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Material Type: Artigo
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Benzo[f]azino[2,1-a]phthalazinium Cations: Novel DNA Intercalating Chromophores with Antiproliferative ActivityMartínez, Valentín ; Burgos, Carolina ; Alvarez-Builla, Julio ; Fernández, Gerónimo ; Domingo, Alberto ; García-Nieto, Raquel ; Gago, Federico ; Manzanares, Ignacio ; Cuevas, Carmen ; Vaquero, Juan JJournal of medicinal chemistry, 2004-02, Vol.47 (5), p.1136-1148 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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DNA Sequence-Specific Reading by Echinomycin: Role of Hydrogen Bonding and Stacking InteractionsGallego, Jose ; Luque, F. J ; Orozco, Modesto ; Burgos, Carolina ; Alvarez-Builla, Julio ; Rodrigo, M. Melia ; Gago, FedericoJournal of medicinal chemistry, 1994-05, Vol.37 (11), p.1602-1609 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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β-C-Mannosides as Selectin InhibitorsKaila, Neelu ; Chen, Lihren ; Thomas ; Tsao, Desiree ; Tam, Steve ; Bedard, Patricia W ; Camphausen, Raymond T ; Alvarez, Juan C ; Ullas, GiliyarJournal of medicinal chemistry, 2002-04, Vol.45 (8), p.1563-1566 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Synthesis, Structure, and Pharmacological Evaluation of the Stereoisomers of FurnidipineAlajarin, Ramon ; Vaquero, Juan J ; Alvarez-Builla, Julio ; Pastor, Manuel ; Sunkel, Carlos ; Fau de Casa-Juana, Miguel ; Priego, Jaime ; Statkow, Peter R ; Sanz-Aparicio, Julia ; Fonseca, IsabelJournal of medicinal chemistry, 1995-07, Vol.38 (15), p.2830-2841 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Discovery of a Potent and Orally Active Hedgehog Pathway Antagonist (IPI-926)Tremblay, Martin R ; Lescarbeau, André ; Grogan, Michael J ; Tan, Eddy ; Lin, Grace ; Austad, Brian C ; Yu, Lin-Chen ; Behnke, Mark L ; Nair, Somarajan J ; Hagel, Margit ; White, Kerry ; Conley, James ; Manna, Joseph D ; Alvarez-Diez, Teresa M ; Hoyt, Jennifer ; Woodward, Caroline N ; Sydor, Jens R ; Pink, Melissa ; MacDougall, John ; Campbell, Matthew J ; Cushing, Jill ; Ferguson, Jeanne ; Curtis, Michael S ; McGovern, Karen ; Read, Margaret A ; Palombella, Vito J ; Adams, Julian ; Castro, Alfredo CJournal of medicinal chemistry, 2009-07, Vol.52 (14), p.4400-4418 [Periódico revisado por pares]Columbus, OH: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Cheminformatic Models To Predict Binding Affinities to Human Serum AlbuminColmenarejo, Gonzalo ; Alvarez-Pedraglio, Ana ; Lavandera, José-LuisJournal of medicinal chemistry, 2001-12, Vol.44 (25), p.4370-4378 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Nanomolar Inhibitors of the Peptidyl Prolyl Cis/Trans Isomerase Pin1 from Combinatorial Peptide LibrariesWildemann, Dirk ; Erdmann, Frank ; Alvarez, Birte Hernandez ; Stoller, Gerlind ; Zhou, Xiao Z ; Fanghänel, Jörg ; Schutkowski, Mike ; Lu, Kun P ; Fischer, GunterJournal of medicinal chemistry, 2006-04, Vol.49 (7), p.2147-2150 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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1,2,3-Triazole-[2,5-Bis-O-(tert-butyldimethylsilyl)-.beta.-D-ribofuranosyl]-3'-spiro-5''-(4''-amino-1'',2''-oxathiole 2'',2''-dioxide) (TSAO) Analogs: Synthesis and Anti-HIV-1 ActivityAlvarez, Rosa ; Velazquez, Sonsoles ; San-Felix, Ana ; Aquaro, Stefano ; Clercq, Erik De ; Perno, Carlo-Federico ; Karlsson, Anna ; Balzarini, Jan ; Camarasa, Maria JoseJournal of medicinal chemistry, 1994-11, Vol.37 (24), p.4185-4194 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Tricyclic Farnesyl Protein Transferase Inhibitors: Crystallographic and Calorimetric Studies of Structure−Activity RelationshipsStrickland, Corey L ; Weber, Patricia C ; Windsor, William T ; Wu, Zhen ; Le, Hung V ; Albanese, Margaret M ; Alvarez, Carmen S ; Cesarz, David ; del Rosario, Joycelyn ; Deskus, Jeffrey ; Mallams, Alan K ; Njoroge, F. George ; Piwinski, John J ; Remiszewski, Stacy ; Rossman, Randall R ; Taveras, Arthur G ; Vibulbhan, Bancha ; Doll, Ronald J ; Girijavallabhan, Viyyoor M ; Ganguly, Ashit KJournal of medicinal chemistry, 1999-06, Vol.42 (12), p.2125-2135 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Synthesis, in Vitro Antiviral Evaluation, and Stability Studies of Novel α-Borano-Nucleotide Analogues of 9-[2-(Phosphonomethoxy)ethyl]adenine and (R)-9-[2-(Phosphonomethoxy)propyl]adenineBarral, Karine ; Priet, Stéphane ; Sire, Joséphine ; Neyts, Johan ; Balzarini, Jan ; Canard, Bruno ; Alvarez, KarineJournal of medicinal chemistry, 2006-12, Vol.49 (26), p.7799-7806 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |