Structural biology and medicinalchemistry strategies to the discovery of new bioactive compounds applications in infectious diseases
G. M. A Lima A. A Oliveira; R. V Bueno; F. V Maluf; A. C. C Aguiar; L. R Sousa; Glaucius Oliva; Rafael Victorio Carvalho Guido; TWA's General Conference (3. 2015 Vienna); TWA's General Meeting (26. 2015 Vienna)
Abstracts Trieste: The World Academy of Sciences - TWAS, 2015
Trieste The World Academy of Sciences - TWAS 2015
Localização:
IFSC - Inst. Física de São Carlos
(PROD024436 )(Acessar)
Synthesis, molecular modeling and preliminary biological evaluation of a set of 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazole as potential antibacterial, anti-Trypanosoma cruzi and antifungal agents
Marina Ishii Salomão Dória Jorge; Alex Alfredo de Oliveira; Fanny Palace-Berl; Ieda Yuriko Sonehara; Kerly Fernanda Mesquita Pasqualoto; Leoberto Costa Tavares
Bioorganic & Medicinal Chemistry Oxford v. 19, n. 21, p. 6292-6301, 2011
Oxford 2011
Item não circula. Consulte sua biblioteca.(Acessar)
Discovery of 1,2,4-oxadiazole derivatives as a novel class of noncompetitive inhibitors of 3-hydroxykynurenine transaminase (HKT) from Aedes aegypti
Larissa G. Maciel Andrew Albert de Oliveira; Tatiany P Romão; Laylla L. L Leal; Rafael Victorio Carvalho Guido; Maria Helena N. L Silva Filha; Janaína V Anjos; Thereza A Soares
Bioorganic and Medicinal Chemistry Oxford : Elsevier v. 28, n. 2, p. 115252-1-115252-13, Jan. 2020
Oxford 2020
Localização:
IFSC - Inst. Física de São Carlos
(PROD029805 )(Acessar)
Structure-activity relationships of sulfonamides derived from carvacrol and their potential for the treatment of Alzheimer's disease
Márcia Maria de Souza Marina Corrêa Andreolla; Thaís Cecília Ribeiro; Ana Elisa Gonçalves; Alex Rogério Medeiros; Anacleto Silva de Souza; Leonardo Luiz Gomes Ferreira; Adriano Defini Andricopulo; Rosendo Augusto Yunes; Aldo Sena de Oliveira
RSC Medicinal Chemistry Cambridge : Royal Society of Chemistry - RSC v. 11, n. 2, p. 307-316, Feb. 2020
Cambridge 2020
Localização:
IFSC - Inst. Física de São Carlos
(PROD030145 )(Acessar)
Diaminomaleonitrile derivatives as new potential antichagasic compounds a study of structure-activity relationships
Aldo S. Oliveira Lucas dos S Mello; Camila H Ogihara; Thiago H Döring; David Leandro Palomino-Salcedo; Simone Michelan Duarte; Leonardo Luiz Gomes Ferreira; Julia Medeiros Souza; María-José Dávila-Rodríguez; José W. da Cruz Júnior; Edward R Dockal; Adriano Defini Andricopulo
Future Medicinal Chemistry London v. 13, n. 24, p. 2167-2183, Dec. 2021
London 2021
Localização:
IFSC - Inst. Física de São Carlos
(PROD032333-SC )(Acessar)
Novel trypanocidal thiophen-chalcone cruzain inhibitors structure- and ligand-based studies
Aldo Sena de Oliveira Marilia Valli; Leonardo Luiz Gomes Ferreira; Julia Medeiros Souza; Renata Krogh Andricopulo; Lidiane Meier; Heitor R Abreu; Bruna G Voltolini; Luana C Llanes; Ricardo José Nunes; Antonio L Braga; Adriano Defini Andricopulo
Future Medicinal Chemistry London v. 14, n. 11, p. 795-808, June 2022
London 2022
Localização:
IFSC - Inst. Física de São Carlos
(PROD033126-SC )(Acessar)
Pyrazolines as potential anti-Alzheimer's agents DFT, molecular docking, enzyme inhibition and pharmacokinetic studies
Valkiria Machado Arthur R Cenci; Kerolain F Teixeira; Larissa Sens; Tiago Tizziani; Ricardo J Nunes; Leonardo Luiz Gomes Ferreira; Rosendo A Yunes; Louis P Sandjo; Adriano Defini Andricopulo; Aldo S Oliveira
RSC Medicinal Chemistry Cambridge v. 13, n. 12, p. 1644-1656 + supplementary information, Dec. 2022
Cambridge 2022
Localização:
IFSC - Inst. Física de São Carlos
(PROD033792-SC )(Acessar)
DYRK1A inhibitors and perspectives for the treatment of Alzheimer's disease
Márcia Maria de Souza Arthur Ribeiro Cenci; Kerolain Faoro Teixeira; Valkiria Machado; Majory Christina Garcia Mendes; Ana Elisa Gonçalves; Ana Paula Dalmagro; Camila André Cazarin; Leonardo Luiz Gomes Ferreira; Aldo Sena de Oliveira; Adriano Defini Andricopulo
Current Medicinal Chemistry Sharjah v. 30, n. 6, p. 669-688, 2023
Sharjah 2023
Localização:
IFSC - Inst. Física de São Carlos
(PROD033747 )(Acessar)
Synthesis, molecular modeling and preliminary biological evaluation of a set of 3-acetyl-2,5-disubstituted-2,3-dihydro-1,3,4-oxadiazole as potential antibacterial, anti-Trypanosoma cruzi and antifungal agents
Marina Ishii Salomão Dória Jorge; Alex Alfredo de Oliveira; Fanny Palace-Berl; Ieda Yuriko Sonehara; Kerly Fernanda Mesquita Pasqualoto; Leoberto Costa Tavares
Bioorganic & Medicinal Chemistry Oxford v. 19, n. 21, p. 6292-6301, 2011
Oxford 2011
Item não circula. Consulte sua biblioteca.(Acessar)