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Material Type: Artigo
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Substituted tetraazaacenaphthylenes as potent CRF1 receptor antagonists for the treatment of depression and anxietySt-Denis, Y ; Di Fabio, R ; Bernasconi, G ; Castiglioni, E ; Contini, S ; Donati, D ; Fazzolari, E ; Gentile, G ; Ghirlanda, D ; Marchionni, C ; Messina, F ; Micheli, F ; Pavone, F ; Pasquarello, A ; Sabbatini, F M ; Zampori, M G ; Arban, R ; Vitulli, GBioorganic & medicinal chemistry letters, 2005-08, Vol.15 (16), p.3713-3716 [Periódico revisado por pares]EnglandTexto completo disponível |
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Material Type: Artigo
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Enantiomerically pure tetrahydroquinoline derivatives as in vivo potent antagonists of the glycine binding site associated to the NMDA receptorDI FABIO, Romano ; TRANQUILLINI, Elvira ; DONATI, Daniele ; RATTI, Emiliangelo ; ARBAN, Roberto ; DAL FORNO, Giovanna ; REGGIANI, Angelo ; BARNABY, Robert J ; BERTANI, Barbara ; ALVARO, Giuseppe ; MICHELI, Fabrizio ; SABBATINI, Fabio ; PIZZI, Maria Domenica ; PENTASSUGLIA, Giorgio ; PASQUARELLO, Alessandra ; MESSERI, TommasoBioorganic & medicinal chemistry letters, 2003-11, Vol.13 (21), p.3863-3866 [Periódico revisado por pares]Oxford: ElsevierTexto completo disponível |
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Material Type: Artigo
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Substituted tetraazaacenaphthylenes as potent CRF1 receptor antagonists for the treatment of depression and anxiety: G-protein-coupled receptors in drug discoveryST-DENIS, Y ; DI FABIO, R ; MESSINA, F ; MICHELI, F ; PAVONE, F ; PASQUARELLO, A ; SABBATINI, F. M ; ZAMPORI, M. G ; ARBAN, R ; VITULLI, G ; BERNASCONI, G ; CASTIGLIONI, E ; CONTINI, S ; DONATI, D ; FAZZOLARI, E ; GENTILE, G ; GHIRLANDA, D ; MARCHIONNI, CBioorganic & medicinal chemistry letters, 2005, Vol.15 (16), p.3713-3716 [Periódico revisado por pares]Oxford: ElsevierTexto completo disponível |
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Material Type: Artigo
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From pyrroles to pyrrolo[1,2- a]pyrazinones: A new class of mGluR1 antagonistsMicheli, Fabrizio ; Cavanni, Paolo ; Di Fabio, Romano ; Marchioro, Carla ; Donati, Daniele ; Faedo, Stefania ; Maffeis, Micaela ; Sabbatini, Fabio Maria ; Tranquillini, Maria ElviraBioorganic & medicinal chemistry letters, 2006-03, Vol.16 (5), p.1342-1345 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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2,4-Dicarboxy-pyrroles as selective non-Competitive mGluR1 antagonists: further characterization of 3,5-Dimethyl pyrrole-2,4-dicarboxylic acid 2-propyl ester 4-(1,2,2-Trimethyl-propyl) ester and structure–Activity relationshipsMicheli, Fabrizio ; Di Fabio, Romano ; Bordi, Fabio ; Cavallini, Palmina ; Cavanni, Paolo ; Donati, Daniele ; Faedo, Stefania ; Maffeis, Micaela ; Sabbatini, Fabio Maria ; Tarzia, Giorgio ; Tranquillini, Maria ElviraBioorganic & medicinal chemistry letters, 2003-07, Vol.13 (13), p.2113-2118 [Periódico revisado por pares]England: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Discovery and structure–activity relationship of 2-phenyl-oxazole-4-carboxamide derivatives as potent apoptosis inducersTai, Vincent W.-F. ; Sperandio, David ; Shelton, Emma J. ; Litvak, Joane ; Pararajasingham, Keith ; Cebon, Ben ; Lohman, Julia ; Eksterowicz, John ; Kantak, Seema ; Sabbatini, Peter ; Brown, Cindy ; Zeitz, Jennifer ; Reed, Chris ; Maske, Bill ; Graupe, Doris ; Estevez, Alberto ; Oeh, Jason ; Wong, Darren ; Ni, Yong ; Sprengeler, Paul ; Yee, Robert ; Magill, Catherine ; Neri, Anthony ; Cai, Sui Xiong ; Drewe, John ; Qiu, Ling ; Herich, John ; Tseng, Ben ; Kasibhatla, Shailaja ; Spencer, Jeffrey R.Bioorganic & medicinal chemistry letters, 2006-09, Vol.16 (17), p.4554-4558 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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Substituted tetraazaacenaphthylenes as potent CRF 1 receptor antagonists for the treatment of depression and anxietySt-Denis, Y. ; Fabio, R. Di ; Bernasconi, G. ; Castiglioni, E. ; Contini, S. ; Donati, D. ; Fazzolari, E. ; Gentile, G. ; Ghirlanda, D. ; Marchionni, C. ; Messina, F. ; Micheli, F. ; Pavone, F. ; Pasquarello, A. ; Sabbatini, F.M. ; Zampori, M.G. ; Arban, R. ; Vitulli, G.Bioorganic & medicinal chemistry letters, 2005, Vol.15 (16), p.3713-3716 [Periódico revisado por pares]Elsevier LtdTexto completo disponível |