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Material Type: Artigo
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Evaluation of a human bio-engineered skin equivalent for drug permeation studiesASBILL, Charles ; NANHYE KIM ; EL-KATTAN, Ayman ; CREEK, Kim ; WERTZ, Philip ; MICHNIAK, BozenaPharmaceutical research, 2000-09, Vol.17 (9), p.1092-1097 [Periódico revisado por pares]New York, NY: SpringerTexto completo disponível |
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Material Type: Artigo
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Evaluation of derivatives of 3-(2-oxo-1-pyrrolidine) hexahydro-1H-azepine-2-one as dermal penetration enhancers : side chain length variation and molecular modelingKIM, N ; EL-KATTAN, A. F ; ASBILL, C. S ; KENNETTE, R. J ; SOWELL, J. W ; LATOUR, R ; MICHNIAK, B. BJournal of controlled release, 2001-06, Vol.73 (2-3), p.183-196 [Periódico revisado por pares]Amsterdam: ElsevierTexto completo disponível |
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Material Type: Artigo
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Carboxylate bioisosteres of gabapentinBurgos-Lepley, Carmen E. ; Thompson, Lisa R. ; Kneen, Clare O. ; Osborne, Simon A. ; Bryans, Justin S. ; Capiris, Thomas ; Suman-Chauhan, Nirmala ; Dooley, David J. ; Donovan, Cindy M. ; Field, Mark J. ; Vartanian, Mark G. ; Kinsora, Jack J. ; Lotarski, Susan M. ; El-Kattan, Ayman ; Walters, Karen ; Cherukury, Madhu ; Taylor, Charles P. ; Wustrow, David J. ; Schwarz, Jacob B.Bioorganic & medicinal chemistry letters, 2006-05, Vol.16 (9), p.2333-2336 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Carboxylate bioisosteres of pregabalinSchwarz, Jacob B. ; Colbry, Norman L. ; Zhu, Zhijian ; Nichelson, Brian ; Barta, Nancy S. ; Lin, Kristin ; Hudack, Raymond A. ; Gibbons, Sian E. ; Galatsis, Paul ; DeOrazio, Russell J. ; Manning, David D. ; Vartanian, Mark G. ; Kinsora, Jack J. ; Lotarski, Susan M. ; Li, Zheng ; Dickerson, Melvin R. ; El-Kattan, Ayman ; Thorpe, Andrew J. ; Donevan, Sean D. ; Taylor, Charles P. ; Wustrow, David J.Bioorganic & medicinal chemistry letters, 2006-07, Vol.16 (13), p.3559-3563 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |