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1
Ado-trastuzumab Emtansine (T-DM1): An Antibody–Drug Conjugate (ADC) for HER2-Positive Breast Cancer
Ado-trastuzumab Emtansine (T-DM1): An Antibody–Drug Conjugate (ADC) for HER2-Positive Breast Cancer
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Ado-trastuzumab Emtansine (T-DM1): An Antibody–Drug Conjugate (ADC) for HER2-Positive Breast Cancer

Lambert, John M ; Chari, Ravi V. J

Journal of medicinal chemistry, 2014-08, Vol.57 (16), p.6949-6964 [Periódico revisado por pares]

United States: American Chemical Society

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2
Synthesis, Pharmacological and Structural Characterization, and Thermodynamic Aspects of GluA2-Positive Allosteric Modulators with a 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxide Scaffold
Synthesis, Pharmacological and Structural Characterization, and Thermodynamic Aspects of GluA2-Positive Allosteric Modulators with a 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxide Scaffold
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Synthesis, Pharmacological and Structural Characterization, and Thermodynamic Aspects of GluA2-Positive Allosteric Modulators with a 3,4-Dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxide Scaffold

Nørholm, Ann-Beth ; Francotte, Pierre ; Olsen, Lars ; Krintel, Christian ; Frydenvang, Karla ; Goffin, Eric ; Challal, Sylvie ; Danober, Laurence ; Botez-Pop, Iuliana ; Lestage, Pierre ; Pirotte, Bernard ; Kastrup, Jette S

Journal of medicinal chemistry, 2013-11, Vol.56 (21), p.8736-8745 [Periódico revisado por pares]

United States: American Chemical Society

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3
Positive Allosteric Modulators of 2‑Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors Belonging to 4‑Cyclopropyl-3,4-dihydro‑2H‑1,2,4-pyridothiadiazine Dioxides and Diversely Chloro-Substituted 4‑Cyclopropyl-3,4-dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides
Positive Allosteric Modulators of 2‑Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors Belonging to 4‑Cyclopropyl-3,4-dihydro‑2H‑1,2,4-pyridothiadiazine Dioxides and Diversely Chloro-Substituted 4‑Cyclopropyl-3,4-dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides
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Positive Allosteric Modulators of 2‑Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors Belonging to 4‑Cyclopropyl-3,4-dihydro‑2H‑1,2,4-pyridothiadiazine Dioxides and Diversely Chloro-Substituted 4‑Cyclopropyl-3,4-dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides

Francotte, Pierre ; Nørholm, Ann-Beth ; Deva, Taru ; Olsen, Lars ; Frydenvang, Karla ; Goffin, Eric ; Fraikin, Pierre ; de Tullio, Pascal ; Challal, Sylvie ; Thomas, Jean-Yves ; Iop, Fabrice ; Louis, Caroline ; Botez-Pop, Iuliana ; Lestage, Pierre ; Danober, Laurence ; Kastrup, Jette S ; Pirotte, Bernard

Journal of medicinal chemistry, 2014-11, Vol.57 (22), p.9539-9553 [Periódico revisado por pares]

United States: American Chemical Society

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4
Development of Thiophenic Analogues of Benzothiadiazine Dioxides as New Powerful Potentiators of 2‑Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid (AMPA) Receptors
Development of Thiophenic Analogues of Benzothiadiazine Dioxides as New Powerful Potentiators of 2‑Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid (AMPA) Receptors
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Development of Thiophenic Analogues of Benzothiadiazine Dioxides as New Powerful Potentiators of 2‑Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid (AMPA) Receptors

Francotte, Pierre ; Goffin, Eric ; Fraikin, Pierre ; Graindorge, E ; Lestage, Pierre ; Danober, Laurence ; Challal, Sylvie ; Rogez, Nathalie ; Nosjean, Olivier ; Caignard, Daniel-Henri ; Pirotte, Bernard ; de Tullio, Pascal

Journal of medicinal chemistry, 2013-10, Vol.56 (20), p.7838-7850 [Periódico revisado por pares]

United States: American Chemical Society

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5
Cubanes in Medicinal Chemistry
Cubanes in Medicinal Chemistry
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Cubanes in Medicinal Chemistry

Reekie, Tristan A ; Williams, Craig M ; Rendina, Louis M ; Kassiou, Michael

Journal of medicinal chemistry, 2019-02, Vol.62 (3), p.1078-1095 [Periódico revisado por pares]

United States: American Chemical Society

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6
New Fluorinated 1,2,4-Benzothiadiazine 1,1-Dioxides: Discovery of an Orally Active Cognitive Enhancer Acting through Potentiation of the 2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors
New Fluorinated 1,2,4-Benzothiadiazine 1,1-Dioxides: Discovery of an Orally Active Cognitive Enhancer Acting through Potentiation of the 2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors
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New Fluorinated 1,2,4-Benzothiadiazine 1,1-Dioxides: Discovery of an Orally Active Cognitive Enhancer Acting through Potentiation of the 2-Amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic Acid Receptors

Francotte, Pierre ; Goffin, Eric ; Fraikin, Pierre ; Lestage, Pierre ; Van Heugen, Jean-Claude ; Gillotin, Florian ; Danober, Laurence ; Thomas, Jean-Yves ; Chiap, Patrice ; Caignard, Daniel-Henri ; Pirotte, Bernard ; de Tullio, Pascal

Journal of medicinal chemistry, 2010-02, Vol.53 (4), p.1700-1711 [Periódico revisado por pares]

Columbus, OH: American Chemical Society

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7
pkCSM: Predicting Small-Molecule Pharmacokinetic and Toxicity Properties Using Graph-Based Signatures
pkCSM: Predicting Small-Molecule Pharmacokinetic and Toxicity Properties Using Graph-Based Signatures
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pkCSM: Predicting Small-Molecule Pharmacokinetic and Toxicity Properties Using Graph-Based Signatures

Pires, Douglas E. V ; Blundell, Tom L ; Ascher, David B

Journal of medicinal chemistry, 2015-05, Vol.58 (9), p.4066-4072 [Periódico revisado por pares]

United States: American Chemical Society

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8
New Pyridobenzoxazepine Derivatives Derived from 5-(4-Methylpiperazin-1-yl)-8-chloro-pyrido[2,3-b][1,5]benzoxazepine (JL13): Chemical Synthesis and Pharmacological Evaluation
New Pyridobenzoxazepine Derivatives Derived from 5-(4-Methylpiperazin-1-yl)-8-chloro-pyrido[2,3-b][1,5]benzoxazepine (JL13): Chemical Synthesis and Pharmacological Evaluation
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New Pyridobenzoxazepine Derivatives Derived from 5-(4-Methylpiperazin-1-yl)-8-chloro-pyrido[2,3-b][1,5]benzoxazepine (JL13): Chemical Synthesis and Pharmacological Evaluation

Liégeois, Jean-François ; Deville, Marine ; Dilly, Sébastien ; Lamy, Cédric ; Mangin, Floriane ; Résimont, Mélissa ; Tarazi, Frank I

Journal of medicinal chemistry, 2012-02, Vol.55 (4), p.1572-1582 [Periódico revisado por pares]

United States: American Chemical Society

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9
Physicochemical Property Determinants of Oral Absorption for PROTAC Protein Degraders
Physicochemical Property Determinants of Oral Absorption for PROTAC Protein Degraders
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Physicochemical Property Determinants of Oral Absorption for PROTAC Protein Degraders

Hornberger, Keith R. ; Araujo, Erika M. V.

Journal of medicinal chemistry, 2023-06, Vol.66 (12), p.8281-8287 [Periódico revisado por pares]

United States: American Chemical Society

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10
Synthesis and Pharmacology of Mono‑, Di‑, and Trialkyl-Substituted 7‑Chloro-3,4-dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides Combined with X‑ray Structure Analysis to Understand the Unexpected Structure–Activity Relationship at AMPA Receptors
Synthesis and Pharmacology of Mono‑, Di‑, and Trialkyl-Substituted 7‑Chloro-3,4-dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides Combined with X‑ray Structure Analysis to Understand the Unexpected Structure–Activity Relationship at AMPA Receptors
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Synthesis and Pharmacology of Mono‑, Di‑, and Trialkyl-Substituted 7‑Chloro-3,4-dihydro‑2H‑1,2,4-benzothiadiazine 1,1-Dioxides Combined with X‑ray Structure Analysis to Understand the Unexpected Structure–Activity Relationship at AMPA Receptors

Larsen, Anja Probst ; Francotte, Pierre ; Frydenvang, Karla ; Tapken, Daniel ; Goffin, Eric ; Fraikin, Pierre ; Caignard, Daniel-Henri ; Lestage, Pierre ; Danober, Laurence ; Pirotte, Bernard ; Kastrup, Jette Sandholm

ACS chemical neuroscience, 2016-03, Vol.7 (3), p.378-390 [Periódico revisado por pares]

United States: American Chemical Society

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