Molecular design aided by random forests and synthesis of potent trypanocidal agents as cruzain inhibitors for Chagas disease treatment
Sérgio de Albuquerque Lorenzo Cianni; Daniela de Vita; Carla Duque Lopes; Ana S. M Gomes; Paula Gomes; Charles Laughton; Andrei Leitão; Carlos Alberto Montanari; Raphael Montanari; Jean Francisco Rosa Ribeiro; João Santana da Silva; Cátia Teixeira
Chemical Biology & Drug Design Hoboken: Wiley-Blackwell v. 96, p. 948–960, October 2020
Hoboken 2020
Localização:
FCFRP - Fac. Ciên. Farm. Ribeirão Preto
(pcd 3008255 Acervo Digital ) e outros locais(Acessar)
Heterobimetallic nickel(II) and palladium(II) complexes derived from S-benzyl-N- (ferrocenyl)methylenedithiocarbazate: Trypanocidal activity and interaction with Trypanosoma cruzi Old Yellow Enzyme (TcOYE)
Zumira A Carneiro Ana P S Gaspari; Jackelinne C Lima; Carla D Lopes; Ana P S Gaspari; Sérgio de Albuquerque; Luis R Dinelli; Laudimir Leonardo Walbert Veloso da Silva; Marcella Oliva Paganelli; Silvia Helena Libardi; Victor Marcelo Deflon; Carolina G Oliveira; Ronaldo J Oliveira; Julio Cesar Borges; Pedro I. S Maia
European Journal of Medicinal Chemistry Paris v. 180, p.213-223, 2019
Paris 2019
Localização:
FCFRP - Fac. Ciên. Farm. Ribeirão Preto
(pcd 2952478 Estantes Deslizantes ) e outros locais(Acessar)
Dipeptidyl nitrile derivatives suppress the Trypanosoma cruzi in vitro infection
José Carlos Quilles Junior Anwar Shamim; Daiane Yukie Tezuka; Pedro Henrique Jatai Batista; Carla Duque Lopes; Sérgio de Albuquerque; Carlos Alberto Montanari; Andrei Leitão
Experimental Parasitology San Diego v. 219, art. 108032, dec. 2020
San Diego 2020
Localização:
FCFRP - Fac. Ciên. Farm. Ribeirão Preto
(pcd 3009701 Acervo Digital ) e outros locais(Acessar)
Mapping the S1 and S1’ subsites of cysteine proteases with new dipeptidyl nitrile inhibitors as trypanocidal agents
Lorenzo Cianni Carina Lemke; Erik Gilberg; Christian Feldmann; Fabiana Rosini; Fernanda dos Reis Rocho; Jean Francisco Rosa Ribeiro; Daiane Yukie Tezuka; Carla Duque Lopes; Sérgio de Albuquerque; Jürgen Bajorath; Stefan Laufer Eberhard Karls University Tübingen,, Germany Department of Pharmaceutical/Medicinal Chemistry, Tübingen,; Andrei Leitão Gütschow Michaell; Carlos Alberto Montanari
PLoS Neglected Tropical Diseases San Francisco v. 14, n. 3, art. e0007755, p. 1-36, Mar., 2020
San Francisco 2020
Localização:
FCFRP - Fac. Ciên. Farm. Ribeirão Preto
(pcd 2994422 Acervo Digital ) e outros locais(Acessar)