synthesis, antichagasic in vitro evaluation, cytotoxicity assays, molecular modeling and SAR/QSAR studies of a 2-phenyl-3-(1-phenyl-1H-pyrazol-4-yl)-acrylic acid benzylidene-carbohydrazide series
Maria A. F. Vera DiVaio Antônio C. C Freitas; Helena C Castro; Sérgio de Albuquerque; Lucio M Cabral; Carlos Ribeiro Rodrigues; Magaly G Albuquerque; Rita C. A Martins; Maria das Graças M. O Henriques; Luiza R. S Dias
Bioorganic and Medicinal Chemistry Oxford v. 17, n. 1, p. 295-302, 2009
synthesis, antichagasic in vitro evaluation, cytotoxicity assays, molecular modeling and SAR/QSAR studies of a 2-phenyl-3-(1-phenyl-1H-pyrazol-4-yl)-acrylic acid benzylidene-carbohydrazide series
Maria A. F. Vera DiVaio Antônio C. C Freitas; Helena C Castro; Sérgio de Albuquerque; Lucio M Cabral; Carlos Ribeiro Rodrigues; Magaly G Albuquerque; Rita C. A Martins; Maria das Graças M. O Henriques; Luiza R. S Dias
Bioorganic and Medicinal Chemistry Oxford v. 17, n. 1, p. 295-302, 2009
Novel 6-methanesulfonamide-3,4-methylenedioxyphenyl-N-acylhydrazones orally effective anti-inflammatory drug candidates
Jorge L. M. Tributino Carolina D Duarte; Rodrigo S Corrêa; Antonio C Doriguetto; Javier Ellena; Nelilma C Romeiro; Newton G Castro; Ana Luisa P Miranda; Eliezer J Barreiro; Carlos A. M Fraga
Bioorganic and Medicinal Chemistry Oxford v. 17, n. 3, p. 1125-1131, Feb. 2009
Oxford 2009
Localização:
IFSC - Inst. Física de São Carlos
(PROD015694 )(Acessar)
Novel 6-methanesulfonamide-3,4-methylenedioxyphenyl-N-acylhydrazones orally effective anti-inflammatory drug candidates
Jorge L. M. Tributino Carolina D Duarte; Rodrigo S Corrêa; Antonio C Doriguetto; Javier Ellena; Nelilma C Romeiro; Newton G Castro; Ana Luisa P Miranda; Eliezer J Barreiro; Carlos A. M Fraga
Bioorganic and Medicinal Chemistry Oxford v. 17, n. 3, p. 1125-1131, Feb. 2009
Oxford 2009
Localização:
IFSC - Inst. Física de São Carlos
(PROD015694 )(Acessar)
Design, synthesis and stepwise optimization of nitrile-based inhibitors of cathepsins B and L
Lorenzo Cianni Fernanda dos Reis Rocho; Vinícius Bonatto; Felipe Cardoso Prado Martins; Jerônimo Lameira; Andrei Leitão; Carlos Alberto Montanari; Anwar Shamim
Bioorganic and Medicinal Chemistry Oxford : Elsevier v. 29, p. 115827,
Oxford 2021
Localização:
IQSC - Inst. Química de São Carlos
(P19087 )(Acessar)