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Refinado por: Nome da Publicação: Journal Of Medicinal Chemistry remover
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1
1,2,3-Triazoles as Amide Bioisosteres: Discovery of a New Class of Potent HIV‑1 Vif Antagonists
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1,2,3-Triazoles as Amide Bioisosteres: Discovery of a New Class of Potent HIV‑1 Vif Antagonists

Mohammed, Idrees ; Kummetha, Indrasena Reddy ; Singh, Gatikrushna ; Sharova, Natalia ; Lichinchi, Gianluigi ; Dang, Jason ; Stevenson, Mario ; Rana, Tariq M

Journal of medicinal chemistry, 2016-08, Vol.59 (16), p.7677-7682 [Periódico revisado por pares]

United States: American Chemical Society

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2
Vanadium–Flavonoid Complexes: A Promising Class of Molecules for Therapeutic Applications
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Artigo
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Vanadium–Flavonoid Complexes: A Promising Class of Molecules for Therapeutic Applications

Selvaraj, Stalin ; Krishnan, Uma Maheswari

Journal of medicinal chemistry, 2021-09, Vol.64 (17), p.12435-12452 [Periódico revisado por pares]

United States: American Chemical Society

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3
Quantitative Structure–Activity Relationship (QSAR) Study Predicts Small-Molecule Binding to RNA Structure
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Artigo
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Quantitative Structure–Activity Relationship (QSAR) Study Predicts Small-Molecule Binding to RNA Structure

Cai, Zhengguo ; Zafferani, Martina ; Akande, Olanrewaju M. ; Hargrove, Amanda E.

Journal of medicinal chemistry, 2022-05, Vol.65 (10), p.7262-7277 [Periódico revisado por pares]

United States: American Chemical Society

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4
Nitro-Group-Containing Drugs
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Artigo
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Nitro-Group-Containing Drugs

Nepali, Kunal ; Lee, Hsueh-Yun ; Liou, Jing-Ping

Journal of medicinal chemistry, 2019-03, Vol.62 (6), p.2851-2893 [Periódico revisado por pares]

United States: American Chemical Society

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5
Learning Molecular Representations for Medicinal Chemistry
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Artigo
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Learning Molecular Representations for Medicinal Chemistry

Chuang, Kangway V ; Gunsalus, Laura M ; Keiser, Michael J

Journal of medicinal chemistry, 2020-08, Vol.63 (16), p.8705-8722 [Periódico revisado por pares]

United States

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6
Human Neuraminidases: Structures and Stereoselective Inhibitors
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Artigo
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Human Neuraminidases: Structures and Stereoselective Inhibitors

Bourguet, Erika ; Figurska, Sylwia ; Fra̧czek, Manuela Maria

Journal of medicinal chemistry, 2022-02, Vol.65 (4), p.3002-3025 [Periódico revisado por pares]

United States: American Chemical Society

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7
Structure-Activity Relationship Study of the High-Affinity Neuropeptide Y 4 Receptor Positive Allosteric Modulator VU0506013
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Artigo
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Structure-Activity Relationship Study of the High-Affinity Neuropeptide Y 4 Receptor Positive Allosteric Modulator VU0506013

Schüß, Corinna ; Vu, Oanh ; Mishra, Nigam M ; Tough, Iain R ; Du, Yu ; Stichel, Jan ; Cox, Helen M ; Weaver, C David ; Meiler, Jens ; Emmitte, Kyle A ; Beck-Sickinger, Annette G

Journal of medicinal chemistry, 2023-07, Vol.66 (13), p.8745-8766 [Periódico revisado por pares]

United States

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8
Polypharmacology: challenges and opportunities in drug discovery
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Polypharmacology: challenges and opportunities in drug discovery

Anighoro, Andrew ; Bajorath, Jürgen ; Rastelli, Giulio

Journal of medicinal chemistry, 2014-10, Vol.57 (19), p.7874-7887 [Periódico revisado por pares]

United States

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9
An Empirical Quantitative Structure-Activity Relationship Equation Assists the Discovery of High-Affinity Phosphodiesterase 4D Inhibitors as Leads to PET Radioligands
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An Empirical Quantitative Structure-Activity Relationship Equation Assists the Discovery of High-Affinity Phosphodiesterase 4D Inhibitors as Leads to PET Radioligands

Jiang, Meijuan ; Lu, Shuiyu ; Telu, Sanjay ; Pike, Victor W.

Journal of medicinal chemistry, 2023-01, Vol.66 (2), p.1543-1561 [Periódico revisado por pares]

United States: American Chemical Society

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10
Amide Bond Bioisosteres: Strategies, Synthesis, and Successes
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Artigo
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Amide Bond Bioisosteres: Strategies, Synthesis, and Successes

Kumari, Shikha ; Carmona, Angelica V ; Tiwari, Amit K ; Trippier, Paul C

Journal of medicinal chemistry, 2020-11, Vol.63 (21), p.12290-12358 [Periódico revisado por pares]

United States: American Chemical Society

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