Hit-to-lead optimization of a benzene sulfonamide series for potential antileishmanial agents
Paul J. Koovits Marcos A Dessoy; An Matheeussen; Louis Maes; Guy Caljon; Leonardo Luiz Gomes Ferreira; Rafael Consolin Chelucci; Simone Michelan Duarte; Adriano Defini Andricopulo; Simon Campbell; Jadel M Kratz; Charles E Mowbray; Luiz C Dias https://orcid.org/0000-0003-0628-9928
RSC Medicinal Chemistry Cambridge : Royal Society of Chemistry - RSC v. 11, n. 11, p. 1267-1274, Nov. 2020
Cambridge 2020
Localização:
IFSC - Inst. Física de São Carlos
(PROD030698 )(Acessar)
2-aminobenzimidazoles for leishmaniasis from initial hit discovery to in vivo profiling
Rafael Augusto Alves Ferreira Celso de Rezende Junior; Pablo David Grigol Martinez; Paul John Koovits; Bruna Miranda Soares; Leonardo Luiz Gomes Ferreira; Simone Michelan Duarte; Rafael Consolin Chelucci; Adriano Defini Andricopulo; Mariana Kolos Galuppo; Silvia Reni Bortolin Uliana; An Matheeussen; Guy Caljon; Louis Maes; Simon Campbell; Jadel M Kratz; Charles E Mowbray; Luiz Carlos Dias https://orcid.org/0000-0003-0628-9928
PLOS Neglected Tropical Diseases San Francisco v. 15, n. 2, p. e0009196-1-e0009196-20, Feb. 2021
San Francisco 2021
Localização:
IFSC - Inst. Física de São Carlos
(PROD031370 )(Acessar)
Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease
Celso de Oliveira Rezende Junior Pablo David Grigol Martinez; Rafael Augusto Alves Ferreira; Paul John Koovits; Bruna Miranda Soares; Leonardo Luiz Gomes Ferreira; Simone Michelan Duarte; Rafael Consolin Chelucci; Adriano Defini Andricopulo; An Matheeussen; Natascha Van Pelt; Guy Caljon; Louis Maes; Simon Campbell; Jadel Muller Kratz; Charles E Mowbray; Luiz Carlos Dias
European Journal of Medicinal Chemistry Issy-les-Moulineaux v. 246, p. 114925-1-114925-10 + supplementary data, Jan. 2023
Issy-les-Moulineaux 2023
Localização:
IFSC - Inst. Física de São Carlos
(PROD033848 )(Acessar)