Discovery and preclinical pharmacology of INE963, a potent and fast-acting blood-stage antimalarial with a high barrier to resistance and potential for single-dose cures in uncomplicated malaria
Benjamin R. Taft Anna Caroline Campos Aguiar
Journal of Medicinal Chemistry Washington, DC v. 65, n. 5, p. 3798-3813, Mar. 2022
Washington, DC 2022
Localização:
IFSC - Inst. Física de São Carlos
(PROD032852 )(Acessar)
Mode of peroxisome proliferator-activated receptor 'gama' activation by luteolin
Ana C. Puhl Amanda Bernardes; Rodrigo L Silveira; Jing Yuan; Jéssica L. O Campos; Daniel Menezes Saidemberg; Mario S Palma; Aleksandra Cvoro; Stephen D Ayers; Paul Webb; Peter S Reinach; Munir S Skaf; Igor Polikarpov
Molecular Pharmacology Bethesda : American Society for Pharmacology and Experimental Therapeutics - ASPET v. 81, n. 6, p. 788-799, June 2012
Bethesda 2012
Localização:
IFSC - Inst. Física de São Carlos
(PROD019556 )(Acessar)
Mode of peroxisome proliferator-activated receptor 'gama' activation by luteolin
Ana C. Puhl Amanda Bernardes; Rodrigo L Silveira; Jing Yuan; Jéssica L. O Campos; Daniel Menezes Saidemberg; Mario S Palma; Aleksandra Cvoro; Stephen D Ayers; Paul Webb; Peter S Reinach; Munir S Skaf; Igor Polikarpov
Molecular Pharmacology Bethesda : American Society for Pharmacology and Experimental Therapeutics - ASPET v. 81, n. 6, p. 788-799, June 2012
Bethesda 2012
Localização:
IFSC - Inst. Física de São Carlos
(PROD019556 )(Acessar)
On the mechanisms of phenothiazine-induced mitochondrial permeability transition thiol oxidation, strict 'Ca POT.2+' dependence, and cyt c release
Thiago S. Cruz Priscila A Faria; Débora P Santana; Juliana C Ferreira; Vitor Oliveira; Otaciro Rangel Nascimento; Giselle Cerchiaro; Carlos Curti; Iseli L Nantes; Tiago Rodrigues
Biochemical Pharmacology Philadelphia : Elsevier v. 80, n. 8, p. 1284-1295, 2010
Philadelphia 2010
Localização:
FCFRP - Fac. Ciên. Farm. Ribeirão Preto
(pcd 2125319 Estantes Deslizantes ) e outros locais(Acessar)
On the mechanisms of phenothiazine-induced mitochondrial permeability transition thiol oxidation, strict 'Ca POT.2+' dependence, and cyt c release
Thiago S. Cruz Priscila A Faria; Débora P Santana; Juliana C Ferreira; Vitor Oliveira; Otaciro Rangel Nascimento; Giselle Cerchiaro; Carlos Curti; Iseli L Nantes; Tiago Rodrigues
Biochemical Pharmacology Philadelphia : Elsevier v. 80, n. 8, p. 1284-1295, 2010
Philadelphia 2010
Localização:
FCFRP - Fac. Ciên. Farm. Ribeirão Preto
(pcd 2125319 Estantes Deslizantes ) e outros locais(Acessar)
Synthetic cyclopenta[b]indoles exhibit antineoplastic activity by targeting microtubule dynamics in acute myeloid leukemia cells
Hugo Passos Vicari Keli Lima; Ralph da Costa Gomes; Daniara Cristina Fernandes; Jean Carlos Lipreri da Silva; Manoel Trindade Rodrigues Junior; Aline Silva Barroso de Oliveira; Ricardo Nascimento dos Santos; Adriano Defini Andricopulo; Fernando Coelho; Leticia Veras Costa Lotufo; João Agostinho Machado Neto
European Journal of Pharmacology Amsterdam v. 894, p. 173853-1-173853-10, Mar. 2021
Amsterdam 2021
Localização:
IFSC - Inst. Física de São Carlos
(PROD030951 )(Acessar)
Antioxidant activity, molecular docking, quantum studies and in vivo antinociceptive activity of sulfonamides derived from carvacrol
Aldo Sena de Oliveira Luana C Llanes; Ricardo J Nunes; Catharina Nucci-Martins; Anacleto Silva de Souza; David Leandro Palomino-Salcedo; María-José Dávila-Rodríguez; Leonardo Luiz Gomes Ferreira; Adair R. S Santos; Adriano Defini Andricopulo
Frontiers in Pharmacology Lausanne v. 12, p. 788850-1-788850-16 + supplementary material, Nov. 2021
Lausanne 2021
Localização:
IFSC - Inst. Física de São Carlos
(PROD032526 )(Acessar)