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Application of Pictet–Spengler Reaction to Indole-Based Alkaloids Containing Tetrahydro-β-carboline Scaffold in Combinatorial Chemistry
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Application of Pictet–Spengler Reaction to Indole-Based Alkaloids Containing Tetrahydro-β-carboline Scaffold in Combinatorial Chemistry

Rao, R. Nishanth ; Maiti, Barnali ; Chanda, Kaushik

ACS combinatorial science, 2017-04, Vol.19 (4), p.199-228 [Periódico revisado por pares]

United States: American Chemical Society

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2
Identification of RAD51–BRCA2 Inhibitors Using N‑Acylhydrazone-Based Dynamic Combinatorial Chemistry
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Artigo
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Identification of RAD51–BRCA2 Inhibitors Using N‑Acylhydrazone-Based Dynamic Combinatorial Chemistry

Bagnolini, Greta ; Balboni, Beatrice ; Schipani, Fabrizio ; Gioia, Dario ; Veronesi, Marina ; De Franco, Francesca ; Kaya, Cansu ; Jumde, Ravindra P. ; Ortega, Jose Antonio ; Girotto, Stefania ; Hirsch, Anna K. H. ; Roberti, Marinella ; Cavalli, Andrea

ACS medicinal chemistry letters, 2022-08, Vol.13 (8), p.1262-1269 [Periódico revisado por pares]

American Chemical Society

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3
Development of Urease Inhibitors by Fragment‐Based Dynamic Combinatorial Chemistry
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Development of Urease Inhibitors by Fragment‐Based Dynamic Combinatorial Chemistry

Wu, Yao ; Zhao, Shuang ; Liu, Changming ; Hu, Lei

ChemMedChem, 2022-10, Vol.17 (19), p.e202200307-n/a [Periódico revisado por pares]

Weinheim: Wiley Subscription Services, Inc

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4
Identification and synthesis of an efficient multivalent E. coli heat labile toxin inhibitor __ A dynamic combinatorial chemistry approach
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Identification and synthesis of an efficient multivalent E. coli heat labile toxin inhibitor __ A dynamic combinatorial chemistry approach

Xu, Jintao ; Zhang, Shixin ; Zhao, Shuang ; Hu, Lei

Bioorganic & medicinal chemistry, 2020-05, Vol.28 (9), p.115436-115436, Article 115436 [Periódico revisado por pares]

England: Elsevier Ltd

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5
Fragment-Based Dynamic Combinatorial Chemistry for Identification of Selective α‑Glucosidase Inhibitors
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Fragment-Based Dynamic Combinatorial Chemistry for Identification of Selective α‑Glucosidase Inhibitors

Wu, Yao ; Liu, Changming ; Hu, Lei

ACS medicinal chemistry letters, 2022-11, Vol.13 (11), p.1791-1796 [Periódico revisado por pares]

American Chemical Society

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6
Identification of HuR–RNA Interfering Compounds by Dynamic Combinatorial Chemistry and Fluorescence Polarization
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Identification of HuR–RNA Interfering Compounds by Dynamic Combinatorial Chemistry and Fluorescence Polarization

Volpe, Serena Della ; Listro, Roberta ; Ambrosio, Francesca Alessandra ; Garbagnoli, Martina ; Linciano, Pasquale ; Rossi, Daniela ; Costa, Giosuè ; Alcaro, Stefano ; Vasile, Francesca ; Hirsch, Anna K. H. ; Collina, Simona

ACS medicinal chemistry letters, 2023-11, Vol.14 (11), p.1509-1516 [Periódico revisado por pares]

American Chemical Society

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7
Dynamic Generation of G‑Quadruplex DNA Ligands by Target-Guided Combinatorial Chemistry on a Magnetic Nanoplatform
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Dynamic Generation of G‑Quadruplex DNA Ligands by Target-Guided Combinatorial Chemistry on a Magnetic Nanoplatform

Jana, Snehasish ; Panda, Deepanjan ; Saha, Puja ; Pantos̨, G. Dan ; Dash, Jyotirmayee

Journal of medicinal chemistry, 2019-01, Vol.62 (2), p.762-773 [Periódico revisado por pares]

United States: American Chemical Society

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8
Discovery of Small-Molecule Stabilizers of 14-3-3 Protein–Protein Interactions via Dynamic Combinatorial Chemistry
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Discovery of Small-Molecule Stabilizers of 14-3-3 Protein–Protein Interactions via Dynamic Combinatorial Chemistry

Hartman, Alwin M ; Elgaher, Walid A. M ; Hertrich, Nathalie ; Andrei, Sebastian A ; Ottmann, Christian ; Hirsch, Anna K. H

ACS medicinal chemistry letters, 2020-05, Vol.11 (5), p.1041-1046 [Periódico revisado por pares]

United States: American Chemical Society

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9
Current Parallel Solid-Phase Synthesis of Drug-like Oxadiazole and Thiadiazole Derivatives for Combinatorial Chemistry
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Current Parallel Solid-Phase Synthesis of Drug-like Oxadiazole and Thiadiazole Derivatives for Combinatorial Chemistry

Abdildinova, Aizhan ; Gong, Young-Dae

ACS combinatorial science, 2018-06, Vol.20 (6), p.309-329 [Periódico revisado por pares]

United States: American Chemical Society

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10
(Chlorosulfonyl)benzenesulfonyl FluoridesVersatile Building Blocks for Combinatorial Chemistry: Design, Synthesis and Evaluation of a Covalent Inhibitor Library
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(Chlorosulfonyl)benzenesulfonyl FluoridesVersatile Building Blocks for Combinatorial Chemistry: Design, Synthesis and Evaluation of a Covalent Inhibitor Library

Tolmachova, Kateryna A ; Moroz, Yurii S ; Konovets, Angelika ; Platonov, Maxim O ; Vasylchenko, Oleksandr V ; Borysko, Petro ; Zozulya, Sergey ; Gryniukova, Anastasia ; Bogolubsky, Andrey V ; Pipko, Sergey ; Mykhailiuk, Pavel K ; Brovarets, Volodymyr S ; Grygorenko, Oleksandr O

ACS combinatorial science, 2018-11, Vol.20 (11), p.672-680 [Periódico revisado por pares]

United States: American Chemical Society

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