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1
Agelastatin E, Agelastatin F, and Benzosceptrin C from the Marine Sponge Agelas dendromorpha
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Agelastatin E, Agelastatin F, and Benzosceptrin C from the Marine Sponge Agelas dendromorpha

Tilvi, Supriya ; Moriou, Céline ; Martin, Marie-Thérèse ; Gallard, Jean-François ; Sorres, Jonathan ; Patel, Kirti ; Petek, Sylvain ; Debitus, Cécile ; Ermolenko, Ludmila ; Al-Mourabit, Ali

Journal of natural products (Washington, D.C.), 2010-04, Vol.73 (4), p.720-723 [Periódico revisado por pares]

Northbrook, IL: American Chemical Society and American Society of Pharmacognosy

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2
Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success
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Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success

Lovering, Frank ; Bikker, Jack ; Humblet, Christine

Journal of medicinal chemistry, 2009-11, Vol.52 (21), p.6752-6756 [Periódico revisado por pares]

Columbus, OH: American Chemical Society

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3
The Many Roles for Fluorine in Medicinal Chemistry
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The Many Roles for Fluorine in Medicinal Chemistry

Hagmann, William K

Journal of medicinal chemistry, 2008-08, Vol.51 (15), p.4359-4369 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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4
Covalent Modifiers: An Orthogonal Approach to Drug Design
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Covalent Modifiers: An Orthogonal Approach to Drug Design

Potashman, Michele H ; Duggan, Mark E

Journal of medicinal chemistry, 2009-03, Vol.52 (5), p.1231-1246 [Periódico revisado por pares]

Columbus, OH: American Chemical Society

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5
Recent Developments in Fragment-Based Drug Discovery
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Recent Developments in Fragment-Based Drug Discovery

Congreve, Miles ; Chessari, Gianni ; Tisi, Dominic ; Woodhead, Andrew J

Journal of medicinal chemistry, 2008-07, Vol.51 (13), p.3661-3680 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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6
MolDock:  A New Technique for High-Accuracy Molecular Docking
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MolDock:  A New Technique for High-Accuracy Molecular Docking

Thomsen, René ; Christensen, Mikael H

Journal of medicinal chemistry, 2006-06, Vol.49 (11), p.3315-3321 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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7
Discovery of 6α-Ethyl-23(S)-methylcholic Acid (S-EMCA, INT-777) as a Potent and Selective Agonist for the TGR5 Receptor, a Novel Target for Diabesity
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Discovery of 6α-Ethyl-23(S)-methylcholic Acid (S-EMCA, INT-777) as a Potent and Selective Agonist for the TGR5 Receptor, a Novel Target for Diabesity

Pellicciari, Roberto ; Gioiello, Antimo ; Macchiarulo, Antonio ; Thomas, Charles ; Rosatelli, Emiliano ; Natalini, Benedetto ; Sardella, Roccaldo ; Pruzanski, Mark ; Roda, Aldo ; Pastorini, Elisabetta ; Schoonjans, Kristina ; Auwerx, Johan

Journal of medicinal chemistry, 2009-12, Vol.52 (24), p.7958-7961 [Periódico revisado por pares]

Columbus, OH: American Chemical Society

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8
Novel Procedure for Modeling Ligand/Receptor Induced Fit Effects
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Novel Procedure for Modeling Ligand/Receptor Induced Fit Effects

Sherman, Woody ; Day, Tyler ; Jacobson, Matthew P ; Friesner, Richard A ; Farid, Ramy

Journal of medicinal chemistry, 2006-01, Vol.49 (2), p.534-553 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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9
Modern Natural Products Drug Discovery and Its Relevance to Biodiversity Conservation
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Modern Natural Products Drug Discovery and Its Relevance to Biodiversity Conservation

Kingston, David G. I

Journal of natural products (Washington, D.C.), 2011-03, Vol.74 (3), p.496-511 [Periódico revisado por pares]

Northbrook, IL: American Chemical Society and American Society of Pharmacognosy

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10
Extra Precision Glide:  Docking and Scoring Incorporating a Model of Hydrophobic Enclosure for Protein−Ligand Complexes
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Extra Precision Glide:  Docking and Scoring Incorporating a Model of Hydrophobic Enclosure for Protein−Ligand Complexes

Friesner, Richard A ; Murphy, Robert B ; Repasky, Matthew P ; Frye, Leah L ; Greenwood, Jeremy R ; Halgren, Thomas A ; Sanschagrin, Paul C ; Mainz, Daniel T

Journal of medicinal chemistry, 2006-10, Vol.49 (21), p.6177-6196 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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