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Material Type: Artigo
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Geometrically and Conformationally Restrained Cinnamoyl Compounds as Inhibitors of HIV-1 Integrase: Synthesis, Biological Evaluation, and Molecular ModelingArtico, Marino ; Di Santo, Roberto ; Costi, Roberta ; Novellino, Ettore ; Greco, Giovanni ; Massa, Silvio ; Tramontano, Enzo ; Marongiu, Maria E ; De Montis, Antonella ; La Colla, PaoloJournal of medicinal chemistry, 1998-10, Vol.41 (21), p.3948-3960 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Routes to Covalent Catalysis by Reactive Selection for Nascent Protein NucleophilesReshetnyak, Andrey V ; Armentano, Maria Francesca ; Ponomarenko, Natalia A ; Vizzuso, Domenica ; Durova, Oxana M ; Ziganshin, Rustam ; Serebryakova, Marina ; Govorun, Vadim ; Gololobov, Gennady ; Morse, Herbert C ; Friboulet, Alain ; Makker, Sudesh P ; Gabibov, Alexander G ; Tramontano, AlfonsoJournal of the American Chemical Society, 2007-12, Vol.129 (51), p.16175-16182 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |
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3 |
Material Type: Artigo
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5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones: Novel Potent and Selective Dihydro-alkoxy-benzyl-oxopyrimidine DerivativesMai, Antonello ; Artico, Marino ; Sbardella, Gianluca ; Massa, Silvio ; Novellino, Ettore ; Greco, Giovanni ; Loi, Anna Giulia ; Tramontano, Enzo ; Marongiu, Maria Elena ; La Colla, PaoloJournal of medicinal chemistry, 1999-02, Vol.42 (4), p.619-627 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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4 |
Material Type: Artigo
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Antitumor Agents. 1. Synthesis, Biological Evaluation, and Molecular Modeling of 5H-Pyrido[3,2-a]phenoxazin-5-one, a Compound with Potent Antiproliferative ActivityBolognese, Adele ; Correale, Gaetano ; Manfra, Michele ; Lavecchia, Antonio ; Mazzoni, Orazio ; Novellino, Ettore ; Barone, Vincenzo ; Pani, Alessandra ; Tramontano, Enzo ; La Colla, Paolo ; Murgioni, Chiara ; Serra, Ilaria ; Setzu, Giovanna ; Loddo, RobertaJournal of medicinal chemistry, 2002-11, Vol.45 (24), p.5205-5216 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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5 |
Material Type: Artigo
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A Zinc Binding Site in Viral Serine ProteinasesDe Francesco, Raffaele ; Urbani, Andrea ; Nardi, Maria Chiara ; Tomei, Licia ; Steinkühler, Christian ; Tramontano, AnnaBiochemistry (Easton), 1996-10, Vol.35 (41), p.13282-13287 [Periódico revisado por pares]United States: American Chemical SocietyTexto completo disponível |