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1
Molecular docking and structure-based drug design strategies
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Molecular docking and structure-based drug design strategies

Ferreira, Leonardo G ; Dos Santos, Ricardo N ; Oliva, Glaucius ; Andricopulo, Adriano D

Molecules, 2015-07, Vol.20 (7), p.13384-13421 [Periódico revisado por pares]

Switzerland: MDPI AG

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2
Antifungal compounds from Streptomyces associated with attine ants also inhibit Leishmania donovani
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Antifungal compounds from Streptomyces associated with attine ants also inhibit Leishmania donovani

Ortega, Humberto E ; Ferreira, Leonardo L G ; Melo, Weilan G P ; Oliveira, Ana Ligia L ; Ramos Alvarenga, René F ; Lopes, Norberto P ; Bugni, Tim S ; Andricopulo, Adriano D ; Pupo, Mônica T Fischer, Katja

PLoS neglected tropical diseases, 2019-08, Vol.13 (8), p.e0007643-e0007643 [Periódico revisado por pares]

United States: Public Library of Science

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3
Identification of natural cytochalasins as leads for neglected tropical diseases drug discovery
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Identification of natural cytochalasins as leads for neglected tropical diseases drug discovery

Valli, Marilia ; Souza, Julia Medeiros ; Chelucci, Rafael Consolin ; Biasetto, Carolina Rabal ; Araujo, Angela Regina ; Bolzani, Vanderlan da Silva ; Andricopulo, Adriano Defini Saha, Bhaskar

PloS one, 2022-10, Vol.17 (10), p.e0275002-e0275002 [Periódico revisado por pares]

San Francisco: Public Library of Science

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4
Discovery of a Series of Acridinones as Mechanism-Based Tubulin Assembly Inhibitors with Anticancer Activity
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Artigo
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Discovery of a Series of Acridinones as Mechanism-Based Tubulin Assembly Inhibitors with Anticancer Activity

Magalhaes, Luma G ; Marques, Fernando B ; da Fonseca, Marina B ; Rogério, Kamilla R ; Graebin, Cedric S ; Andricopulo, Adriano D Lebedeva, Irina V

PloS one, 2016-08, Vol.11 (8), p.e0160842-e0160842 [Periódico revisado por pares]

United States: Public Library of Science

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5
H1-antihistamines as antischistosomal drugs: in vitro and in vivo studies
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Artigo
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H1-antihistamines as antischistosomal drugs: in vitro and in vivo studies

Xavier, Rogério P ; Mengarda, Ana C ; Silva, Marcos P ; Roquini, Daniel B ; Salvadori, Maria C ; Teixeira, Fernanda S ; Pinto, Pedro L ; Morais, Thiago R ; Ferreira, Leonardo L G ; Andricopulo, Adriano D ; de Moraes, Josué

Parasites & vectors, 2020-06, Vol.13 (1), p.278-278, Article 278 [Periódico revisado por pares]

England: BioMed Central Ltd

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6
Structure-Based Virtual Screening, Molecular Dynamics and Binding Free Energy Calculations of Hit Candidates as ALK-5 Inhibitors
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Structure-Based Virtual Screening, Molecular Dynamics and Binding Free Energy Calculations of Hit Candidates as ALK-5 Inhibitors

Araujo, Sheila C ; Maltarollo, Vinicius G ; Almeida, Michell O ; Ferreira, Leonardo L G ; Andricopulo, Adriano D ; Honorio, Kathia M

Molecules (Basel, Switzerland), 2020-01, Vol.25 (2), p.264 [Periódico revisado por pares]

Switzerland: MDPI AG

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7
Identification of a Prenyl Chalcone as a Competitive Lipoxygenase Inhibitor: Screening, Biochemical Evaluation and Molecular Modeling Studies
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Identification of a Prenyl Chalcone as a Competitive Lipoxygenase Inhibitor: Screening, Biochemical Evaluation and Molecular Modeling Studies

Zeraik, Maria Luiza ; Pauli, Ivani ; Dutra, Luiz A ; Cruz, Raquel S ; Valli, Marilia ; Paracatu, Luana C ; de Faria, Carolina M Q G ; Ximenes, Valdecir F ; Regasini, Luis O ; Andricopulo, Adriano D ; Bolzani, Vanderlan S

Molecules (Basel, Switzerland), 2021-04, Vol.26 (8), p.2205 [Periódico revisado por pares]

Switzerland: MDPI AG

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8
Antiplasmodial and trypanocidal activity of violacein and deoxyviolacein produced from synthetic operons
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Artigo
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Antiplasmodial and trypanocidal activity of violacein and deoxyviolacein produced from synthetic operons

Bilsland, Elizabeth ; Tavella, Tatyana A ; Krogh, Renata ; Stokes, Jamie E ; Roberts, Annabelle ; Ajioka, James ; Spring, David R ; Andricopulo, Adriano D ; Costa, Fabio T M ; Oliver, Stephen G

BMC biotechnology, 2018-04, Vol.18 (1), p.22-22, Article 22 [Periódico revisado por pares]

England: BioMed Central Ltd

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9
2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profiling
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Artigo
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2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profiling

Ferreira, Rafael Augusto Alves ; Junior, Celso de Oliveira Rezende ; Martinez, Pablo David Grigol ; Koovits, Paul John ; Soares, Bruna Miranda ; Ferreira, Leonardo L G ; Michelan-Duarte, Simone ; Chelucci, Rafael Consolin ; Andricopulo, Adriano D ; Galuppo, Mariana K ; Uliana, Silvia R B ; Matheeussen, An ; Caljon, Guy ; Maes, Louis ; Campbell, Simon ; Kratz, Jadel M ; Mowbray, Charles E ; Dias, Luiz Carlos Croft, Simon L.

PLoS neglected tropical diseases, 2021-02, Vol.15 (2), p.e0009196 [Periódico revisado por pares]

United States: Public Library of Science

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10
Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum
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Evaluation and discovery of novel benzothiazole derivatives as promising hits against Leishmania infantum

Lapierre, Thibault Joseph William Jacques Dit ; Farago, Danilo Nascimento ; de Moura Lodi Cruz, Mariza Gabriela Faleiro ; de Melo Resende, Daniela ; de Oliveira, Adriane Cristina Rosa ; Dos Santos, Brenda Rosa Macedo ; de Oliveira Souza, Felipe ; Michelan-Duarte, Simone ; Chelucci, Rafael C ; Andricopulo, Adriano D ; Ferreira, Leonardo L G ; Pilau, Eduardo Jorge ; Murta, Silvane Maria Fonseca ; de Oliveira Rezende Júnior, Celso

Chemical biology & drug design, 2024-04, Vol.103 (4), p.e14525-e14525 [Periódico revisado por pares]

England

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