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1 |
Material Type: Artigo
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Bisphosphonates Inhibit the Growth of Trypanosoma brucei, Trypanosoma cruzi, Leishmania donovani, Toxoplasma gondii, and Plasmodium falciparum: A Potential Route to ChemotherapyMARTIN, Michael B. ; GRIMLEY, Joshua S. ; LEWIS, Jared C. ; HEATH, Huel T. ; BAILEY, Brian N. ; KENDRICK, Howard ; YARDLEY, Vanessa ; CALDERA, Aura ; LIRA, Renee ; URBINA, Julio A. ; MORENO, Silvia N. J. ; DOCAMPO, Roberto ; CROFT, Simon L. ; OLDFIELD, EricJournal of medicinal chemistry, 2001-03, Vol.44 (6), p.909-916 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Amiodarone Has Intrinsic Anti-Trypanosoma cruzi Activity and Acts Synergistically with PosaconazoleBENAIM, Gustavo ; SANDERS, John M. ; GARCIA-MARCHáN, Yael ; COLINA, Claudia ; LIRA, Renee ; CALDERA, Aura R. ; PAYARES, Gilberto ; SANOJA, Cristina ; BURGOS, Juan Miguel ; LEON-ROSSELL, Annette ; CONCEPCION, Juan Luis ; SCHIJMAN, Alejandro G. ; LEVIN, Mariano ; OLDFIELD, Eric ; URBINA, Julio A.Journal of medicinal chemistry, 2006-02, Vol.49 (3), p.892-899 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Informant consensus factor and antibacterial activity of the medicinal plants used by the people of San Rafael Coxcatlán, Puebla, MéxicoCanales, M. ; Hernández, T. ; Caballero, J. ; Vivar, A. Romo de ; Avila, G. ; Duran, A. ; Lira, R.Journal of ethnopharmacology, 2005-03, Vol.97 (3), p.429-439 [Periódico revisado por pares]Shannon: Elsevier Ireland LtdTexto completo disponível |
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Material Type: Artigo
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The antinociceptive and anti-inflammatory activities of Piptadenia stipulacea Benth. (Fabaceae)de Queiroz, Aline Cavalcanti ; de Lira, Daysianne Pereira ; Dias, Thays de Lima Matos Freire ; de Souza, Éverton Tenório ; da Matta, Carolina Barbosa Brito ; de Aquino, Anansa Bezerra ; Silva, Luiz Henrique Agra Cavalcante ; da Silva, Diogo José Costa ; Mella, Eliane Aparecida Campessato ; Agra, Maria de Fátima ; Filho, José Maria Barbosa ; de Araújo-Júnior, João Xavier ; Santos, Bárbara Viviana de Oliveira ; Alexandre-Moreira, Magna SuzanaJournal of ethnopharmacology, 2010-03, Vol.128 (2), p.377-383 [Periódico revisado por pares]Shannon: Elsevier Ireland LtdTexto completo disponível |
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Material Type: Artigo
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Composition and antibacterial activity of essential oil of Lantana achyranthifolia Desf. (Verbenaceae)Hernández, T. ; Canales, M. ; Avila, J.G. ; García, A.M. ; Martínez, A. ; Caballero, J. ; Vivar, A. Romo de ; Lira, R.Journal of ethnopharmacology, 2005-01, Vol.96 (3), p.551-554 [Periódico revisado por pares]Shannon: Elsevier Ireland LtdTexto completo disponível |
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Material Type: Artigo
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Design and synthesis of dihydrobenzofuran amides as orally bioavailable, centrally active γ-secretase modulatorsPettersson, Martin ; Johnson, Douglas S. ; Subramanyam, Chakrapani ; Bales, Kelly R. ; am Ende, Christopher W. ; Fish, Benjamin A. ; Green, Michael E. ; Kauffman, Gregory W. ; Lira, Ricardo ; Mullins, Patrick B. ; Navaratnam, Thayalan ; Sakya, Subas M. ; Stiff, Cory M. ; Tran, Tuan P. ; Vetelino, Beth C. ; Xie, Longfei ; Zhang, Liming ; Pustilnik, Leslie R. ; Wood, Kathleen M. ; O’Donnell, Christopher J.Bioorganic & medicinal chemistry letters, 2012-04, Vol.22 (8), p.2906-2911 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Novel CCR1 antagonists with improved metabolic stabilityBROWN, Matthew F ; AVERY, Mike ; LIRA, Paul D ; LILLIE, Brett M ; LUNDQUIST, Greg D ; MAIRS, Erin N ; MCELROY, Eric B ; MCGLYNN, Molly A ; PARADIS, Timothy J ; POSS, Christopher S ; ROSSULEK, Michelle I ; SHEPARD, Richard M ; BRISSETTE, William H ; SIMS, Jeff ; STRELEVITZ, Timothy J ; TRUESDELL, Susan ; TYLASKA, Laurie A ; YOON, Kwansik ; DEYE ZHENG ; CHANG, J. H ; COLIZZA, Kevin ; CONKLYN, Maryrose ; DIRICO, Amy P ; GLADUE, Ronald P ; KATH, John C ; KRUEGER, Suzanne SBioorganic & medicinal chemistry letters, 2004-05, Vol.14 (9), p.2175-2179 [Periódico revisado por pares]Oxford: ElsevierTexto completo disponível |
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Material Type: Artigo
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Piperazinyl CCR1 antagonists—optimization of human liver microsome stabilityBrown, Matthew F. ; Bahnck, Kevin B. ; Blumberg, Laura C. ; Brissette, William H. ; Burrell, Sara A. ; Driscoll, James P. ; Fedeles, Flavia ; Fisher, Michael B. ; Foti, Robert S. ; Gladue, Ronald P. ; Guzman-Martinez, Aikomari ; Hayward, Matthew M. ; Lira, Paul D. ; Lillie, Brett M. ; Lu, Yi ; Lundquist, Greg D. ; McElroy, Eric B. ; McGlynn, Molly A. ; Paradis, Timothy J. ; Poss, Christopher S. ; Roache, James H. ; Shavnya, Andrei ; Shepard, Richard M. ; Trevena, Kristen A. ; Tylaska, Laurie A.Bioorganic & medicinal chemistry letters, 2007-06, Vol.17 (11), p.3109-3112 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and evaluation of 9-anilinothiazolo[5,4-b]quinoline derivatives as potential antitumoralsRodríguez-Loaiza, Pilar ; Quintero, Angelina ; Rodríguez-Sotres, Rogelio ; Solano, José D ; Lira-Rocha, AlfonsoEuropean journal of medicinal chemistry, 2004, Vol.39 (1), p.5-10 [Periódico revisado por pares]Oxford: Elsevier Masson SASTexto completo disponível |
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Material Type: Artigo
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Solid-Phase Library Synthesis, Screening, and Selection of Tight-Binding Reduced Peptide Bond Inhibitors of a Recombinant Leishmania mexicana Cysteine Protease BST. HILAIRE, Phaedria M. ; ALVES, Lira C. ; HERRERA, Fatima ; RENIL, Manat ; SANDERSON, Sanya J. ; MOTTRAM, Jeremy C. ; COOMBS, Graham H. ; JULIANO, Maria A. ; JULIANO, Luiz ; AREVALO, Jorge ; MELDAL, MortenJournal of medicinal chemistry, 2002-05, Vol.45 (10), p.1971-1982 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |