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11
A nontoxic pain killer designed by modeling of pathological receptor conformations
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Artigo
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A nontoxic pain killer designed by modeling of pathological receptor conformations

Spahn, V. ; Del Vecchio, G. ; Labuz, D. ; Rodriguez-Gaztelumendi, A. ; Massaly, N. ; Temp, J. ; Durmaz, V. ; Sabri, P. ; Reidelbach, M. ; Machelska, H. ; Weber, M. ; Stein, C.

Science (American Association for the Advancement of Science), 2017-03, Vol.355 (6328), p.966-969 [Periódico revisado por pares]

United States: American Association for the Advancement of Science

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12
Biochemical Pharmacology of the Sigma-1 Receptor
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Artigo
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Biochemical Pharmacology of the Sigma-1 Receptor

Chu, Uyen B ; Ruoho, Arnold E

Molecular pharmacology, 2016-01, Vol.89 (1), p.142-153 [Periódico revisado por pares]

United States

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13
A bifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates
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Artigo
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A bifunctional nociceptin and mu opioid receptor agonist is analgesic without opioid side effects in nonhuman primates

Ding, Huiping ; Kiguchi, Norikazu ; Yasuda, Dennis ; Daga, Pankaj R ; Polgar, Willma E ; Lu, James J ; Czoty, Paul W ; Kishioka, Shiroh ; Zaveri, Nurulain T ; Ko, Mei-Chuan

Science translational medicine, 2018-08, Vol.10 (456) [Periódico revisado por pares]

United States: The American Association for the Advancement of Science

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14
Biased Opioid Ligands
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Artigo
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Biased Opioid Ligands

Faouzi, Abdelfattah ; Varga, Balazs R ; Majumdar, Susruta

Molecules (Basel, Switzerland), 2020-09, Vol.25 (18), p.4257 [Periódico revisado por pares]

Switzerland: MDPI

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15
Time-Series Analysis of Fentanyl Concentration in the Unregulated Opioid Drug Supply in a Canadian Setting
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Time-Series Analysis of Fentanyl Concentration in the Unregulated Opioid Drug Supply in a Canadian Setting

Tobias, Samuel ; Grant, Cameron J ; Laing, Richard ; Arredondo, Jaime ; Lysyshyn, Mark ; Buxton, Jane ; Tupper, Kenneth W ; Wood, Evan ; Ti, Lianping

American journal of epidemiology, 2022-01, Vol.191 (2), p.241-247 [Periódico revisado por pares]

United States: Oxford University Press

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16
Design, Synthesis, and Biological Evaluation of NAP Isosteres: A Switch from Peripheral to Central Nervous System Acting Mu-Opioid Receptor Antagonists
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Artigo
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Design, Synthesis, and Biological Evaluation of NAP Isosteres: A Switch from Peripheral to Central Nervous System Acting Mu-Opioid Receptor Antagonists

Pagare, Piyusha P ; Li, Mengchu ; Zheng, Yi ; Kulkarni, Abhishek S ; Obeng, Samuel ; Huang, Boshi ; Ruiz, Christian ; Gillespie, James C ; Mendez, Rolando E ; Stevens, David L ; Poklis, Justin L ; Halquist, Matthew S ; Dewey, William L ; Selley, Dana E ; Zhang, Yan

Journal of medicinal chemistry, 2022-03, Vol.65 (6), p.5095-5112 [Periódico revisado por pares]

United States: American Chemical Society

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17
Molecular insights into the biased signaling mechanism of the μ-opioid receptor
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Molecular insights into the biased signaling mechanism of the μ-opioid receptor

Cong, Xiaojing ; Maurel, Damien ; Déméné, Hélène ; Vasiliauskaité-Brooks, Ieva ; Hagelberger, Joanna ; Peysson, Fanny ; Saint-Paul, Julie ; Golebiowski, Jérôme ; Granier, Sébastien ; Sounier, Rémy

Molecular cell, 2021-10, Vol.81 (20), p.4165-4175.e6 [Periódico revisado por pares]

United States: Elsevier Inc

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18
PLA-PCL Microsphere Formulation to Deter Abuse of Prescription Opioids by Smoking
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Artigo
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PLA-PCL Microsphere Formulation to Deter Abuse of Prescription Opioids by Smoking

Vasiukhina, Anastasiia ; Gad, Sheryhan F. ; Wellington, Elyssia N. ; Wilmes, Danielle M. ; Yeo, Yoon ; Solorio, Luis

International journal of pharmaceutics, 2022-10, Vol.626, p.122151-122151, Article 122151 [Periódico revisado por pares]

Netherlands: Elsevier B.V

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19
Optimization of a Series of Mu Opioid Receptor (MOR) Agonists with High G Protein Signaling Bias
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Optimization of a Series of Mu Opioid Receptor (MOR) Agonists with High G Protein Signaling Bias

Kennedy, Nicole M ; Schmid, Cullen L ; Ross, Nicolette C ; Lovell, Kimberly M ; Yue, Zhizhou ; Chen, Yen Ting ; Cameron, Michael D ; Bohn, Laura M ; Bannister, Thomas D

Journal of medicinal chemistry, 2018-10, Vol.61 (19), p.8895-8907 [Periódico revisado por pares]

United States: American Chemical Society

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20
Designing Safer Analgesics via μ-Opioid Receptor Pathways
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Designing Safer Analgesics via μ-Opioid Receptor Pathways

Chan, H.C. Stephen ; McCarthy, Dillon ; Li, Jianing ; Palczewski, Krzysztof ; Yuan, Shuguang

Trends in pharmacological sciences (Regular ed.), 2017-11, Vol.38 (11), p.1016-1037 [Periódico revisado por pares]

England: Elsevier Ltd

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