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1 |
Material Type: Artigo
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Tacripyrimidines, the first tacrine-dihydropyrimidine hybrids, as multi-target-directed ligands for Alzheimer's diseaseChioua, Mourad ; Buzzi, Eleonora ; Moraleda, Ignacio ; Iriepa, Isabel ; Maj, Maciej ; Wnorowski, Artur ; Giovannini, Catia ; Tramarin, Anna ; Portali, Federica ; Ismaili, Lhassane ; López-Alvarado, Pilar ; Bolognesi, Maria Laura ; Jóźwiak, Krzysztof ; Menéndez, J. Carlos ; Marco-Contelles, José ; Bartolini, ManuelaEuropean journal of medicinal chemistry, 2018-07, Vol.155, p.839-846 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
2 |
Material Type: Artigo
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Developing steroidal aromatase inhibitors-an effective armament to win the battle against breast cancerYadav, Mange Ram ; Barmade, Mahesh A. ; Tamboli, Riyaj S. ; Murumkar, Prashant R.European journal of medicinal chemistry, 2015-11, Vol.105, p.1-38 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
3 |
Material Type: Artigo
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Tetrahydropyranodiquinolin-8-amines as new, non hepatotoxic, antioxidant, and acetylcholinesterase inhibitors for Alzheimer's disease therapyDgachi, Youssef ; Sokolov, Olga ; Luzet, Vincent ; Godyń, Justyna ; Panek, Dawid ; Bonet, Alexandre ; Martin, Hélène ; Iriepa, Isabel ; Moraleda, Ignacio ; García-Iriepa, Cristina ; Janockova, Jana ; Richert, Lysiane ; Soukup, Ondrej ; Malawska, Barbara ; Chabchoub, Fakher ; Marco-Contelles, José ; Ismaili, LhassaneEuropean journal of medicinal chemistry, 2017-01, Vol.126, p.576-589 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
4 |
Material Type: Artigo
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Synthesis and biological evaluation of new 3-(6-hydroxyindol-2-yl)-5-(Phenyl) pyridine or pyrazine V-Shaped molecules as kinase inhibitors and cytotoxic agentsKassis, Pamela ; Brzeszcz, Joanna ; Bénéteau, Valérie ; Lozach, Olivier ; Meijer, Laurent ; Le Guével, Rémi ; Guillouzo, Christiane ; Lewiński, Krzysztof ; Bourg, Stéphane ; Colliandre, Lionel ; Routier, Sylvain ; Mérour, Jean-YvesEuropean journal of medicinal chemistry, 2011-11, Vol.46 (11), p.5416-5434 [Periódico revisado por pares]Kidlington: Elsevier Masson SASTexto completo disponível |
5 |
Material Type: Artigo
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Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moietiesSpadoni, Gilberto ; Bedini, Annalida ; Bartolucci, Silvia ; Pala, Daniele ; Mor, Marco ; Riccioni, Teresa ; Borsini, Franco ; Cabri, Walter ; Celona, Diana ; Marzi, Mauro ; Tarzia, Giorgio ; Rivara, Silvia ; Minetti, PatriziaEuropean journal of medicinal chemistry, 2014-06, Vol.80, p.8-35 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
6 |
Material Type: Artigo
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Novel 9-oxo-thiazolo[5,4- f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studiesLogé, Cédric ; Testard, Alexandra ; Thiéry, Valérie ; Lozach, Olivier ; Blairvacq, Mélina ; Robert, Jean-Michel ; Meijer, Laurent ; Besson, ThierryEuropean journal of medicinal chemistry, 2008-07, Vol.43 (7), p.1469-1477 [Periódico revisado por pares]Oxford: Elsevier Masson SASTexto completo disponível |
7 |
Material Type: Artigo
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Type IIA - Type IIB protein tyrosine kinase inhibitors hybridization as an efficient approach for potent multikinase inhibitor development: Design, synthesis, anti-proliferative activity, multikinase inhibitory activity and molecular modeling of novel indolinone-based ureides and amidesEldehna, Wagdy M. ; El Kerdawy, Ahmed M. ; Al-Ansary, Ghada H. ; Al-Rashood, Sara T. ; Ali, Mamdouh M. ; Mahmoud, Abeer E.European journal of medicinal chemistry, 2019-02, Vol.163, p.37-53 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
8 |
Material Type: Artigo
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Synthesis, cytotoxicity, antioxidant activity and molecular modeling of new NSAIDs-EBS derivativesZhong, Min ; Lu, Ying ; Li, Shaolei ; Li, Xiaolong ; Liu, Zhenming ; He, Xianran ; Zhang, YongminEuropean journal of medicinal chemistry, 2023-11, Vol.259, p.115662-115662, Article 115662 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
9 |
Material Type: Artigo
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2,4-Disubstituted quinazolines as amyloid-β aggregation inhibitors with dual cholinesterase inhibition and antioxidant properties: Development and structure-activity relationship (SAR) studiesMohamed, Tarek ; Rao, Praveen P.N.European journal of medicinal chemistry, 2017-01, Vol.126, p.823-843 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |
10 |
Material Type: Artigo
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Recent advances in small organic molecules as DNA intercalating agents: Synthesis, activity, and modelingRescifina, Antonio ; Zagni, Chiara ; Varrica, Maria Giulia ; Pistarà, Venerando ; Corsaro, AntoninoEuropean journal of medicinal chemistry, 2014-03, Vol.74, p.95-115 [Periódico revisado por pares]France: Elsevier Masson SASTexto completo disponível |