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Material Type: Artigo
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Design, synthesis, and biological evaluation of dinaciclib and CAN508 hybrids as CDK inhibitorsOdeh, Dana M. ; Allam, Heba Abdelrasheed ; Baselious, Fady ; Mahmoud, Walaa R. ; Odeh, Mohanad M. ; Ibrahim, Hany S. ; Abdel‐Aziz, Hatem A. ; Mohammed, Eman R.Drug development research, 2024-05, Vol.85 (3), p.e22193-n/a [Periódico revisado por pares]United States: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Novel Antiviral Compounds against Gastroenteric Viral InfectionsMohamed, Mosaad S. ; Abd El-Hameed, Rania H. ; Sayed, Amira I. ; Soror, Sameh H.Archiv der Pharmazie (Weinheim), 2015-03, Vol.348 (3), p.194-205 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |
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Material Type: Artigo
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Preferential Inhibition of JAK1 Relative to JAK3 by Upadacitinib: Exposure‐Response Analyses of Ex Vivo Data From 2 Phase 1 Clinical Trials and Comparison to TofacitinibMohamed, Mohamed‐Eslam F. ; Beck, Denise ; Camp, Heidi S. ; Othman, Ahmed A.Journal of clinical pharmacology, 2020-02, Vol.60 (2), p.188-197 [Periódico revisado por pares]England: American College of Clinical PharmacologyTexto completo disponível |
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Material Type: Artigo
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Design, synthesis, and in vitro biological evaluation of novel thiazolopyrimidine derivatives as antileishmanial compoundsIstanbullu, Huseyin ; Bayraktar, Gulsah ; Akbaba, Hasan ; Cavus, Ibrahim ; Coban, Gunes ; Debelec Butuner, Bilge ; Kilimcioglu, Ali Ahmet ; Ozbilgin, Ahmet ; Alptuzun, Vildan ; Erciyas, ErcinArchiv der Pharmazie (Weinheim), 2020-08, Vol.353 (8), p.e1900325-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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1,2,4‐Triazole and benzimidazole fused dihydropyrimidine derivatives: Design, green synthesis, antibacterial, antitubercular, and antimalarial activitiesMokariya, Jaydeep A. ; Rajani, Dhanji P. ; Patel, Manish P.Archiv der Pharmazie (Weinheim), 2023-04, Vol.356 (4), p.e2200545-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Population Pharmacokinetics and Exposure‐Response Analyses for the Most Frequent Adverse Events Following Treatment With Lemborexant, an Orexin Receptor Antagonist, in Subjects With Insomnia DisorderLalovic, Bojan ; Majid, Oneeb ; Aluri, Jagadeesh ; Landry, Ishani ; Moline, Margaret ; Hussein, ZiadJournal of clinical pharmacology, 2020-12, Vol.60 (12), p.1642-1654 [Periódico revisado por pares]England: American College of Clinical PharmacologyTexto completo disponível |
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Material Type: Artigo
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Synthesis, molecular docking studies, and biological evaluation of novel alkyl bis(4‐amino‐5‐cyanopyrimidine) derivativesBoualia, Imen ; Derabli, Chamseddine ; Boulcina, Raouf ; Bensouici, Chawki ; Yildirim, Muhammet ; Birinci Yildirim, Arzu ; Mokrani, El Hassen ; Debache, AbdelmadjidArchiv der Pharmazie (Weinheim), 2019-11, Vol.352 (11), p.e1900027-n/a [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Sensitive CE‐MS method for monitoring of riociguat and desmethylriociguat levels in human serumHložek, Tomáš ; Štícha, Martin ; Bursová, Miroslava ; Jelínek, Ivan ; Tůma, Petr ; Čabala, RadomírElectrophoresis, 2020-10, Vol.41 (18-19), p.1564-1567 [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Design, synthesis, and antiviral evaluation of novel hydrazone‐substituted thiophene[3,2‐d]pyrimidine derivatives as potent human immunodeficiency virus‐1 inhibitorsWang, Zhao ; Kang, Dongwei ; Chen, Meng ; Wu, Gaochan ; Feng, Da ; Zhao, Tong ; Zhou, Zhongxia ; Huo, Zhipeng ; Jing, Lanlan ; Zuo, Xiaofang ; Daelemans, Dirk ; De Clercq, Erik ; Pannecouque, Christophe ; Zhan, Peng ; Liu, XinyongChemical biology & drug design, 2018-12, Vol.92 (6), p.2009-2021 [Periódico revisado por pares]EnglandTexto completo disponível |
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Material Type: Artigo
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Herpes Zoster and Tofacitinib Therapy in Patients With Rheumatoid ArthritisWinthrop, Kevin L. ; Yamanaka, Hisashi ; Valdez, Hernan ; Mortensen, Eric ; Chew, Robert ; Krishnaswami, Sriram ; Kawabata, Thomas ; Riese, RichardArthritis & rheumatology (Hoboken, N.J.), 2014-10, Vol.66 (10), p.2675-2684 [Periódico revisado por pares]United States: Wiley Subscription Services, IncTexto completo disponível |