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1 |
Material Type: Artigo
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Design and synthesis of dihydrobenzofuran amides as orally bioavailable, centrally active γ-secretase modulatorsPettersson, Martin ; Johnson, Douglas S. ; Subramanyam, Chakrapani ; Bales, Kelly R. ; am Ende, Christopher W. ; Fish, Benjamin A. ; Green, Michael E. ; Kauffman, Gregory W. ; Lira, Ricardo ; Mullins, Patrick B. ; Navaratnam, Thayalan ; Sakya, Subas M. ; Stiff, Cory M. ; Tran, Tuan P. ; Vetelino, Beth C. ; Xie, Longfei ; Zhang, Liming ; Pustilnik, Leslie R. ; Wood, Kathleen M. ; O’Donnell, Christopher J.Bioorganic & medicinal chemistry letters, 2012-04, Vol.22 (8), p.2906-2911 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Novel CCR1 antagonists with improved metabolic stabilityBROWN, Matthew F ; AVERY, Mike ; LIRA, Paul D ; LILLIE, Brett M ; LUNDQUIST, Greg D ; MAIRS, Erin N ; MCELROY, Eric B ; MCGLYNN, Molly A ; PARADIS, Timothy J ; POSS, Christopher S ; ROSSULEK, Michelle I ; SHEPARD, Richard M ; BRISSETTE, William H ; SIMS, Jeff ; STRELEVITZ, Timothy J ; TRUESDELL, Susan ; TYLASKA, Laurie A ; YOON, Kwansik ; DEYE ZHENG ; CHANG, J. H ; COLIZZA, Kevin ; CONKLYN, Maryrose ; DIRICO, Amy P ; GLADUE, Ronald P ; KATH, John C ; KRUEGER, Suzanne SBioorganic & medicinal chemistry letters, 2004-05, Vol.14 (9), p.2175-2179 [Periódico revisado por pares]Oxford: ElsevierTexto completo disponível |
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Material Type: Artigo
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Piperazinyl CCR1 antagonists—optimization of human liver microsome stabilityBrown, Matthew F. ; Bahnck, Kevin B. ; Blumberg, Laura C. ; Brissette, William H. ; Burrell, Sara A. ; Driscoll, James P. ; Fedeles, Flavia ; Fisher, Michael B. ; Foti, Robert S. ; Gladue, Ronald P. ; Guzman-Martinez, Aikomari ; Hayward, Matthew M. ; Lira, Paul D. ; Lillie, Brett M. ; Lu, Yi ; Lundquist, Greg D. ; McElroy, Eric B. ; McGlynn, Molly A. ; Paradis, Timothy J. ; Poss, Christopher S. ; Roache, James H. ; Shavnya, Andrei ; Shepard, Richard M. ; Trevena, Kristen A. ; Tylaska, Laurie A.Bioorganic & medicinal chemistry letters, 2007-06, Vol.17 (11), p.3109-3112 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Potent small molecule CCR1 antagonistsKATH, John C ; BRISSETTE, William H ; MARTIN, William H ; MCELROY, Eric B ; MCGLYNN, Molly A ; PARADIS, Timothy J ; POSS, Christopher S ; STOCK, Ingrid A ; TYLASKA, Laurie A ; DEYE ZHENG ; BROWN, Matthew F ; CONKLYN, Maryrose ; DIRICO, Amy P ; DORFF, Peter ; GLADUE, Ronald P ; LILLIE, Brett M ; LIRA, Paul D ; MAIRS, Erin NBioorganic & medicinal chemistry letters, 2004-05, Vol.14 (9), p.2169-2173 [Periódico revisado por pares]Oxford: ElsevierTexto completo disponível |
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Material Type: Artigo
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Pyrimidine benzamide-based thrombopoietin receptor agonistsReiter, Lawrence A. ; Subramanyam, Chakrapani ; Mangual, Emilio J. ; Jones, Christopher S. ; Smeets, Marc I. ; Brissette, William H. ; McCurdy, Sandra P. ; Lira, Paul D. ; Linde, Robert G. ; Li, Qifang ; Zhang, Fangning ; Antipas, Amy S. ; Blumberg, Laura C. ; Doty, Jonathan L. ; Driscoll, James P. ; Munchhof, Michael J. ; Ripp, Sharon L. ; Shavnya, Andrei ; Shepard, Richard M. ; Sperger, Diana ; Thomasco, Lisa M. ; Trevena, Kristen A. ; Wolf-Gouveia, Lilli A. ; Zhang, LilingBioorganic & medicinal chemistry letters, 2007-10, Vol.17 (19), p.5447-5454 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |