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Material Type: Artigo
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Structure-activity relationship of a series of diaminoalkyl substituted benzimidazole as neuropeptide Y Y1 receptor antagonistsZarrinmayeh, Hamideh ; Zimmerman, Dennis M. ; Cantrell, Buddy E. ; Schober, Douglas A. ; Bruns, Robert E. ; Gackenheimer, Susan L. ; Ornstein, Paul L. ; Hipskind, Philip A. ; Britton, Thomas C. ; Gehlert, Donald R.Bioorganic & medicinal chemistry letters, 1999-03, Vol.9 (5), p.647-652 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Privileged structure based ligands for melanocortin receptors—4,4-Disubstituted piperidine derivativesKuklish, Steven L. ; Backer, Ryan T. ; Briner, Karin ; Doecke, Christopher W. ; Husain, Saba ; Mullaney, Jeffrey T. ; Ornstein, Paul L. ; Zgombick, John M. ; O’Brien, Thomas P. ; Fisher, Matthew J.Bioorganic & medicinal chemistry letters, 2006-07, Vol.16 (14), p.3843-3846 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Synthesis and structure–activity relationships of novel dipeptides and reduced dipeptides as ligands for melanocortin subtype-4 receptorShi, Qing ; Ornstein, Paul L. ; Briner, Karin ; Richardson, Timothy I. ; Arnold, Macklin B. ; Backer, Ryan T. ; Buckmaster, Jennifer L. ; Canada, Emily J. ; Doecke, Christopher W. ; Hertel, Larry W. ; Honigschmidt, Nick ; Hsiung, Hansen M. ; Husain, Saba ; Kuklish, Steve L. ; Martinelli, Michael J. ; Mullaney, Jeffrey T. ; O’Brien, Thomas P. ; Reinhard, Matt R. ; Rothhaar, Roger ; Shah, Jikesh ; Wu, Zhipei ; Xie, Chaoyu ; Zgombick, John M. ; Fisher, Matthew J.Bioorganic & medicinal chemistry letters, 2006-05, Vol.16 (9), p.2341-2346 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Privileged structure based ligands for melanocortin-4 receptors—Aliphatic piperazine derivativesBriner, Karin ; Collado, Iván ; Fisher, Matthew J. ; García-Paredes, Cristina ; Husain, Saba ; Kuklish, Steven L. ; Mateo, Ana I. ; O’Brien, Thomas P. ; Ornstein, Paul L. ; Zgombick, John ; de Frutos, ÓscarBioorganic & medicinal chemistry letters, 2006-07, Vol.16 (13), p.3449-3453 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |