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The pKBHX Database: Toward a Better Understanding of Hydrogen-Bond Basicity for Medicinal ChemistsLAURENCE, Christian ; BRAMELD, Ken A ; GRATON, Jérôme ; LE QUESTEL, Jean-Yves ; RENAULT, EricJournal of medicinal chemistry, 2009-07, Vol.52 (14), p.4073-4086 [Periódico revisado por pares]Columbus, OH: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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The Many Roles for Fluorine in Medicinal ChemistryHagmann, William KJournal of medicinal chemistry, 2008-08, Vol.51 (15), p.4359-4369 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical SuccessLovering, Frank ; Bikker, Jack ; Humblet, ChristineJournal of medicinal chemistry, 2009-11, Vol.52 (21), p.6752-6756 [Periódico revisado por pares]Columbus, OH: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Designed Multiple Ligands. An Emerging Drug Discovery ParadigmMorphy, Richard ; Rankovic, ZoranJournal of medicinal chemistry, 2005-10, Vol.48 (21), p.6523-6543 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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The Identification of 2-(1H-Indazol-4-yl)-6-(4-methanesulfonyl-piperazin-1-ylmethyl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidine (GDC-0941) as a Potent, Selective, Orally Bioavailable Inhibitor of Class I PI3 Kinase for the Treatment of CancerFolkes, Adrian J ; Ahmadi, Khatereh ; Alderton, Wendy K ; Alix, Sonia ; Baker, Stewart J ; Box, Gary ; Chuckowree, Irina S ; Clarke, Paul A ; Depledge, Paul ; Eccles, Suzanne A ; Friedman, Lori S ; Hayes, Angela ; Hancox, Timothy C ; Kugendradas, Arumugam ; Lensun, Letitia ; Moore, Pauline ; Olivero, Alan G ; Pang, Jodie ; Patel, Sonal ; Pergl-Wilson, Giles H ; Raynaud, Florence I ; Robson, Anthony ; Saghir, Nahid ; Salphati, Laurent ; Sohal, Sukhjit ; Ultsch, Mark H ; Valenti, Melanie ; Wallweber, Heidi J.A ; Wan, Nan Chi ; Wiesmann, Christian ; Workman, Paul ; Zhyvoloup, Alexander ; Zvelebil, Marketa J ; Shuttleworth, Stephen JJournal of medicinal chemistry, 2008-09, Vol.51 (18), p.5522-5532 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Multi-target-Directed Ligands To Combat Neurodegenerative DiseasesCavalli, Andrea ; Bolognesi, Maria Laura ; Minarini, Anna ; Rosini, Michela ; Tumiatti, Vincenzo ; Recanatini, Maurizio ; Melchiorre, CarloJournal of medicinal chemistry, 2008-02, Vol.51 (3), p.347-372 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Physicochemical Properties of Antibacterial Compounds: Implications for Drug DiscoveryO’Shea, Rosemarie ; Moser, Heinz EJournal of medicinal chemistry, 2008-05, Vol.51 (10), p.2871-2878 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Recent Developments in Fragment-Based Drug DiscoveryCongreve, Miles ; Chessari, Gianni ; Tisi, Dominic ; Woodhead, Andrew JJournal of medicinal chemistry, 2008-07, Vol.51 (13), p.3661-3680 [Periódico revisado por pares]Washington, DC: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Covalent Modifiers: An Orthogonal Approach to Drug DesignPotashman, Michele H ; Duggan, Mark EJournal of medicinal chemistry, 2009-03, Vol.52 (5), p.1231-1246 [Periódico revisado por pares]Columbus, OH: American Chemical SocietyTexto completo disponível |
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Material Type: Artigo
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Structure−Activity Relationship of New Anti-Hepatitis C Virus Agents: Heterobicycle−Coumarin ConjugatesNeyts, Johan ; Clercq, Erik De ; Singha, Raghunath ; Chang, Yung Hsiung ; Das, Asish R ; Chakraborty, Subhasish K ; Hong, Shih Ching ; Tsay, Shwu-Chen ; Hsu, Ming-Hua ; Hwu, Jih RuJournal of medicinal chemistry, 2009-03, Vol.52 (5), p.1486-1490 [Periódico revisado por pares]Columbus, OH: American Chemical SocietyTexto completo disponível |