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1
Bicyclic α-Iminophosphonates as High Affinity Imidazoline I 2 Receptor Ligands for Alzheimer's Disease
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Bicyclic α-Iminophosphonates as High Affinity Imidazoline I 2 Receptor Ligands for Alzheimer's Disease

Abás, Sònia ; Rodríguez-Arévalo, Sergio ; Bagán, Andrea ; Griñán-Ferré, Christian ; Vasilopoulou, Foteini ; Brocos-Mosquera, Iria ; Muguruza, Carolina ; Pérez, Belén ; Molins, Elies ; Luque, F Javier ; Pérez-Lozano, Pilar ; de Jonghe, Steven ; Daelemans, Dirk ; Naesens, Lieve ; Brea, José ; Loza, M Isabel ; Hernández-Hernández, Elena ; García-Sevilla, Jesús A ; García-Fuster, M Julia ; Radan, Milica ; Djikic, Teodora ; Nikolic, Katarina ; Pallàs, Mercè ; Callado, Luis F ; Escolano, Carmen

Journal of medicinal chemistry, 2020-04, Vol.63 (7), p.3610-3633 [Periódico revisado por pares]

United States

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2
Bicyclic α‑Iminophosphonates as High Affinity Imidazoline I2 Receptor Ligands for Alzheimer’s Disease
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Artigo
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Bicyclic α‑Iminophosphonates as High Affinity Imidazoline I2 Receptor Ligands for Alzheimer’s Disease

Abás, Sònia ; Rodríguez-Arévalo, Sergio ; Bagán, Andrea ; Griñán-Ferré, Christian ; Vasilopoulou, Foteini ; Brocos-Mosquera, Iria ; Muguruza, Carolina ; Pérez, Belén ; Molins, Elies ; Luque, F. Javier ; Pérez-Lozano, Pilar ; de Jonghe, Steven ; Daelemans, Dirk ; Naesens, Lieve ; Brea, José ; Loza, M. Isabel ; Hernández-Hernández, Elena ; García-Sevilla, Jesús A ; García-Fuster, M. Julia ; Radan, Milica ; Djikic, Teodora ; Nikolic, Katarina ; Pallàs, Mercè ; Callado, Luis F ; Escolano, Carmen

Journal of medicinal chemistry, 2020-04, Vol.63 (7), p.3610-3633 [Periódico revisado por pares]

American Chemical Society

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3
α2‑Adrenoceptor Antagonists: Synthesis, Pharmacological Evaluation, and Molecular Modeling Investigation of Pyridinoguanidine, Pyridino-2-aminoimidazoline and Their Derivatives
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Artigo
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α2‑Adrenoceptor Antagonists: Synthesis, Pharmacological Evaluation, and Molecular Modeling Investigation of Pyridinoguanidine, Pyridino-2-aminoimidazoline and Their Derivatives

Kelly, Brendan ; McMullan, Michela ; Muguruza, Carolina ; Ortega, Jorge E ; Meana, J. Javier ; Callado, Luis F ; Rozas, Isabel

Journal of medicinal chemistry, 2015-01, Vol.58 (2), p.963-977 [Periódico revisado por pares]

United States: American Chemical Society

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4
Guanidine and 2-Aminoimidazoline Aromatic Derivatives as α2-Adrenoceptor Antagonists. 2. Exploring Alkyl Linkers for New Antidepressants
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Guanidine and 2-Aminoimidazoline Aromatic Derivatives as α2-Adrenoceptor Antagonists. 2. Exploring Alkyl Linkers for New Antidepressants

Rodriguez, Fernando ; Rozas, Isabel ; Ortega, Jorge E ; Erdozain, Amaia M ; Meana, J. Javier ; Callado, Luis F

Journal of medicinal chemistry, 2008-06, Vol.51 (11), p.3304-3312 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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5
Guanidine and 2-Aminoimidazoline Aromatic Derivatives as α2-Adrenoceptor Ligands: Searching for Structure−Activity Relationships
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Guanidine and 2-Aminoimidazoline Aromatic Derivatives as α2-Adrenoceptor Ligands: Searching for Structure−Activity Relationships

Rodriguez, Fernando ; Rozas, Isabel ; Ortega, Jorge E ; Erdozain, Amaia M ; Meana, J. Javier ; Callado, Luis F

Journal of medicinal chemistry, 2009-02, Vol.52 (3), p.601-609 [Periódico revisado por pares]

Columbus, OH: American Chemical Society

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6
Guanidine and 2-aminoimidazoline aromatic derivatives as alpha(2)-adrenoceptor antagonists, 1: toward new antidepressants with heteroatomic linkers
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Artigo
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Guanidine and 2-aminoimidazoline aromatic derivatives as alpha(2)-adrenoceptor antagonists, 1: toward new antidepressants with heteroatomic linkers

