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Material Type: Artigo
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Cyclin dependent kinase (CDK) inhibitors as anticancer drugs: Recent advances (2015–2019)Sánchez-Martínez, Concepción ; Lallena, María José ; Sanfeliciano, Sonia Gutiérrez ; de Dios, AlfonsoBioorganic & medicinal chemistry letters, 2019-10, Vol.29 (20), p.126637-126637, Article 126637 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Discovery of the pan-genotypic hepatitis C virus NS3/4A protease inhibitor voxilaprevir (GS-9857): A component of VoseviTaylor, James G. ; Zipfel, Sheila ; Ramey, Kyla ; Vivian, Randy ; Schrier, Adam ; Karki, Kapil K. ; Katana, Ashley ; Kato, Darryl ; Kobayashi, Tetsuya ; Martinez, Ruben ; Sangi, Michael ; Siegel, Dustin ; Tran, Chinh V. ; Yang, Zheng-Yu ; Zablocki, Jeff ; Yang, Cheng Y. ; Wang, Yujin ; Wang, Kelly ; Chan, Katie ; Barauskas, Ona ; Cheng, Guofeng ; Jin, Debi ; Schultz, Brian E. ; Appleby, Todd ; Villaseñor, Armando G. ; Link, John O.Bioorganic & medicinal chemistry letters, 2019-08, Vol.29 (16), p.2428-2436 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Semisynthesis and insecticidal bioactivities of benzoxazole and benzoxazolone derivatives of honokiol, a naturally occurring neolignan derived from Magnolia officinalisZhi, Xiao-yan ; Jiang, Ling-yun ; Li, Ting ; Song, Li-li ; Wang, Yi ; Cao, Hui ; Yang, ChunBioorganic & medicinal chemistry letters, 2020-05, Vol.30 (9), p.127086-127086, Article 127086 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Screening for tyrosinase inhibitors from actinomycetes; identification of trichostatin derivatives from Streptomyces sp. CA-129531 and scale up production in bioreactorGeorgousaki, Katerina ; Tsafantakis, Nikolaos ; Gumeni, Sentiljana ; Gonzalez, Ignacio ; Mackenzie, Thomas Andrew ; Reyes, Fernando ; Lambert, Carole ; Trougakos, Ioannis P. ; Genilloud, Olga ; Fokialakis, NikolasBioorganic & medicinal chemistry letters, 2020-03, Vol.30 (6), p.126952-126952, Article 126952 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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C–H activation reactions as useful tools for medicinal chemistsCaro-Diaz, Eduardo J.E. ; Urbano, Mariangela ; Buzard, Daniel J. ; Jones, Robert M.Bioorganic & medicinal chemistry letters, 2016-11, Vol.26 (22), p.5378-5383 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Development of curcumin–cyclodextrin/cellulose nanocrystals complexes: New anticancer drug delivery systemsNdong Ntoutoume, Gautier M.A. ; Granet, Robert ; Mbakidi, Jean Pierre ; Brégier, Frédérique ; Léger, David Y. ; Fidanzi-Dugas, Chloë ; Lequart, Vincent ; Joly, Nicolas ; Liagre, Bertrand ; Chaleix, Vincent ; Sol, VincentBioorganic & medicinal chemistry letters, 2016-02, Vol.26 (3), p.941-945 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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The SARS-CoV-2 main protease as drug targetUllrich, Sven ; Nitsche, ChristophBioorganic & medicinal chemistry letters, 2020-09, Vol.30 (17), p.127377-127377, Article 127377 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Discovery of velpatasvir (GS-5816): A potent pan-genotypic HCV NS5A inhibitor in the single-tablet regimens Vosevi® and EpclusaLink, John O. ; Taylor, James G. ; Trejo-Martin, Alejandra ; Kato, Darryl ; Katana, Ashley A. ; Krygowski, Evan S. ; Yang, Zheng-Yu ; Zipfel, Sheila ; Cottell, Jeromy J. ; Bacon, Elizabeth M. ; Tran, Chinh V. ; Yang, Cheng Y. ; Wang, Yujin ; Wang, Kelly W. ; Zhao, Guangyu ; Cheng, Guofeng ; Tian, Yang ; Gong, Ruoyu ; Lee, Yu-Jen ; Yu, Mei ; Gorman, Eric ; Mogalian, Erik ; Perry, Jason K.Bioorganic & medicinal chemistry letters, 2019-08, Vol.29 (16), p.2415-2427 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis of a heterotrifunctional linker for the site-specific preparation of antibody-drug conjugates with two distinct warheadsKumar, Amit ; Kinneer, Krista ; Masterson, Luke ; Ezeadi, Ebele ; Howard, Philip ; Wu, Herren ; Gao, Changshou ; Dimasi, NazzarenoBioorganic & medicinal chemistry letters, 2018-12, Vol.28 (23-24), p.3617-3621 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and antioxidant activities of novel 4-Schiff base-7-benzyloxy-coumarin derivativesZhang, Ye ; Zou, Biqun ; Chen, Zhenfeng ; Pan, Yingming ; Wang, Hengshan ; Liang, Hong ; Yi, XianghuiBioorganic & medicinal chemistry letters, 2011-11, Vol.21 (22), p.6811-6815 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |