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1 |
Material Type: Artigo
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Efficient synthesis of 5-(hydroxymethyl)piperazin-2-ones using automatically prepared chiral bromocarboxylic acid and Garner’s aldehyde as versatile building blocksMasui, Hisashi ; Naito, Kohei ; Minoshima, Mai ; Kusayanagi, Akira ; Yosugi, Sae ; Shoji, Mitsuru ; Takahashi, TakashiBioorganic & medicinal chemistry letters, 2021-05, Vol.40, p.127961-127961, Article 127961 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
2 |
Material Type: Artigo
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Synthesis, antituberculosis studies and biological evaluation of new quinoline derivatives carrying 1,2,4-oxadiazole moietyShruthi, T.G. ; Eswaran, Sumesh ; Shivarudraiah, Prasad ; Narayanan, Shridhar ; Subramanian, SangeethaBioorganic & medicinal chemistry letters, 2019-01, Vol.29 (1), p.97-102 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
3 |
Material Type: Artigo
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New natural products as new leads for antibacterial drug discoveryBrown, Dean G. ; Lister, Troy ; May-Dracka, Tricia L.Bioorganic & medicinal chemistry letters, 2014-01, Vol.24 (2), p.413-418 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
4 |
Material Type: Artigo
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Biocatalytic synthesis and evaluation of antioxidant and antibacterial activities of hydroxyequolsNozawa, Daiki ; Matsuyama, Akinobu ; Furuya, ToshikiBioorganic & medicinal chemistry letters, 2022-10, Vol.73, p.128908-128908, Article 128908 [Periódico revisado por pares]Elsevier LtdTexto completo disponível |
5 |
Material Type: Artigo
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Ultrasonication-ionic liquid synergy for the synthesis of new potent anti-tuberculosis 1,2,4-triazol-1-yl-pyrazole based spirooxindolopyrrolizidinesPogaku, Vinay ; Krishna, Vagolu Siva ; Sriram, Dharmarajan ; Rangan, Krishnan ; Basavoju, SrinivasBioorganic & medicinal chemistry letters, 2019-07, Vol.29 (13), p.1682-1687 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
6 |
Material Type: Artigo
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Design, synthesis and biological evaluation of potent EGFR kinase inhibitors against 19D/T790M/C797S mutationSu, Zhicheng ; Yang, Tingyuan ; Wang, Jie ; Lai, Mengzhen ; Tong, Linjiang ; Wumaier, Gulinuer ; Chen, Zhuo ; Li, Shengqing ; Li, Honglin ; Xie, Hua ; Zhao, ZhenjiangBioorganic & medicinal chemistry letters, 2020-08, Vol.30 (16), p.127327-127327, Article 127327 [Periódico revisado por pares]Elsevier LtdTexto completo disponível |
7 |
Material Type: Artigo
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Synthesis of mitochondria-targeted coumarin-3-carboxamide fluorescent derivatives: Inhibiting mitochondrial TrxR2 and cell proliferation on breast cancer cellsLi, Yuanyuan ; Tang, Qun ; Xie, Yu ; He, Dian ; Yang, Kun ; Zheng, LifangBioorganic & medicinal chemistry letters, 2021-02, Vol.33, p.127750-127750, Article 127750 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
8 |
Material Type: Artigo
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Discovery of benzo[d]oxazol-2(3H)-one derivatives as a new class of TNIK inhibitors for the treatment of colorectal cancerLuo, Xinling ; Yang, Ruicheng ; Li, Yueshan ; Zhang, Liting ; Yang, Shengyong ; Li, LinliBioorganic & medicinal chemistry letters, 2022-07, Vol.67, p.128745-128745, Article 128745 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
9 |
Material Type: Artigo
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Design, synthesis and activity evaluation of Hedgehog inhibitor Itraconazole derivatives in A549 cellsCai, Jin ; Chen, Xixi ; You, Haoyuan ; Li, Xiaojing ; Ji, MinBioorganic & medicinal chemistry letters, 2022-11, Vol.76, p.129011-129011, Article 129011 [Periódico revisado por pares]Texto completo disponível |
10 |
Material Type: Artigo
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Essential structure of orexin 1 receptor antagonist YNT-707: Conversion of the 16-cyclopropylmethyl group to the 16-sulfonamide group in d-nor-nalfurafine derivativesKatoh, Koki ; Kutsumura, Noriki ; Yamamoto, Naoshi ; Nagumo, Yasuyuki ; Saitoh, Tsuyoshi ; Ishikawa, Yukiko ; Irukayama-Tomobe, Yoko ; Tanimura, Ryuji ; Yanagisawa, Masashi ; Nagase, HiroshiBioorganic & medicinal chemistry letters, 2022-03, Vol.59, p.128550-128550, Article 128550 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |