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Material Type: Artigo
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Specific inhibitors of Plasmodium falciparum thioredoxin reductase as potential antimalarial agentsAndricopulo, A.D. ; Akoachere, M.B. ; Krogh, R. ; Nickel, C. ; McLeish, M.J. ; Kenyon, G.L. ; Arscott, L.D. ; Williams, C.H. ; Davioud-Charvet, E. ; Becker, K.Bioorganic & medicinal chemistry letters, 2006-04, Vol.16 (8), p.2283-2292 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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CoMFA and CoMSIA 3D QSAR Models for a Series of Cyclic Imides with Analgesic ActivityBorchhardt, D M ; Andricopulo, A DMedicinal chemistry (Shp-sariqah, United Arab Emirates), 2009-01, Vol.5 (1), p.66-73 [Periódico revisado por pares]Netherlands: Bentham Science Publishers LtdTexto completo disponível |
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Material Type: Artigo
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Structure−Activity Relationships for a Class of Inhibitors of Purine Nucleoside PhosphorylaseFarutin, Victor ; Masterson, Lori ; Andricopulo, Adriano D ; Cheng, Jianming ; Riley, Brad ; Hakimi, Ryan ; Frazer, Jack W ; Cordes, Eugene HJournal of medicinal chemistry, 1999-07, Vol.42 (13), p.2422-2431 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Structure-Activity Relationships for a Collection of Structurally Diverse Inhibitors of Purine Nucleoside PhosphorylaseANDRICOPULO, Adriano D. ; YUNES, Rosendo A.Chemical and Pharmaceutical Bulletin, 2001, Vol.49(1), pp.10-17 [Periódico revisado por pares]Tokyo: The Pharmaceutical Society of JapanTexto completo disponível |
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Material Type: Artigo
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Classical and Fragment-Based Hologram Structure-Activity Relationships for a Series of Analgesic Cyclic ImidesAndricopulo, A. ; Borchhardt, D. ; Castilho, M.Letters in drug design & discovery, 2008-01, Vol.5 (1), p.57-64 [Periódico revisado por pares]Bentham Science Publishers LtdTexto completo disponível |
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Material Type: Artigo
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Hologram QSAR model for the prediction of human oral bioavailabilityModa, Tiago L. ; Montanari, Carlos A. ; Andricopulo, Adriano D.Bioorganic & medicinal chemistry, 2007-12, Vol.15 (24), p.7738-7745 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Structure-Activity Relationships for the Design of Small-Molecule InhibitorsAndricopulo, Adriano D ; Montanari, Carlos AMini reviews in medicinal chemistry, 2005-06, Vol.5 (6), p.585-593 [Periódico revisado por pares]Netherlands: Bentham Science Publishers LtdTexto completo disponível |
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Material Type: Artigo
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Two- and three-dimensional quantitative structure–activity relationships for a series of purine nucleoside phosphorylase inhibitorsCastilho, Marcelo S. ; Postigo, Matheus P. ; de Paula, Caroline B.V. ; Montanari, Carlos A. ; Oliva, Glaucius ; Andricopulo, Adriano D.Bioorganic & medicinal chemistry, 2006-01, Vol.14 (2), p.516-527 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Hologram quantitative structure–activity relationships for a series of farnesoid X receptor activatorsHonorio, Kathia M. ; Garratt, Richard C. ; Andricopulo, Adriano D.Bioorganic & medicinal chemistry letters, 2005-06, Vol.15 (12), p.3119-3125 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Structure-activity relationships of novel inhibitors of glyceraldehyde-3-phosphate dehydrogenaseLEITAO, Andrei ; ANDRICOPULO, Adriano D ; MORAES, Valéria R. S ; MONTANARI, Carlos A ; OLIVA, Glaucius ; PUPO, Monica T ; DE MARCHI, Anderson A ; VIEIRA, Paulo C ; DA SILVA, Maria Fatima G. F ; FERREIRA, Vitor F ; DE SOUZA, Maria Cecilia B. V ; SA, Marcus MBioorganic & medicinal chemistry letters, 2004-05, Vol.14 (9), p.2199-2204 [Periódico revisado por pares]Oxford: ElsevierTexto completo disponível |