Result Number | Material Type | Add to My Shelf Action | Record Details and Options |
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1 |
Material Type: Artigo
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Biased agonism: An emerging paradigm in GPCR drug discoveryRankovic, Zoran ; Brust, Tarsis F. ; Bohn, Laura M.Bioorganic & medicinal chemistry letters, 2016-01, Vol.26 (2), p.241-250 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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2 |
Material Type: Artigo
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2′,4′-BNA/LNA aptamers: CE-SELEX using a DNA-based library of full-length 2′-O,4′-C-methylene-bridged/linked bicyclic ribonucleotidesKasahara, Yuuya ; Irisawa, Yuuta ; Ozaki, Hiroaki ; Obika, Satoshi ; Kuwahara, MasayasuBioorganic & medicinal chemistry letters, 2013-03, Vol.23 (5), p.1288-1292 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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3 |
Material Type: Artigo
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Minimum structural requirements for inhibitors of the zinc finger protein TRAF6Radwan, Mohamed O. ; Koga, Ryoko ; Hida, Tomohiro ; Ejima, Tomohiko ; Kanemaru, Yosuke ; Tateishi, Hiroshi ; Okamoto, Yoshinari ; Inoue, Jun-ichiro ; Fujita, Mikako ; Otsuka, MasamiBioorganic & medicinal chemistry letters, 2019-08, Vol.29 (16), p.2162-2167 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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4 |
Material Type: Artigo
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Sulfonamide derivatives as multi-target agents for complex diseasesApaydın, Sinem ; Török, MariannaBioorganic & medicinal chemistry letters, 2019-08, Vol.29 (16), p.2042-2050 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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5 |
Material Type: Artigo
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Proteolysis targeting chimeras (PROTACs) in ‘beyond rule-of-five’ chemical space: Recent progress and future challengesEdmondson, Scott D. ; Yang, Bin ; Fallan, CharleneBioorganic & medicinal chemistry letters, 2019-07, Vol.29 (13), p.1555-1564 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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6 |
Material Type: Artigo
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Pyridones in drug discovery: Recent advancesZhang, Yun ; Pike, AndrewBioorganic & medicinal chemistry letters, 2021-04, Vol.38, p.127849-127849, Article 127849 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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7 |
Material Type: Artigo
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The SARS-CoV-2 main protease as drug targetUllrich, Sven ; Nitsche, ChristophBioorganic & medicinal chemistry letters, 2020-09, Vol.30 (17), p.127377-127377, Article 127377 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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8 |
Material Type: Artigo
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Structural hybridization as a facile approach to new drug candidatesSampath Kumar, Halmuthur M. ; Herrmann, Lars ; Tsogoeva, Svetlana B.Bioorganic & medicinal chemistry letters, 2020-12, Vol.30 (23), p.127514, Article 127514 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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9 |
Material Type: Artigo
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Selective degradation of CDK6 by a palbociclib based PROTACRana, Sandeep ; Bendjennat, Mourad ; Kour, Smit ; King, Hannah M. ; Kizhake, Smitha ; Zahid, Muhammad ; Natarajan, AmarnathBioorganic & medicinal chemistry letters, 2019-06, Vol.29 (11), p.1375-1379 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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10 |
Material Type: Artigo
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A first-in-class clinical G-quadruplex-targeting drug. The bench-to-bedside translation of the fluoroquinolone QQ58 to CX-5461 (Pidnarulex)Xu, Hong ; Hurley, Laurence H.Bioorganic & medicinal chemistry letters, 2022-12, Vol.77, p.129016-129016, Article 129016 [Periódico revisado por pares]Elsevier LtdTexto completo disponível |