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Material Type: Artigo
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1-(2-Ethoxyethyl)-1H-pyrazolo[4,3-d]pyrimidines as potent phosphodiesterase 5 (PDE5) inhibitorsTOLLEFSON, Michael B ; ACKER, Brad A ; JACOBSEN, E. J ; HUGHES, Robert O ; WALKER, John K ; FOX, David N. A ; PALMER, Michael J ; FREEMAN, Sandra K ; YING YU ; BOND, Brian RBioorganic & medicinal chemistry letters, 2010-05, Vol.20 (10), p.3120-3124 [Periódico revisado por pares]Amsterdam: ElsevierTexto completo disponível |
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Material Type: Artigo
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1-(4-Aminophenyl)isoquinoline derivatives: Potent inhibitors of calcium-independent and calcium-dependent phosphodiesterases from rat cerebral cortexDavis, Craig W. ; Walker, Kathleen A.Biochemical pharmacology, 1984-04, Vol.33 (8), p.1205-1212 [Periódico revisado por pares]New York, NY: Elsevier IncTexto completo disponível |
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Material Type: Artigo
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14‐Deoxyandrographolide desensitizes hepatocytes to tumour necrosis factor‐alpha‐induced apoptosis through calcium‐dependent tumour necrosis factor receptor superfamily member 1A release via the NO/cGMP pathwayRoy, DN ; Mandal, S ; Sen, G ; Mukhopadhyay, S ; Biswas, TBritish journal of pharmacology, 2010-08, Vol.160 (7), p.1823-1843 [Periódico revisado por pares]Oxford, UK: Blackwell Publishing LtdTexto completo disponível |
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Material Type: Artigo
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1,7- and 2,7-naphthyridine derivatives as potent and highly specific PDE5 inhibitorsUkita, Tatsuzo ; Nakamura, Yoshinori ; Kubo, Akira ; Yamamoto, Yasuo ; Moritani, Yasunori ; Saruta, Kunio ; Higashijima, Takanori ; Kotera, Jun ; Fujishige, Kotomi ; Takagi, Michino ; Kikkawa, Kohei ; Omori, KenjiBioorganic & medicinal chemistry letters, 2003-07, Vol.13 (14), p.2341-2345 [Periódico revisado por pares]Oxford: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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1H-[1, 2, 4]Oxadiazolo[4, 3-a]quinoxalin-1-one(ODQ)Inhibits Cyclic GMP-PKG Pathway-Independent Nonadrenergic, Noncholinergic Relaxation in Longitudinal Muscle of the Rectum of Wistar-ST RatsNakagawa, Masashi ; Takeuchi, Tadayoshi ; Niioka, Satomi ; Yamaji, Michiru ; Okishio, Yutaka ; Nishio, Hideaki ; Hata, FumiakiThe Japanese Journal of Pharmacology, 2000, Vol.82(2), pp.164-167Japan: The Japanese Pharmacological SocietyTexto completo disponível |
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Material Type: Artigo
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2-Aryl- and 2-amido-benzothiazoles as multifunctional vasodilators on rat artery preparationsFusi, Fabio ; Durante, Miriam ; Sgaragli, Giampietro ; Cuong, Nguyen Manh ; Dung, Phan Thi Phuong ; Nam, Nguyen HaiEuropean journal of pharmacology, 2013-08, Vol.714 (1-3), p.178-187 [Periódico revisado por pares]Netherlands: Elsevier B.VTexto completo disponível |
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Material Type: Artigo
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2-Ethylpyrazine Induces Vasodilatation by Releasing Nitric Oxide in the EndotheliumAshigai, Hiroshi ; Ikeshima, Emiko ; Koizumi, Kumiko ; Nakashima, Keiko ; Mizutani, Mai ; Yajima, HiroakiBiological and Pharmaceutical Bulletin, 2017/12/01, Vol.40(12), pp.2153-2157 [Periódico revisado por pares]Japan: The Pharmaceutical Society of JapanTexto completo disponível |
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Material Type: Artigo
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2-Phenylquinazolin-4(3 H)-one, a class of potent PDE5 inhibitors with high selectivity versus PDE6Duan, Hongliang ; Zheng, Jin ; Lai, Qinglin ; Liu, Zheng ; Tian, Guanghui ; Wang, Zhen ; Li, Jianfeng ; Shen, JingshanBioorganic & medicinal chemistry letters, 2009-05, Vol.19 (10), p.2777-2779 [Periódico revisado por pares]Amsterdam: Elsevier LtdTexto completo disponível |
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Material Type: Artigo
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2’,4’‐LNA‐Functionalized 5′‐S‐Phosphorothioester CDNs as STING AgonistsYeboah, Simpa K. ; Zigli, Abdulai ; Sintim, Herman O.Chembiochem : a European journal of chemical biology, 2024-07, Vol.25 (13), p.e202400321-n/a [Periódico revisado por pares]Texto completo disponível |
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Material Type: Artigo
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2′/3′ Regioselectivity of Enzyme‐Free Copying of RNA Detected by NMRMotsch, Sebastian ; Pfeffer, Daniel ; Richert, ClemensChembiochem : a European journal of chemical biology, 2020-07, Vol.21 (14), p.2013-2018 [Periódico revisado por pares]Germany: Wiley Subscription Services, IncTexto completo disponível |