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1 |
Material Type: Artigo
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Investigations on the 1-(2-biphenyl)piperazine motif: identification of new potent and selective ligands for the serotonin(7) (5-HT(7)) receptor with agonist or antagonist action in vitro or ex vivoLacivita, Enza ; Patarnello, Daniela ; Stroth, Nikolas ; Caroli, Antonia ; Niso, Mauro ; Contino, Marialessandra ; De Giorgio, Paola ; Di Pilato, Pantaleo ; Colabufo, Nicola A ; Berardi, Francesco ; Perrone, Roberto ; Svenningsson, Per ; Hedlund, Peter B ; Leopoldo, MarcelloJournal of medicinal chemistry, 2012-07, Vol.55 (14), p.6375-6380 [Periódico revisado por pares]United StatesTexto completo disponível |
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Material Type: Artigo
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New σ and 5-HT1A Receptor Ligands: ω-(Tetralin-1-yl)-n-alkylamine DerivativesBerardi, Francesco ; Colabufo, Nicola A ; Giudice, Giuseppe ; Perrone, Roberto ; Tortorella, Vincenzo ; Govoni, Stefano ; Lucchi, LauraJournal of medicinal chemistry, 1996-01, Vol.39 (1), p.176-182 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Structure−Affinity Relationship Study on N -[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamides as Potent and Selective Dopamine D 3 Receptor LigandsLeopoldo, Marcello ; Berardi, Francesco ; Colabufo, Nicola A. ; De Giorgio, Paola ; Lacivita, Enza ; Perrone, Roberto ; Tortorella, VincenzoJournal of medicinal chemistry, 2002-12, Vol.45 (26), p.5727-5735 [Periódico revisado por pares]Texto completo disponível |
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Material Type: Artigo
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First Structure−Activity Relationship Study on Dopamine D 3 Receptor Agents with N -[4-(4-Arylpiperazin-1-yl)butyl]arylcarboxamide StructureLeopoldo, Marcello ; Lacivita, Enza ; Colabufo, Nicola A. ; Contino, Marialessandra ; Berardi, Francesco ; Perrone, RobertoJournal of medicinal chemistry, 2005-12, Vol.48 (25), p.7919-7922 [Periódico revisado por pares]Texto completo disponível |
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Material Type: Artigo
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Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma(1) receptorBerardi, Francesco ; Ferorelli, Savina ; Abate, Carmen ; Pedone, Maria P ; Colabufo, Nicola A ; Contino, Marialessandra ; Perrone, RobertoJournal of medicinal chemistry, 2005-12, Vol.48 (26), p.8237-8244 [Periódico revisado por pares]United StatesTexto completo disponível |
6 |
Material Type: Artigo
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Synthesis and Structure−Affinity Relationships of 1-[ω-(4-Aryl-1-piperazinyl)alkyl]-1-aryl Ketones as 5-HT7 Receptor LigandsPerrone, Roberto ; Berardi, Francesco ; Colabufo, Nicola A ; Lacivita, Enza ; Leopoldo, Marcello ; Tortorella, VincenzoJournal of medicinal chemistry, 2003-02, Vol.46 (4), p.646-649 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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A Structure−Affinity Relationship Study on Derivatives of N -[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide, a High-Affinity and Selective D 4 Receptor LigandPerrone, Roberto ; Berardi, Francesco ; Colabufo, Nicola A. ; Leopoldo, Marcello ; Tortorella, VincenzoJournal of medicinal chemistry, 2000-01, Vol.43 (2), p.270-277 [Periódico revisado por pares]Texto completo disponível |
8 |
Material Type: Artigo
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N -[2-[4-(4-Chlorophenyl)piperazin-1-yl]ethyl]-3-methoxybenzamide: A Potent and Selective Dopamine D 4 LigandPerrone, Roberto ; Berardi, Francesco ; Colabufo, Nicola A. ; Leopoldo, Marcello ; Tortorella, VincenzoJournal of medicinal chemistry, 1998-11, Vol.41 (24), p.4903-4909 [Periódico revisado por pares]Texto completo disponível |
9 |
Material Type: Artigo
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Structure−Activity Relationship Studies on the 5-HT1A Receptor Affinity of 1-Phenyl-4-[ω-(α- or β-tetralinyl)alkyl]piperazines. 4Perrone, Roberto ; Berardi, Francesco ; Colabufo, Nicola A ; Leopoldo, Marcello ; Tortorella, Vincenzo ; Fornaretto, Maria Gioia ; Caccia, Carla ; McArthur, Robert AJournal of medicinal chemistry, 1996-12, Vol.39 (25), p.4928-4934 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
10 |
Material Type: Artigo
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Mixed 5-HT1A/D-2 activity of a new model of arylpiperazines: 1-aryl-4-[3-(1,2-dihydronaphthalen-4-yl)-n-propyl]piperazines. 1. Synthesis and structure-activity relationshipsPerrone, Roberto ; Berardi, Francesco ; Colabufo, Nicola A ; Tortorella, Vincenzo ; Fiorentini, Francesco ; Olgiati, Vincenzo ; Vanotti, Ermes ; Govoni, StefanoJournal of medicinal chemistry, 1994-01, Vol.37 (1), p.99-104 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |