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1
Discovery and SAR of Novel 2,3-Dihydroimidazo[1,2-c]quinazoline PI3K Inhibitors: Identification of Copanlisib (BAY 80-6946)
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Discovery and SAR of Novel 2,3-Dihydroimidazo[1,2-c]quinazoline PI3K Inhibitors: Identification of Copanlisib (BAY 80-6946)

Scott, William J. ; Hentemann, Martin F. ; Rowley, R. Bruce ; Bull, Cathy O. ; Jenkins, Susan ; Bullion, Ann M. ; Johnson, Jeffrey ; Redman, Anikó ; Robbins, Arthur H. ; Esler, William ; Fracasso, R. Paul ; Garrison, Timothy ; Hamilton, Mark ; Michels, Martin ; Wood, Jill E. ; Wilkie, Dean P. ; Xiao, Hong ; Levy, Joan ; Stasik, Enrico ; Liu, Ningshu ; Schaefer, Martina ; Brands, Michael ; Lefranc, Julien

ChemMedChem, 2016-07, Vol.11 (14), p.1517-1530 [Periódico revisado por pares]

Germany: Blackwell Publishing Ltd

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2
An Efficient Synthesis of bi‐Aryl Pyrimidine Heterocycles: Potential New Drug Candidates to Treat Alzheimer's Disease
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An Efficient Synthesis of bi‐Aryl Pyrimidine Heterocycles: Potential New Drug Candidates to Treat Alzheimer's Disease

Rehman, Tanzeel Ur ; Khan, Islam Ullah ; Ashraf, Muhammad ; Tarazi, Hamadeh ; Riaz, Sadaf ; Yar, Muhammad

Archiv der Pharmazie (Weinheim), 2017-04, Vol.350 (3-4), p.n/a [Periódico revisado por pares]

Germany: Wiley Subscription Services, Inc

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3
Pyrazolopyrimidines: Potent Inhibitors Targeting the Capsid of Rhino- and Enteroviruses
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Pyrazolopyrimidines: Potent Inhibitors Targeting the Capsid of Rhino- and Enteroviruses

Makarov, Vadim A. ; Braun, Heike ; Richter, Martina ; Riabova, Olga B. ; Kirchmair, Johannes ; Kazakova, Elena S. ; Seidel, Nora ; Wutzler, Peter ; Schmidtke, Michaela

ChemMedChem, 2015-10, Vol.10 (10), p.1629-1634 [Periódico revisado por pares]

Weinheim: WILEY-VCH Verlag

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4
Structure-Activity Relationships of 2-Sufonylpyrimidines as Quorum-Sensing Inhibitors to Tackle Biofilm Formation and eDNA Release of Pseudomonas aeruginosa
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Structure-Activity Relationships of 2-Sufonylpyrimidines as Quorum-Sensing Inhibitors to Tackle Biofilm Formation and eDNA Release of Pseudomonas aeruginosa

Thomann, Andreas ; Brengel, Christian ; Börger, Carsten ; Kail, Dagmar ; Steinbach, Anke ; Empting, Martin ; Hartmann, Rolf W.

ChemMedChem, 2016-11, Vol.11 (22), p.2522-2533 [Periódico revisado por pares]

Germany: Blackwell Publishing Ltd

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5
Microwave Assisted Synthesis of Pyrimidines in Ionic Liquid and Their Potency as Non-Classical Malarial Antifolates
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Microwave Assisted Synthesis of Pyrimidines in Ionic Liquid and Their Potency as Non-Classical Malarial Antifolates

Bhatt, Jaimin D. ; Chudasama, Chaitanya J. ; Patel, Kanuprasad D.

Archiv der Pharmazie (Weinheim), 2016-10, Vol.349 (10), p.791-800 [Periódico revisado por pares]

Germany: Blackwell Publishing Ltd

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6
Design, Synthesis and Biological Evaluation of 4-Amino-N-(4-aminophenyl)benzamide Analogues of Quinoline-Based SGI-1027 as Inhibitors of DNA Methylation
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Design, Synthesis and Biological Evaluation of 4-Amino-N-(4-aminophenyl)benzamide Analogues of Quinoline-Based SGI-1027 as Inhibitors of DNA Methylation

Rilova, Elodie ; Erdmann, Alexandre ; Gros, Christina ; Masson, Véronique ; Aussagues, Yannick ; Poughon-Cassabois, Valérie ; Rajavelu, Arumugam ; Jeltsch, Albert ; Menon, Yoann ; Novosad, Natacha ; Gregoire, Jean-Marc ; Vispé, Stéphane ; Schambel, Philippe ; Ausseil, Fréderic ; Sautel, François ; Arimondo, Paola B. ; Cantagrel, Frédéric

ChemMedChem, 2014-03, Vol.9 (3), p.590-601 [Periódico revisado por pares]

Weinheim: WILEY-VCH Verlag

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7
Novel Antiviral Compounds against Gastroenteric Viral Infections
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Novel Antiviral Compounds against Gastroenteric Viral Infections

Mohamed, Mosaad S. ; Abd El-Hameed, Rania H. ; Sayed, Amira I. ; Soror, Sameh H.

Archiv der Pharmazie (Weinheim), 2015-03, Vol.348 (3), p.194-205 [Periódico revisado por pares]

Germany: Blackwell Publishing Ltd

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8
Design and Synthesis of 4-Anilinothieno[2,3-d]pyrimidine-Based Compounds as Dual EGFR/HER-2 Inhibitors
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Design and Synthesis of 4-Anilinothieno[2,3-d]pyrimidine-Based Compounds as Dual EGFR/HER-2 Inhibitors

Abd El Hadi, Soha R. ; Lasheen, Deena S. ; Hassan, Mahmoud A. ; Abouzid, Khaled A. M.

Archiv der Pharmazie (Weinheim), 2016-11, Vol.349 (11), p.827-847 [Periódico revisado por pares]

Germany: Blackwell Publishing Ltd

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9
Synthesis of Some Pyrazolines and Pyrimidines Derived from Polymethoxy Chalcones as Anticancer and Antimicrobial Agents
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Synthesis of Some Pyrazolines and Pyrimidines Derived from Polymethoxy Chalcones as Anticancer and Antimicrobial Agents

Rostom, Sherif A.F. ; Badr, Mona H. ; Abd El Razik, Heba A. ; Ashour, Hayam M.A. ; Abdel Wahab, Abeer E.

Archiv der Pharmazie (Weinheim), 2011-09, Vol.344 (9), p.572-587 [Periódico revisado por pares]

Weinheim: WILEY-VCH Verlag

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10
Synthesis and Biological Evaluation of Novel 6-Hydrazinyl-2,4-bismorpholino pyrimidine and 1,3,5-Triazine Derivatives as Potential Antitumor Agents
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Synthesis and Biological Evaluation of Novel 6-Hydrazinyl-2,4-bismorpholino pyrimidine and 1,3,5-Triazine Derivatives as Potential Antitumor Agents

Zhu, Wufu ; Liu, Yajing ; Zhao, Yanfang ; Wang, Haiyan ; Tan, Li ; Fan, Weijie ; Gong, Ping

Archiv der Pharmazie (Weinheim), 2012-10, Vol.345 (10), p.812-821 [Periódico revisado por pares]

Weinheim: WILEY-VCH Verlag

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