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1 |
Material Type: Artigo
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Synthesis and biological evaluation of novel mono- and bivalent ASGP-R-targeted drug-conjugatesPetrov, Rostislav A. ; Maklakova, Svetlana Yu ; Ivanenkov, Yan A. ; Petrov, Stanislav A. ; Sergeeva, Olga V. ; Yamansarov, Emil Yu ; Saltykova, Irina V. ; Kireev, Igor I. ; Alieva, Irina B. ; Deyneka, Ekaterina V. ; Sofronova, Alina A. ; Aladinskaia, Anastasiia V. ; Trofimenko, Alexandre V. ; Yamidanov, Renat S. ; Kovalev, Sergey V. ; Kotelianski, Victor E. ; Zatsepin, Timofey S. ; Beloglazkina, Elena K. ; Majouga, Alexander G.Bioorganic & medicinal chemistry letters, 2018-02, Vol.28 (3), p.382-387 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and biological evaluation of novel doxorubicin-containing ASGP-R-targeted drug-conjugatesIvanenkov, Yan A. ; Majouga, Alexander G. ; Petrov, Rostislav A. ; Petrov, Stanislav A. ; Kovalev, Sergey V. ; Maklakova, Svetlana Yu ; Yamansarov, Emil Yu ; Saltykova, Irina V. ; Deyneka, Ekaterina V. ; Filkov, Gleb I. ; Kotelianski, Victor E. ; Zatsepin, Timofey S. ; Beloglazkina, Elena K.Bioorganic & medicinal chemistry letters, 2018-02, Vol.28 (3), p.503-508 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and initial in vitro evaluation of PSMA-targeting ligands with a modified aromatic moiety at the lysine ε-nitrogen atomZyk, Nikolai Y. ; Ber, Anton P. ; Nimenko, Ekaterina A. ; Shafikov, Radik R. ; Evteev, Sergei A. ; Petrov, Stanislav A. ; Uspenskaya, Anastasia A. ; Dashkova, Natalia S. ; Ivanenkov, Yan A. ; Skvortsov, Dmitry A. ; Beloglazkina, Elena K. ; Majouga, Alexander G. ; Machulkin, Aleksei E.Bioorganic & medicinal chemistry letters, 2022-09, Vol.71, p.128840-128840, Article 128840 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Novel potent pyridoxine-based inhibitors of AChE and BChE, structural analogs of pyridostigmine, with improved in vivo safety profileStrelnik, Alexey D. ; Petukhov, Alexey S. ; Zueva, Irina V. ; Zobov, Vladimir V. ; Petrov, Konstantin A. ; Nikolsky, Evgeny E. ; Balakin, Konstantin V. ; Bachurin, Sergey O. ; Shtyrlin, Yurii G.Bioorganic & medicinal chemistry letters, 2016-08, Vol.26 (16), p.4092-4094 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis, SAR and molecular docking study of novel non-β-lactam inhibitors of TEM type β-lactamaseAntipin, Roman L. ; Beshnova, Daria A. ; Petrov, Rostislav A. ; Shiryaeva, Anna S. ; Andreeva, Irina P. ; Grigorenko, Vitaly G. ; Rubtsova, Maya Yu ; Majouga, Alexander G. ; Lamzin, Victor S. ; Egorov, Alexey M.Bioorganic & medicinal chemistry letters, 2017-04, Vol.27 (7), p.1588-1592 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Fluoropyrrolidine amides as dipeptidyl peptidase IV inhibitorsCALDWELL, Charles G ; PING CHEN ; HUAIBING HE ; LYONS, Kathryn A ; THORNBERRY, Nancy A ; WEBER, Ann E ; JIAFANG HE ; PARMEE, Emma R ; LEITING, Barbara ; MARSILIO, Frank ; PATEL, Reshma A ; WU, Joseph K ; EIERMANN, George J ; PETROV, AleksandrBioorganic & medicinal chemistry letters, 2004-03, Vol.14 (5), p.1265-1268 [Periódico revisado por pares]Oxford: ElsevierTexto completo disponível |
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Material Type: Artigo
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Discovery of potent and selective orally bioavailable β-substituted phenylalanine derived dipeptidyl peptidase IV inhibitorsEdmondson, Scott D. ; Mastracchio, Anthony ; Duffy, Joseph L. ; Eiermann, George J. ; He, Huaibing ; Ita, Ida ; Leiting, Barbara ; Leone, Joseph F. ; Lyons, Kathryn A. ; Makarewicz, Amanda M. ; Patel, Reshma A. ; Petrov, Aleksandr ; Wu, Joseph K. ; Thornberry, Nancy A. ; Weber, Ann E.Bioorganic & medicinal chemistry letters, 2005-06, Vol.15 (12), p.3048-3052 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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4-Amino cyclohexylglycine analogues as potent dipeptidyl peptidase IV inhibitorsParmee, Emma R. ; He, Jiafang ; Mastracchio, Anthony ; Edmondson, Scott D. ; Colwell, Larry ; Eiermann, George ; Feeney, William P. ; Habulihaz, Bahanu ; He, Huaibing ; Kilburn, Ruth ; Leiting, Barbara ; Lyons, Kathryn ; Marsilio, Frank ; Patel, Reshma A. ; Petrov, Aleksandr ; Di Salvo, Jerry ; Wu, Joseph K. ; Thornberry, Nancy A. ; Weber, Ann E.Bioorganic & medicinal chemistry letters, 2004-01, Vol.14 (1), p.43-46 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Discovery of potent, selective, and orally bioavailable pyridone-based dipeptidyl peptidase-4 inhibitorsXu, Jinyou ; Wei, Lan ; Mathvink, Robert ; Edmondson, Scott D. ; Mastracchio, Anthony ; Eiermann, George J. ; He, Huaibing ; Leone, Joseph F. ; Leiting, Barbara ; Lyons, Kathryn A. ; Marsilio, Frank ; Patel, Reshma A. ; Petrov, Aleksandr ; Wu, Joseph K. ; Thornberry, Nancy A. ; Weber, Ann E.Bioorganic & medicinal chemistry letters, 2006-03, Vol.16 (5), p.1346-1349 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Incorporation of a pyrene nucleoside analogue into synthetic oligodeoxynucleotides using a nucleoside-like synthonProkhorenko, Igor A. ; Korshun, Vladimir A. ; Petrov, Andrei A. ; Gontarev, Sergei V. ; Berlin, Yuri A.Bioorganic & medicinal chemistry letters, 1995-09, Vol.5 (18), p.2081-2084 [Periódico revisado por pares]Elsevier LtdTexto completo disponível |