Rodriguez, Fernando ; Rozas, Isabel ; Ortega, Jorge E ; Meana, J Javier ; Callado, Luis F

Journal of medicinal chemistry, 2007-09, Vol.50 (18), p.4516-4527 [Periódico revisado por pares]

United States

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7
Correction to Bicyclic α-Iminophosphonates as High Affinity Imidazoline I 2 Receptor Ligands for Alzheimer’s Disease
Material Type:
Artigo
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Correction to Bicyclic α-Iminophosphonates as High Affinity Imidazoline I 2 Receptor Ligands for Alzheimer’s Disease

Abás, Sònia ; Rodríguez-Arévalo, Sergio ; Bagán, Andrea ; Griñán-Ferré, Christian ; Vasilopoulou, Foteini ; Brocos-Mosquera, Iria ; Muguruza, Carolina ; Pérez, Belén ; Molins, Elies ; Luque, F. Javier ; Pérez-Lozano, Pilar ; de Jonghe, Steven ; Daelemans, Dirk ; Naesens, Lieve ; Brea, José ; Loza, M. Isabel ; Hernández-Hernández, Elena ; García-Sevilla, Jesús A. ; García-Fuster, M. Julia ; Radan, Milica ; Djikic, Teodora ; Nikolic, Katarina ; Pallàs, Mercè ; Callado, Luis F. ; Escolano, Carmen

Journal of medicinal chemistry, 2020-09, Vol.63 (18), p.10529-10529 [Periódico revisado por pares]

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8
Bicyclic α-Iminophosphonates as High Affinity Imidazoline I2 Receptor Ligands for Alzheimer's Disease
Material Type:
Artigo
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Bicyclic α-Iminophosphonates as High Affinity Imidazoline I2 Receptor Ligands for Alzheimer's Disease

Abas, Sonia ; Rodriguez-Arevalo, Sergio ; Bagan, Andrea ; Grinan-Ferre, Christian ; Vasilopoulou, Foteini ; Brocos-Mosquera, Iria ; Muguruza, Carolina ; Perez, Belen ; Molins, Elies ; Javier Luque, F ; Perez-Lozano, Pilar ; de Jonghe, Steven ; Daelemans, Dirk ; Naesens, Lieve ; Brea, Jose ; Isabel Loza, M ; Hernandez-Hernandez, Elena ; Garcia-Sevilla, Jesus A ; Julia Garcia-Fuster, M ; Radan, Milica ; Djikic, Teodora ; Nikolic, Katarina ; Pallas, Merce ; Callado, Luis F ; Escolano, Carmen

JOURNAL OF MEDICINAL CHEMISTRY, 2020-04, Vol.63 (7), p.3610-3633 [Periódico revisado por pares]

AMER CHEMICAL SOC

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9
Correction to Bicyclic α‑Iminophosphonates as High Affinity Imidazoline I2 Receptor Ligands for Alzheimer’s Disease
Material Type:
Artigo
Adicionar ao Meu Espaço

Correction to Bicyclic α‑Iminophosphonates as High Affinity Imidazoline I2 Receptor Ligands for Alzheimer’s Disease

Abás, Sònia ; Rodríguez-Arévalo, Sergio ; Bagán, Andrea ; Griñán-Ferré, Christian ; Vasilopoulou, Foteini ; Brocos-Mosquera, Iria ; Muguruza, Carolina ; Pérez, Belén ; Molins, Elies ; Luque, F. Javier ; Pérez-Lozano, Pilar ; de Jonghe, Steven ; Daelemans, Dirk ; Naesens, Lieve ; Brea, José ; Loza, M. Isabel ; Hernández-Hernández, Elena ; García-Sevilla, Jesús A ; García-Fuster, M. Julia ; Radan, Milica ; Djikic, Teodora ; Nikolic, Katarina ; Pallàs, Mercè ; Callado, Luis F ; Escolano, Carmen

Journal of medicinal chemistry, 2020-09, Vol.63 (18), p.10529-10529 [Periódico revisado por pares]

American Chemical Society

Texto completo disponível

10
Correction to α2‑Adrenoceptor Antagonists: Synthesis, Pharmacological Evaluation, and Molecular Modeling Investigation of Pyridinoguanidine, Pyridino-2-aminoimidazoline and Their Derivatives
Material Type:
Artigo
Adicionar ao Meu Espaço

Correction to α2‑Adrenoceptor Antagonists: Synthesis, Pharmacological Evaluation, and Molecular Modeling Investigation of Pyridinoguanidine, Pyridino-2-aminoimidazoline and Their Derivatives

Kelly, Brendan ; McMullan, Michela ; Muguruza, Carolina ; Ortega, Jorge E ; Meana, J. Javier ; Callado, Luis F ; Rozas, Isabel

Journal of medicinal chemistry, 2015-04, Vol.58 (8), p.3638-3638 [Periódico revisado por pares]

United States: American Chemical Society

Texto completo disponível

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