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1 |
Material Type: Artigo
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1-(3-Aminomethyl-4-hydroxyphenyl)-3-pyridinyl-2-propen-1-ones: A novel group of tumour-selective cytotoxinsBilginer, Sinan ; Gul, Halise Inci ; Mete, Ebru ; Das, Umashankar ; Sakagami, Hiroshi ; Umemura, Naoki ; Dimmock, Jonathan RichardJournal of enzyme inhibition and medicinal chemistry, 2013-10, Vol.28 (5), p.974-980 [Periódico revisado por pares]England: Informa HealthcareTexto completo disponível |
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Material Type: Artigo
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1-(3-C-ETHYNYL-β-D-RIBO-PENTOFURANOSYL)CYTOSINE (ECYD, TAS-106)1: ANTITUMOR EFFECT AND MECHANISM OF ACTIONAzuma, Atsushi ; Matsuda, Akira ; Sasaki, Takuma ; Fukushima, MasakazuNucleosides, nucleotides & nucleic acids, 2001-03, Vol.20 (4-7), p.609-619 [Periódico revisado por pares]United States: Taylor & Francis GroupTexto completo disponível |
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Material Type: Artigo
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1‐(5‐Phospho‐β‐d‐Ribosyl)2′‐Phosphoadenosine 5′‐Phosphate Cyclic Anhydride Induced Ca2+ Release in Human T‐Cell LinesGuse, Andreas H. ; Silva, Cristina P. ; Weber, Karin ; Armah, Charlotte N. ; Ashamu, Gloria A. ; Schulze, Christian ; Potter, Barry V. L. ; Mayr, Georg W. ; Hilz, HelmuthEuropean journal of biochemistry, 1997-04, Vol.245 (2), p.411-417 [Periódico revisado por pares]Oxford, UK: Blackwell Science LtdTexto completo disponível |
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Material Type: Artigo
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1,10-Phenanthroline promotes copper complexes into tumor cells and induces apoptosis by inhibiting the proteasome activityZhang, Zhen ; Bi, Caifeng ; Schmitt, Sara M. ; Fan, Yuhua ; Dong, Lili ; Zuo, Jian ; Dou, Q. PingJournal of biological inorganic chemistry, 2012-12, Vol.17 (8), p.1257-1267 [Periódico revisado por pares]Berlin/Heidelberg: Springer-VerlagTexto completo disponível |
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Material Type: Artigo
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1,2-Bis(methylsulfonyl)-1-(2-chloroethyl)-2-[[1-(4-nitrophenyl)ethoxy]carbonyl]hydrazine (KS119): a Cytotoxic Prodrug with Two Stable Conformations Differing in Biological and Physical PropertiesPenketh, Philip G. ; Baumann, Raymond P. ; Shyam, Krishnamurthy ; Williamson, Hugh S. ; Ishiguro, Kimiko ; Zhu, Rui ; Eriksson, Emma S. E. ; Eriksson, Leif A. ; Sartorelli, Alan C.Chemical biology & drug design, 2011-10, Vol.78 (4), p.513-526 [Periódico revisado por pares]Oxford, UK: Blackwell Publishing LtdTexto completo disponível |
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Material Type: Artigo
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1,2-Diaryl-2-hydroxyiminoethanones as Dual COX-1 and β-Amyloid Aggregation Inhibitors: Biological Evaluation and In Silico StudyIrannejad, Hamid ; Unsal Tan, Oya ; Ozadali, Keriman ; Dadashpour, Sakineh ; Tuylu Kucukkilinc, Tuba ; Ahangar, Nematollah ; Ahmadnejad, Mahsa ; Emami, SaeedChemical biology & drug design, 2015-04, Vol.85 (4), p.494-503 [Periódico revisado por pares]England: Blackwell Publishing LtdTexto completo disponível |
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Material Type: Artigo
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1,2-Dimethylimidazole-4-sulfonyl chloride (DMISC), a novel derivatization strategy for the analysis of propofol by LC-ESI-MS/MSMaas, Alexandra ; Maier, Christoph ; Michel-Lauter, Beate ; Madea, Burkhard ; Hess, CorneliusAnalytical and bioanalytical chemistry, 2017-02, Vol.409 (6), p.1547-1554 [Periódico revisado por pares]Berlin/Heidelberg: Springer Berlin HeidelbergTexto completo disponível |
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Material Type: Artigo
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1,2,3,4‐Tetrahydroisoquinolines as inhibitors of HIV‐1 integrase and human LEDGF/p75 interactionGeorge, Anu ; Gopi Krishna Reddy, Alavala ; Satyanarayana, Gedu ; Raghavendra, Nidhanapati KChemical biology & drug design, 2018-06, