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Material Type: Artigo
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5-Ene-4-thiazolidinones – An efficient tool in medicinal chemistryKaminskyy, Danylo ; Kryshchyshyn, Anna ; Lesyk, RomanEuropean journal of medicinal chemistry, 2017-11, Vol.140, p.542-594 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
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Material Type: Artigo
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Medicinal Chemistry Optimization of a Diaminopurine Chemotype: Toward a Lead for Trypanosoma brucei InhibitorsSingh, Baljinder ; Diaz-Gonzalez, Rosario ; Ceballos-Perez, Gloria ; Rojas-Barros, Domingo I ; Gunaganti, Naresh ; Gillingwater, Kirsten ; Martinez-Martinez, Maria Santos ; Manzano, Pilar ; Navarro, Miguel ; Pollastri, Michael PJournal of medicinal chemistry, 2020-09, Vol.63 (17), p.9912-9927 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Medicinal Chemistry Optimization of Antiplasmodial Imidazopyridazine Hits from High Throughput Screening of a SoftFocus Kinase Library: Part 2Le Manach, Claire ; Paquet, Tanya ; Gonzàlez Cabrera, Diego ; Younis, Yassir ; Taylor, Dale ; Wiesner, Lubbe ; Lawrence, Nina ; Schwager, Sylva ; Waterson, David ; Witty, Michael J ; Wittlin, Sergio ; Street, Leslie J ; Chibale, KellyJournal of medicinal chemistry, 2014-11, Vol.57 (21), p.8839-8848 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Medicinal Chemistry Optimization of Antiplasmodial Imidazopyridazine Hits from High Throughput Screening of a SoftFocus Kinase Library: Part 1Le Manach, Claire ; Gonzàlez Cabrera, Diego ; Douelle, Frederic ; Nchinda, Aloysius T ; Younis, Yassir ; Taylor, Dale ; Wiesner, Lubbe ; White, Karen L ; Ryan, Eileen ; March, Corinne ; Duffy, Sandra ; Avery, Vicky M ; Waterson, David ; Witty, Michael J ; Wittlin, Sergio ; Charman, Susan A ; Street, Leslie J ; Chibale, KellyJournal of medicinal chemistry, 2014-03, Vol.57 (6), p.2789-2798 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Medicinal Chemistry of Hsp90 InhibitorsDrysdale, Martin ; Brough, PaulCurrent topics in medicinal chemistry, 2008-07, Vol.8 (10), p.859-868 [Periódico revisado por pares]Bentham Science Publishers LtdTexto completo disponível |
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Material Type: Artigo
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Medicinal attributes of pyrazolo[3,4-d]pyrimidines: A reviewChauhan, Monika ; Kumar, RajBioorganic & medicinal chemistry, 2013-09, Vol.21 (18), p.5657-5668 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Bioactive Constituents of Glycyrrhiza uralensis (Licorice): Discovery of the Effective Components of a Traditional Herbal MedicineJi, Shuai ; Li, Ziwei ; Song, Wei ; Wang, Yongrui ; Liang, Wenfei ; Li, Kai ; Tang, Shunan ; Wang, Qi ; Qiao, Xue ; Zhou, Demin ; Yu, Siwang ; Ye, MinJournal of natural products (Washington, D.C.), 2016-02, Vol.79 (2), p.281-292 [Periódico revisado por pares]United States: American Chemical Society and American Society of PharmacognosyTexto completo disponível |
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Material Type: Artigo
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Functionalized quinoxalinones as privileged structures with broad-ranging pharmacological activitiesJiang, Xiaoying ; Wu, Kaiyu ; Bai, Renren ; Zhang, Pengfei ; Zhang, YiEuropean journal of medicinal chemistry, 2022-02, Vol.229, p.114085-114085, Article 114085 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
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Material Type: Artigo
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Discovery of a Potent Dual Inhibitor of Acetylcholinesterase and Butyrylcholinesterase with Antioxidant Activity that Alleviates Alzheimer-like Pathology in Old APP/PS1 MiceViayna, Elisabet ; Coquelle, Nicolas ; Cieslikiewicz-Bouet, Monika ; Cisternas, Pedro ; Oliva, Carolina A ; Sánchez-López, Elena ; Ettcheto, Miren ; Bartolini, Manuela ; De Simone, Angela ; Ricchini, Mattia ; Rendina, Marisa ; Pons, Mégane ; Firuzi, Omidreza ; Pérez, Belén ; Saso, Luciano ; Andrisano, Vincenza ; Nachon, Florian ; Brazzolotto, Xavier ; García, Maria Luisa ; Camins, Antoni ; Silman, Israel ; Jean, Ludovic ; Inestrosa, Nibaldo C ; Colletier, Jacques-Philippe ; Renard, Pierre-Yves ; Muñoz-Torrero, DiegoJournal of medicinal chemistry, 2021-01, Vol.64 (1), p.812-839 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Galectin-3-Binding Glycomimetics that Strongly Reduce Bleomycin-Induced Lung Fibrosis and Modulate Intracellular Glycan RecognitionDelaine, Tamara ; Collins, Patrick ; MacKinnon, Alison ; Sharma, G. ; Stegmayr, John ; Rajput, Vishal K. ; Mandal, Santanu ; Cumpstey, Ian ; Larumbe, Amaia ; Salameh, Bader A. ; Kahl-Knutsson, Barbro ; van Hattum, Hilde ; van Scherpenzeel, Monique ; Pieters, Roland J. ; Sethi, Tariq ; Schambye, Hans ; Oredsson, Stina ; Leffler, Hakon ; Blanchard, Helen ; Nilsson, Ulf J.Chembiochem : a European journal of chemical biology, 2016-09, Vol.17 (18), p.1759-1770 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |