Novel trypanocidal thiophen-chalcone cruzain inhibitors structure- and ligand-based studies
Aldo Sena de Oliveira Marilia Valli; Leonardo Luiz Gomes Ferreira; Julia Medeiros Souza; Renata Krogh Andricopulo; Lidiane Meier; Heitor R Abreu; BrunaG Voltolini; Luana C Llanes; Ricardo José Nunes; Antonio L Braga; Adriano Defini Andricopulo
Future Medicinal Chemistry London v. 14, n. 11, p. 795-808, June 2022
London 2022
Localização:
IFSC - Inst. Física de São Carlos
(PROD033126-SC )(Acessar)
2-aminobenzimidazoles for leishmaniasis from initial hit discovery to in vivo profiling
Rafael Augusto Alves Ferreira Celso de Rezende Junior; Pablo David Grigol Martinez; Paul John Koovits; Bruna Miranda Soares; Leonardo Luiz Gomes Ferreira; Simone Michelan Duarte; Rafael Consolin Chelucci; Adriano Defini Andricopulo; Mariana Kolos Galuppo; Silvia Reni Bortolin Uliana; An Matheeussen; Guy Caljon; Louis Maes; Simon Campbell; Jadel M Kratz; Charles E Mowbray; Luiz Carlos Dias https://orcid.org/0000-0003-0628-9928
PLOS Neglected Tropical Diseases San Francisco v. 15, n. 2, p. e0009196-1-e0009196-20, Feb. 2021
San Francisco 2021
Localização:
IFSC - Inst. Física de São Carlos
(PROD031370 )(Acessar)
Hit-to-lead optimization of a 2-aminobenzimidazole series as new candidates for chagas disease
Celso de Oliveira Rezende Junior Pablo David Grigol Martinez; Rafael Augusto Alves Ferreira; Paul John Koovits; Bruna Miranda Soares; Leonardo Luiz Gomes Ferreira; Simone Michelan Duarte; Rafael Consolin Chelucci; Adriano Defini Andricopulo; An Matheeussen; Natascha Van Pelt; Guy Caljon; Louis Maes; Simon Campbell; Jadel Muller Kratz; Charles E Mowbray; Luiz Carlos Dias
European Journal of Medicinal Chemistry Issy-les-Moulineaux v. 246, p. 114925-1-114925-10 + supplementary data, Jan. 2023
Issy-les-Moulineaux 2023
Localização:
IFSC - Inst. Física de São Carlos
(PROD033848 )(Acessar)