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Expanding the medicinally relevant chemical space with compound librariesLópez-Vallejo, Fabian ; Giulianotti, Marc A. ; Houghten, Richard A. ; Medina-Franco, José L.Drug discovery today, 2012-07, Vol.17 (13-14), p.718-726 [Periódico revisado por pares]Kidlington: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Automated high throughput ADME assays for metabolic stability and cytochrome P450 inhibition profiling of combinatorial librariesJenkins, Kelly M. ; Angeles, Reginald ; Quintos, Marianne T. ; Xu, Rongda ; Kassel, Daniel B. ; Rourick, Robyn A.Journal of pharmaceutical and biomedical analysis, 2004-03, Vol.34 (5), p.989-1004 [Periódico revisado por pares]Amsterdam: Elsevier B.VTexto completo disponível |
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Automated medicinal chemistryKoppitz, Marcus ; Eis, KnutDrug discovery today, 2006-06, Vol.11 (11), p.561-568 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Selective Optimization of Side Activities: Another Way for Drug DiscoveryWermuth, Camille GJournal of medicinal chemistry, 2004-03, Vol.47 (6), p.1303-1314 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Lead optimization in the nondrug-like spaceZhao, HongyuDrug discovery today, 2011-02, Vol.16 (3), p.158-163 [Periódico revisado por pares]Kidlington: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Enzymes in the synthesis of bioactive compounds: the prodigious decadesGarcı́a-Junceda, Eduardo ; Garcı́a-Garcı́a, Juan Francisco ; Bastida, Agatha ; Fernández-Mayoralas, AlfonsoBioorganic & Medicinal Chemistry, 2004-04, Vol.12 (8), p.1817-1834 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Bis-Acridines as Lead Antiparasitic Agents: Structure-Activity Analysis of a Discrete Compound Library In VitroCAFFREY, Conor R ; STEVERDING, Dietmar ; LAND, Kirkwood M ; BEAUCHENE, Jessica ; SCHREIBER, Kimberly ; MOLL, Heidrun ; PONTE-SUCRE, Alicia ; SCHIRMEISTER, Tanja ; SARAVANAMUTHU, Ahilan ; FAIRLAMB, Alan H ; COHEN, Fred E ; MCKERROW, James H ; SWENERTON, Ryan K ; WEISMAN, Jennifer L ; MAY, Barnaby C. H ; KELLY, Ben ; WALSHE, Deirdre ; DEBNATH, Anjan ; ZHOU, Yuan-Min ; DOYLE, Patricia S ; FAFARMAN, Aaron T ; ZORN, Julie AAntimicrobial Agents and Chemotherapy, 2007-06, Vol.51 (6), p.2164-2172 [Periódico revisado por pares]Washington, DC: American Society for MicrobiologyTexto completo disponível |
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Material Type: Artigo
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Defining and maintaining a high quality screening collection: the GSK experienceLane, Stephen J. ; Eggleston, Drake S. ; Brinded, Keith A. ; Hollerton, John C. ; Taylor, Nicholas L. ; Readshaw, Simon A.Drug discovery today, 2006-03, Vol.11 (5-6), p.267-272 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Scaffold hopping and optimization towards libraries of glycogen synthase kinase-3 inhibitorsNærum, Lars ; Nørskov-Lauritsen, Leif ; Olesen, Preben HBioorganic & medicinal chemistry letters, 2002-06, Vol.12 (11), p.1525-1528 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Natural Products as Sources of New Drugs over the Last 25 YearsNewman, David J ; Cragg, Gordon MJournal of natural products (Washington, D.C.), 2007-03, Vol.70 (3), p.461-477 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |