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1 |
Material Type: Artigo
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Synthesis and profiling of benzylmorpholine 1,2,4,5-tetraoxane analogue N205: Towards tetraoxane scaffolds with potential for single dose cure of malariaO' Neill, Paul M. ; Stocks, Paul A. ; Sabbani, Sunil ; Roberts, Natalie L. ; Amewu, Richard K. ; Shore, Emma R. ; Aljayyoussi, Ghaith ; Angulo-Barturén, Iñigo ; Belén, María ; Jiménez-Díaz ; Bazaga, Santiago Ferrer ; Martínez, María Santos ; Campo, Brice ; Sharma, Raman ; Charman, Susan A. ; Ryan, Eileen ; Chen, Gong ; Shackleford, David M. ; Davies, Jill ; Nixon, Gemma L. ; Biagini, Giancarlo A. ; Ward, Stephen A.Bioorganic & medicinal chemistry, 2018-07, Vol.26 (11), p.2996-3005 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Antihyperlipidemic morpholine derivatives with antioxidant activity: An investigation of the aromatic substitutionLadopoulou, Eleni M. ; Matralis, Alexios N. ; Nikitakis, Anastasios ; Kourounakis, Angeliki P.Bioorganic & medicinal chemistry, 2015-11, Vol.23 (21), p.7015-7023 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Microwave-assisted synthesis of quinoline, isoquinoline, quinoxaline and quinazoline derivatives as CB2 receptor agonistsSaari, Raimo ; Törmä, Jonna-Carita ; Nevalainen, TapioBioorganic & medicinal chemistry, 2011-01, Vol.19 (2), p.939-950 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis, docking study and neuroprotective effects of some novel pyrano[3,2-c]chromene derivatives bearing morpholine/phenylpiperazine moietySameem, Bilqees ; Saeedi, Mina ; Mahdavi, Mohammad ; Nadri, Hamid ; Moghadam, Farshad Homayouni ; Edraki, Najmeh ; Khan, Muhammad Imran ; Amini, MohsenBioorganic & medicinal chemistry, 2017-08, Vol.25 (15), p.3980-3988 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Optimization and biological evaluation of 2-aminobenzothiazole derivatives as Aurora B kinase inhibitorsLee, Eun ; An, Ying ; Kwon, Junhee ; Kim, Keun Il ; Jeon, RaokBioorganic & medicinal chemistry, 2017-07, Vol.25 (14), p.3614-3622 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis of novel compounds containing morpholine and 5(4H)-oxazolone rings as potent tyrosinase inhibitorsHamidian, Hooshang ; Azizi, SimaBioorganic & medicinal chemistry, 2015-11, Vol.23 (21), p.7089-7094 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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1,2-Benzisothiazol-3-one derivatives as a novel class of small-molecule caspase-3 inhibitorsWu, Lixin ; Lu, Meiqi ; Yan, Zhihui ; Tang, Xiaobin ; Sun, Bo ; Liu, Wei ; Zhou, Honggang ; Yang, ChengBioorganic & medicinal chemistry, 2014-04, Vol.22 (8), p.2416-2426 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma actionBozdag, Murat ; Carta, Fabrizio ; Vullo, Daniela ; Akdemir, Atilla ; Isik, Semra ; Lanzi, Cecilia ; Scozzafava, Andrea ; Masini, Emanuela ; Supuran, Claudiu T.Bioorganic & medicinal chemistry, 2015-05, Vol.23 (10), p.2368-2376 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis, in vitro and in vivo evaluation of fluorine-18 labelled FE-GW405833 as a PET tracer for type 2 cannabinoid receptor imagingEvens, Nele ; Vandeputte, Caroline ; Muccioli, Giulio G. ; Lambert, Didier M. ; Baekelandt, Veerle ; Verbruggen, Alfons M. ; Debyser, Zeger ; Van Laere, Koen ; Bormans, Guy M.Bioorganic & medicinal chemistry, 2011-08, Vol.19 (15), p.4499-4505 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
10 |
Material Type: Artigo
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Design, chemical synthesis and biological evaluation of 3-spiromorpholinone/3-spirocarbamate androsterone derivatives as inhibitors of 17β-hydroxysteroid dehydrogenase type 3Djigoué, Guy Bertrand ; Kenmogne, Lucie Carolle ; Roy, Jenny ; Maltais, René ; Poirier, DonaldBioorganic & medicinal chemistry, 2015-09, Vol.23 (17), p.5433-5451 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |