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1
Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1H-tetrazol-5-amine P2X(7) antagonists
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Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1H-tetrazol-5-amine P2X(7) antagonists

Perez-Medrano, Arturo ; Donnelly-Roberts, Diana L ; Florjancic, Alan S ; Nelson, Derek W ; Li, Tongmei ; Namovic, Marian T ; Peddi, Sridhar ; Faltynek, Connie R ; Jarvis, Michael F ; Carroll, William A

Bioorganic & medicinal chemistry letters, 2011-06, Vol.21 (11), p.3297-3300 [Periódico revisado por pares]

England

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2
Novel and potent 3-(2,3-dichlorophenyl)-4-(benzyl)-4H-1,2,4-triazole P2X7 antagonists
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Artigo
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Novel and potent 3-(2,3-dichlorophenyl)-4-(benzyl)-4H-1,2,4-triazole P2X7 antagonists

CARROLL, William A ; KALVIN, Douglas M ; PEREZ MEDRANO, Arturo ; FLORJANCIC, Alan S ; YING WANG ; DONNELLY-ROBERTS, Diana L ; NAMOVIC, Marian T ; GRAYSON, George ; HONORE, Prisca ; JARVIS, Michael F

Bioorganic & medicinal chemistry letters, 2007-07, Vol.17 (14), p.4044-4048 [Periódico revisado por pares]

Oxford: Elsevier

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3
Synthesis and in vitro activity of 1-(2,3-dichlorophenyl)-N-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-5-amine and 4-(2,3-dichlorophenyl)-N-(pyridin-3-ylmethyl)-4H-1,2,4-triazol-3-amine P2X7 antagonists
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Artigo
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Synthesis and in vitro activity of 1-(2,3-dichlorophenyl)-N-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-5-amine and 4-(2,3-dichlorophenyl)-N-(pyridin-3-ylmethyl)-4H-1,2,4-triazol-3-amine P2X7 antagonists

Florjancic, Alan S ; Peddi, Sridhar ; Perez-Medrano, Arturo ; Li, Biqin ; Namovic, Marian T ; Grayson, George ; Donnelly-Roberts, Diana L ; Jarvis, Michael F ; Carroll, William A

Bioorganic & medicinal chemistry letters, 2008-03, Vol.18 (6), p.2089-2092 [Periódico revisado por pares]

England

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4
Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1H-tetrazol-5-amine P2X sub(7 antagonists)
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Artigo
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Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1H-tetrazol-5-amine P2X sub(7 antagonists)

Perez-Medrano, Arturo ; Donnelly-Roberts, Diana L ; Florjancic, Alan S ; Nelson, Derek W ; Li, Tongmei ; Namovic, Marian T ; Peddi, Sridhar ; Faltynek, Connie R ; Jarvis, Michael F ; Carroll, William A

Bioorganic & medicinal chemistry letters, 2011-06, Vol.21 (11), p.3297-3300 [Periódico revisado por pares]

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5
Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1H-tetrazol-5-amine P2X₇ antagonists
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Artigo
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Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1H-tetrazol-5-amine P2X₇ antagonists

Perez-Medrano, Arturo ; Donnelly-Roberts, Diana L ; Florjancic, Alan S ; Nelson, Derek W ; Li, Tongmei ; Namovic, Marian T ; Peddi, Sridhar ; Faltynek, Connie R ; Jarvis, Michael F ; Carroll, William A

Bioorganic & medicinal chemistry letters, 2011-06, Vol.21 (11), p.3297-3300 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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6
Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1 H-tetrazol-5-amine P2X 7 antagonists
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Artigo
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Synthesis and in vitro activity of N-benzyl-1-(2,3-dichlorophenyl)-1 H-tetrazol-5-amine P2X 7 antagonists

Perez-Medrano, Arturo ; Donnelly-Roberts, Diana L. ; Florjancic, Alan S. ; Nelson, Derek W. ; Li, Tongmei ; Namovic, Marian T. ; Peddi, Sridhar ; Faltynek, Connie R. ; Jarvis, Michael F. ; Carroll, William A.

Bioorganic & medicinal chemistry letters, 2011, Vol.21 (11), p.3297-3300 [Periódico revisado por pares]

Elsevier Ltd

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7
Synthesis and in vitro activity of 1-(2,3-dichlorophenyl)-N-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-5-amine and 4-(2,3-dichlorophenyl)-N-(pyridin-3-ylmethyl)-4H-l,2,4-triazol-3-amine P2X7 antagonists
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Artigo
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Synthesis and in vitro activity of 1-(2,3-dichlorophenyl)-N-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-5-amine and 4-(2,3-dichlorophenyl)-N-(pyridin-3-ylmethyl)-4H-l,2,4-triazol-3-amine P2X7 antagonists

FLORJANCIC, Alan S ; PEDDI, Sridhar ; PEREZ-MEDRANO, Arturo ; BIQIN LI ; NAMOVIC, Marian T ; GRAYSON, George ; DONNELLY-ROBERTS, Diana L ; JARVIS, Michael F ; CARROLL, William A

Bioorganic & medicinal chemistry letters, 2008, Vol.18 (6), p.2089-2092 [Periódico revisado por pares]

Oxford: Elsevier

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8
Design and synthesis of novel cyanoguanidine ATP-sensitive potassium channel openers for the treatment of overactive bladder
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Artigo
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Design and synthesis of novel cyanoguanidine ATP-sensitive potassium channel openers for the treatment of overactive bladder

Perez-Medrano, Arturo ; Buckner, Steven A. ; Coghlan, Michael J. ; Gregg, Robert J. ; Gopalakrishnan, Murali ; Kort, Michael E. ; Lynch, John K. ; Scott, Victoria E. ; Sullivan, James P. ; Whiteaker, Kristi L. ; Carroll, William A.

Bioorganic & medicinal chemistry letters, 2004-01, Vol.14 (2), p.397-400 [Periódico revisado por pares]

Oxford: Elsevier Ltd

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9
Synthesis, pharmacology and pharmacokinetics of 3-(4-aryl-piperazin-1-ylalkyl)-uracils as uroselective α1A-antagonists
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Artigo
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Synthesis, pharmacology and pharmacokinetics of 3-(4-aryl-piperazin-1-ylalkyl)-uracils as uroselective α1A-antagonists

LOPEZ, F. J ; ARIAS, L ; PADILLA, F ; PEREZ-MEDRANO, A ; QUINTERO, C ; ROMERO, M ; SANDOVAL, L ; SMITH, S. A ; WILLIAMS, T. J ; BLUE, D. R ; CHAN, R ; CLARKE, D. E ; ELWORTHY, T. R ; FORD, A. P. D. W ; GUZMAN, A ; JAIME-FIGUEROA, S ; JASPER, J. R ; MORGANS, D. J

Bioorganic & medicinal chemistry letters, 2003-06, Vol.13 (11), p.1873-1878 [Periódico revisado por pares]

Oxford: Elsevier

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10
Synthesis and in vitro activity of 1-(2,3-dichlorophenyl)- N-(pyridin-3-ylmethyl)-1 H-1,2,4-triazol-5-amine and 4-(2,3-dichlorophenyl)- N-(pyridin-3-ylmethyl)-4 H-1,2,4-triazol-3-amine P2X 7 antagonists
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Artigo
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Synthesis and in vitro activity of 1-(2,3-dichlorophenyl)- N-(pyridin-3-ylmethyl)-1 H-1,2,4-triazol-5-amine and 4-(2,3-dichlorophenyl)- N-(pyridin-3-ylmethyl)-4 H-1,2,4-triazol-3-amine P2X 7 antagonists

Florjancic, Alan S. ; Peddi, Sridhar ; Perez-Medrano, Arturo ; Li, Biqin ; Namovic, Marian T. ; Grayson, George ; Donnelly-Roberts, Diana L. ; Jarvis, Michael F. ; Carroll, William A.

Bioorganic & medicinal chemistry letters, 2008, Vol.18 (6), p.2089-2092 [Periódico revisado por pares]

Elsevier Ltd

Texto completo disponível

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