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Material Type: Artigo
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How To Design a Successful p53-MDM2/X Interaction Inhibitor: A Thorough Overview Based on Crystal StructuresEstrada-Ortiz, Natalia ; Neochoritis, Constantinos G. ; Dömling, AlexanderChemMedChem, 2016-04, Vol.11 (8), p.757-772 [Periódico revisado por pares]Germany: Blackwell Publishing LtdTexto completo disponível |
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Material Type: Artigo
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Exhaustive Fluorine Scanning toward Potent p53-Mdm2 AntagonistsHuang, Yijun ; Wolf, Siglinde ; Koes, David ; Popowicz, Grzegorz M. ; Camacho, Carlos J. ; Holak, Tad A. ; Dömling, AlexanderChemMedChem, 2012-01, Vol.7 (1), p.49-52 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
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Material Type: Artigo
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Isocyanides as InfluenzaA Virus Subtype H5N1 Wild-Type M2 Channel InhibitorsWu, Shuwen ; Huang, Jing ; Gazzarrini, Sabrina ; He, Si ; Chen, Lihua ; Li, Jun ; Xing, Li ; Li, Chufang ; Chen, Ling ; Neochoritis, Constantinos G ; Liao, George P ; Zhou, Haibing ; Domling, Alexander ; Moroni, Anna ; Wang, WeiChemMedChem, 2015-11, Vol.10 (11), p.1837-1845 [Periódico revisado por pares]Weinheim: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Two‐Step Synthesis of Complex Artificial Macrocyclic CompoundsMadhavachary, Rudrakshula ; Abdelraheem, Eman M. M. ; Rossetti, Arianna ; Twarda‐Clapa, Aleksandra ; Musielak, Bogdan ; Kurpiewska, Katarzyna ; Kalinowska‐Tłuścik, Justyna ; Holak, Tad A. ; Dömling, AlexanderAngewandte Chemie, 2017-08, Vol.129 (36), p.10865-10869 [Periódico revisado por pares]Weinheim: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Discovery of a Potent Allosteric Kinase Modulator by Combining Computational and Synthetic MethodsKroon, Edwin ; Schulze, Jörg O. ; Süß, Evelyn ; Camacho, Carlos J. ; Biondi, Ricardo M. ; Dömling, AlexanderAngewandte Chemie, 2015-11, Vol.127 (47), p.14139-14142 [Periódico revisado por pares]Weinheim: WILEY‐VCH VerlagTexto completo disponível |
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Material Type: Artigo
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Jetzt wird es ernst: strukturbasiertes Design von Mdm2/Mdmx-p53-InhibitorenPopowicz, Grzegorz M. ; Dömling, Alexander ; Holak, Tad A.Angewandte Chemie, 2011-03, Vol.123 (12), p.2732-2741 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
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Material Type: Artigo
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Robust Generation of Lead Compounds for Protein-Protein Interactions by Computational and MCR Chemistry: p53/Hdm2 AntagonistsCzarna, Anna ; Beck, Barbara ; Srivastava, Stuti ; Popowicz, Grzegorz M. ; Wolf, Siglinde ; Huang, Yijun ; Bista, Michal ; Holak, Tad A. ; Dömling, AlexanderAngewandte Chemie, 2010-07, Vol.122 (31), p.5480-5484 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
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Material Type: Artigo
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Programmed Death-1: therapeutischer Erfolg nach über 100 Jahren KrebsimmuntherapieDömling, Alexander ; Holak, Tad A.Angewandte Chemie, 2014-02, Vol.126 (9), p.2318-2320 [Periódico revisado por pares]Weinheim: WILEY-VCH VerlagTexto completo disponível |
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Material Type: Artigo
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Berichtigung: Efficient Assembly of Iminodicarboxamides by a “Truly” Four‐Component ReactionKhoury, Kareem ; Sinha, Mantosh K. ; Nagashima, Tadamichi ; Herdtweck, Eberhardt ; Dömling, AlexanderAngewandte Chemie, 2013-05, Vol.125 (21), p.5535-5535 [Periódico revisado por pares]Weinheim: Wiley Subscription Services, IncTexto completo disponível |
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Material Type: Artigo
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Ivar Ugi (1930-2005)Dömling, AlexanderNachrichten aus der Chemie, 2006-02, Vol.54 (2), p.159-159 [Periódico revisado por pares]Weinheim/Bergstr: Wiley-VCH Verlag GmbH & Co. KGaATexto completo disponível |