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11 |
Material Type: Artigo
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7‑Phenoxy-Substituted 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar PotencyGoffin, Eric ; Drapier, Thomas ; Larsen, Anja Probst ; Geubelle, Pierre ; Ptak, Christopher P ; Laulumaa, Saara ; Rovinskaja, Karoline ; Gilissen, Julie ; Tullio, Pascal de ; Olsen, Lars ; Frydenvang, Karla ; Pirotte, Bernard ; Hanson, Julien ; Oswald, Robert E ; Kastrup, Jette Sandholm ; Francotte, PierreJournal of medicinal chemistry, 2018-01, Vol.61 (1), p.251-264 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
12 |
Material Type: Artigo
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A review of traditional uses, phytochemistry and pharmacology of the genus IndigoferaGerometta, Elise ; Grondin, Isabelle ; Smadja, Jacqueline ; Frederich, Michel ; Gauvin-Bialecki, AnneJournal of ethnopharmacology, 2020-05, Vol.253, p.112608, Article 112608 [Periódico revisado por pares]Ireland: Elsevier B.VTexto completo disponível |
13 |
Material Type: Artigo
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Coumarins as factor XIIa inhibitors: Potency and selectivity improvements using a fragment-based strategyDavoine, Clara ; Traina, Amandine ; Evrard, Jonathan ; Lanners, Steve ; Fillet, Marianne ; Pochet, LionelEuropean journal of medicinal chemistry, 2023-11, Vol.259, p.115636-115636, Article 115636 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
14 |
Material Type: Artigo
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Oxidative Stress Status in COVID-19 Patients Hospitalized in Intensive Care Unit for Severe Pneumonia. A Pilot StudyPincemail, Joël ; Cavalier, Etienne ; Charlier, Corinne ; Cheramy-Bien, Jean-Paul ; Brevers, Eric ; Courtois, Audrey ; Fadeur, Marjorie ; Meziane, Smail ; Goff, Caroline Le ; Misset, Benoît ; Albert, Adelin ; Defraigne, Jean-Olivier ; Rousseau, Anne-FrançoiseAntioxidants, 2021-02, Vol.10 (2), p.257 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
15 |
Material Type: Artigo
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New insights in the development of positive allosteric modulators of α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptors belonging to 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxides: Introduction of (mono/difluoro)methyl groups at the 2-position of the thiadiazine ringGoffin, Eric ; Fraikin, Pierre ; Abboud, Dayana ; de Tullio, Pascal ; Beaufour, Caroline ; Botez, Iuliana ; Hanson, Julien ; Danober, Laurence ; Francotte, Pierre ; Pirotte, BernardEuropean journal of medicinal chemistry, 2023-03, Vol.250, p.115221-115221, Article 115221 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
16 |
Material Type: Artigo
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Chemical composition, cytotoxicity and in vitro antitrypanosomal and antiplasmodial activity of the essential oils of four Cymbopogon species from BeninKpoviessi, Salomé ; Bero, Joanne ; Agbani, Pierre ; Gbaguidi, Fernand ; Kpadonou-Kpoviessi, Bénédicta ; Sinsin, Brice ; Accrombessi, Georges ; Frédérich, Michel ; Moudachirou, Mansourou ; Quetin-Leclercq, JoëlleJournal of ethnopharmacology, 2014, Vol.151 (1), p.652-659 [Periódico revisado por pares]Ireland: Elsevier Ireland LtdTexto completo disponível |
17 |
Material Type: Artigo
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Natural Phenolic Compounds and Derivatives as Potential Antimalarial AgentsMamede, Lucia ; Ledoux, Allison ; Jansen, Olivia ; Frédérich, MichelPlanta medica, 2020-06, Vol.86 (9), p.585-618 [Periódico revisado por pares]Stuttgart · New York: Georg Thieme Verlag KGTexto completo disponível |
18 |
Material Type: Artigo
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Beware the Receptor VariantsHanson, JulienJournal of medicinal chemistry, 2023-12, Vol.66 (23), p.15671-15673 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
19 |
Material Type: Artigo
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1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activityLegru, Alice ; Verdirosa, Federica ; Hernandez, Jean-François ; Tassone, Giusy ; Sannio, Filomena ; Benvenuti, Manuela ; Conde, Pierre-Alexis ; Bossis, Guillaume ; Thomas, Caitlyn A. ; Crowder, Michael W. ; Dillenberger, Melissa ; Becker, Katja ; Pozzi, Cecilia ; Mangani, Stefano ; Docquier, Jean-Denis ; Gavara, LaurentEuropean journal of medicinal chemistry, 2021-12, Vol.226, p.113873-113873, Article 113873 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
20 |
Material Type: Artigo
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Metabolomics as a Challenging Approach for Medicinal Chemistry and Personalized MedicineFrédérich, Michel ; Pirotte, Bernard ; Fillet, Marianne ; de Tullio, PascalJournal of medicinal chemistry, 2016-10, Vol.59 (19), p.8649-8666 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |