl, Svend P ; Hansen, J. Bondo

Journal of medicinal chemistry, 2002-09, Vol.45 (19), p.4171-4187 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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4
Large Dimeric Ligands with Favorable Pharmacokinetic Properties and Peroxisome Proliferator-Activated Receptor Agonist Activity in Vitro and in Vivo
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Artigo
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Large Dimeric Ligands with Favorable Pharmacokinetic Properties and Peroxisome Proliferator-Activated Receptor Agonist Activity in Vitro and in Vivo

Sauerberg, Per ; Bury, Paul S ; Mogensen, John P ; Deussen, Heinz-Josef ; Pettersson, Ingrid ; Fleckner, Jan ; Nehlin, Jan ; Frederiksen, Klaus S ; Albrektsen, Tatjana ; Din, Nanni ; Svensson, L. Anders ; Ynddal, Lars ; Wulff, Erik M ; Jeppesen, Lone

Journal of medicinal chemistry, 2003-11, Vol.46 (23), p.4883-4894 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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5
Arylcyanoguanidines as Activators of Kir6.2/SUR1KATP Channels and Inhibitors of Insulin Release
Material Type:
Artigo
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Arylcyanoguanidines as Activators of Kir6.2/SUR1KATP Channels and Inhibitors of Insulin Release

Tagmose, Tina M ; Schou, Søren C ; Mogensen, John P ; Nielsen, Flemming E ; Arkhammar, Per O. G ; Wahl, Philip ; Hansen, Birgit S ; Worsaae, Anne ; Boonen, Harrie C. M ; Antoine, Marie-Hélène ; Lebrun, Philippe ; Hansen, John Bondo

Journal of medicinal chemistry, 2004-06, Vol.47 (12), p.3202-3211 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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6
Arylcyanoguanidines as activators of Kir6.2/SUR1K ATP channels and inhibitors of insulin release
Material Type:
Artigo
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Arylcyanoguanidines as activators of Kir6.2/SUR1K ATP channels and inhibitors of insulin release

Tagmose, Tina M ; Schou, Søren C ; Mogensen, John P ; Nielsen, Flemming E ; Arkhammar, Per O G ; Wahl, Philip ; Hansen, Birgit S ; Worsaae, Anne ; Boonen, Harrie C M ; Antoine, Marie-Hélène ; Lebrun, Philippe ; Hansen, John Bondo

Journal of medicinal chemistry, 2004-06, Vol.47 (12), p.3202-3211 [Periódico revisado por pares]

United States

Texto completo disponível

7
Identification and synthesis of a novel selective partial PPARdelta agonist with full efficacy on lipid metabolism in vitro and in vivo
Material Type:
Artigo
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Identification and synthesis of a novel selective partial PPARdelta agonist with full efficacy on lipid metabolism in vitro and in vivo

Sauerberg, Per ; Olsen, Grith S ; Jeppesen, Lone ; Mogensen, John P ; Pettersson, Ingrid ; Jeppesen, Claus B ; Daugaard, Jens R ; Galsgaard, Elisabeth D ; Ynddal, Lars ; Fleckner, Jan ; Panajotova, Vladimira ; Polivka, Zdenek ; Pihera, Pavel ; Havranek, Miroslav ; Wulff, Erik M

Journal of medicinal chemistry, 2007-04, Vol.50 (7), p.1495-1503 [Periódico revisado por pares]

United States

Texto completo disponível

8
6-Chloro-3-alkylamino-4 H -thieno[3,2 -e ]-1,2,4-thiadiazine 1,1-Dioxide Derivatives Potently and Selectively Activate ATP Sensitive Potassium Channels of Pancreatic β-Cells
Material Type:
Artigo
Adicionar ao Meu Espaço

6-Chloro-3-alkylamino-4 H -thieno[3,2 -e ]-1,2,4-thiadiazine 1,1-Dioxide Derivatives Potently and Selectively Activate ATP Sensitive Potassium Channels of Pancreatic β-Cells

Nielsen, Flemming E. ; Bodvarsdottir, Thora B. ; Worsaae, Anne ; MacKay, Peter ; Stidsen, Carsten E. ; Boonen, Harrie C. M. ; Pridal, Lone ; Arkhammar, Per O. G. ; Wahl, Philip ; Ynddal, Lars ; Junager, Finn ; Dragsted, Nils ; Tagmose, Tina M. ; Mogensen, John P. ; Koch, Anette ; Treppendahl, Svend P. ; Hansen, J. Bondo

Journal of medicinal chemistry, 2002-09, Vol.45 (19), p.4171-4187 [Periódico revisado por pares]

Texto completo disponível

9
Novel tricyclic-alpha-alkyloxyphenylpropionic acids: dual PPARalpha/gamma agonists with hypolipidemic and antidiabetic activity
Material Type:
Artigo
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Novel tricyclic-alpha-alkyloxyphenylpropionic acids: dual PPARalpha/gamma agonists with hypolipidemic and antidiabetic activity

Sauerberg, Per ; Pettersson, Ingrid ; Jeppesen, Lone ; Bury, Paul S ; Mogensen, John P ; Wassermann, Karsten ; Brand, Christian L ; Sturis, Jeppe ; Wöldike, Helle F ; Fleckner, Jan ; Andersen, Anne-Sofie T ; Mortensen, Steen B ; Svensson, L Anders ; Rasmussen, Hanne B ; Lehmann, Søren V ; Polivka, Zdenek ; Sindelar, Karel ; Panajotova, Vladimira ; Ynddal, Lars ; Wulff, Erik M

Journal of medicinal chemistry, 2002-02, Vol.45 (4), p.789-804 [Periódico revisado por pares]

United States

Texto completo disponível

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