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1
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Conference Paper
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Structural insights into inorganic NO donors as inhibitors of Trypanosoma cruzi glyceraldehyde-3-phosphate dehydrogenase

T. L. Balliano Rafael Victório Carvalho Guido; F. O. N Silva; L. G. F Lopes; N Silva; Adriano Defini Andricopulo; Glaucius Oliva; International Network of Protein Engineering Centers - INPEC (18. 2009 Ubatuba)

Abstract Book São Carlos : Instituto de Física de São Carlos - USP, 2009

São Carlos Instituto de Física de São Carlos - USP 2009

Available at IFSC - Inst. Física de São Carlos    (PROD016915 ) and other locations(GetIt)

2
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Article
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Structure-activity relationships of novel N-imidazoylpiperazines with potent anti-trypanosoma cruzi activity

Rocio Marisol Espinoza Chávez Celso de Oliveira Rezende Junior; Mariana Laureano de Souza; Ivani Pauli; Marilia Valli; Leonardo Luiz Gomes Ferreira; Rafael Consolin Chelucci; Simone Michelan Duarte; Renata Krogh; Fernando Bezerra Romualdo da Silva; Fábio Cardoso Cruz; Aldo Sena de Oliveira; Adriano Defini Andricopulo; Luiz Carlos Dias

Future Medicinal Chemistry London v. 16, n. 3, p. 253-269, Jan. 2024

London 2024

Available at IFSC - Inst. Física de São Carlos    (PROD035642-SC )(GetIt)

3
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Article
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Multiparameter optimization of Trypanocidal cruzain inhibitors with in vivo activity and favorable pharmacokinetics

Ivani Pauli Celso de Oliveira Rezende Junior; Brian W Slafer; Marco A Dessoy; Mariana Laureano de Souza; Leonardo Luiz Gomes Ferreira; Abraham L. M Adjanohun; Rafaela S Ferreira; Luma Godoy Magalhães; Renata Krogh Andricopulo; Simone Michelan Duarte; Ricardo Vaz Del Pintor; Fernando B. R. da Silva; Fabio C Cruz; Luiz C Dias; Adriano Defini Andricopulo

Frontiers in Pharmacology Lausanne v. 12, p. 774069-1-774069-21 + supplementary material, Jan. 2022

Lausanne 2022

Available at IFSC - Inst. Física de São Carlos    (PROD032730 )(GetIt)

4
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Conference Paper
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Design, synthesis and biochemistry evaluation of novel (E)-Cinnamic N-acylhydrazone antichagasic candidates

Gustavo Henrique Goulart Trossini Elizabeth Igne Ferreira; Samir Carvalho; Larisse Feitosa; Maria Henriques; Kelly Salomão; Solange Castro; Marcel Kaiser; Reto Brun; James Wardell; Solange Wardell; Edson F Silva; Thadeu Costa; Adriano Defini Andricopulo; Carlos Alberto Manssour Fraga; Spring National Meeting and Exposition (243. 2012 San Diego)

Abstracts Washington, DC : American Chemical Society - ACS, 2012

Washington, DC American Chemical Society - ACS 2012

Available at IFSC - Inst. Física de São Carlos    (PROD019405 ) and other locations(GetIt)

5
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Conference Paper
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Discovering the potential of the secondary metabolites from Malouetia tamaquarina (Apocynaceae) and its endophytes against neglected tropical diseases

Kamila T. Yuyama Claudia C Macedo; Weilan Gomes da Paixão Melo; Matheus Henrique da Silva; Icaro N Lima; Thayna M Souza; Yuri B Souza; Jaime P. L Aguiar; Ana C. D Castello; Leonardo Luiz Gomes Ferreira; Adriano Defini Andricopulo; Gilvan F Silva; Thomas J Schmidt; Mônica Tallarico Pupo; Research Network Natural Products against Neglected Diseases - ResNet NPDN - Anniversary Online Symposium (10. 2021 Virtual)

Program and Book of Abstracts Münster : University of Münster, 2021

Münster University of Münster 2021

Available at IFSC - Inst. Física de São Carlos    (PROD032701 )(GetIt)

6
Material Type:
Article
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Discovery of indolizine lactones as anticancer agents and their optimization through late-stage functionalization

Thiago Sabino da Silva Matheus da Silva Souza; Adriano Defini Andricopulo; Fernando Antonio Santos Coelho

RSC Advances Cambridge, UK v. 2023, n. 29, p. 20264-20270 + supplementary information: 1-128, 2023

Cambridge, UK 2023

Available at IFSC - Inst. Física de São Carlos    (PROD034683 )(GetIt)

7
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Conference Paper
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Planejamento de chalconas com atividade antimitótica

Lívia B. Salum Louise D Chiaradia; Laura L Vollmer; Marlon N. S Cordeiro; Evelyn Winter; Fernanda S Pedrini; Hikmat N Daghestani; Maria Cláudia Santos da Silva; Tânia B Creczynski-Pasa; Ricardo J Nunes; Rosendo A Yunes; Adriano Defini Andricopulo; Billy W Day; Andreas Vogt; Reunião Anual Sociedade Brasileira de Química - SBQ (34. 2011 Florianópolis)

Programa e Resumos São Paulo : Sociedade Brasileira de Química - SBQ, 2011

São Paulo Sociedade Brasileira de Química - SBQ 2011

Online access. The library also has physical copies.

8
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Article
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Liquid fungal cocultivation as a strategy to access bioactive metabolites

Airton Damasceno Silva Alessandra Regina Pepe Ambrozin; Ana Flávia Silveira de Camargo; Felipe de Paula Nogueira Cruz; Leonardo Luiz Gomes Ferreira; Renata Krogh Andricopulo; Taynara Lopes Silva; Ilana Lopes Baratella da Cunha Camargo; Adriano Defini Andricopulo; Paulo Cezar Vieira

Planta Medica Stuttgart : Georg Thieme Verlag v. 87, n. 1/2, p. 187-195, Feb. 2021

Stuttgart 2021

Available at FCFRP - Fac. Ciên. Farm. Ribeirão Preto    (pcd 3018357 Acervo Digital ) and other locations(GetIt)

9
Material Type:
Conference Paper
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Structure-activity relationships of β-chalcogenamines synthesis, enzyme inhibition, molecular docking and QSAR studies

Cleiton da Silva Ricardo Beche; Aldo Oliveira; David Salcedo; Adriano Defini Andricopulo; Fabio Galetto; Brazilian Symposium on Medicinal Chemistry - BrazMedChem (9. 2019 Pirenópolis)

Anais eletrônicos Campinas : Galoá

Campinas Galoá 2019

Online access. The library also has physical copies.

10
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Conference Paper
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Triagem in vitro de compostos ativos frente linhagem celular de câncer de mama triplo-negativa e metastática

F. R. F. D. Costa Matheus da Silva Souza; Adriano Defini Andricopulo; Semana Integrada do Instituto de Física de São Carlos - SIFSC (10. 2020 São Carlos)

Livro de Resumos São Carlos : Instituto de Física de São Carlos - IFSC, 2020

São Carlos Instituto de Física de São Carlos - IFSC 2020

Online access. The library also has physical copies.

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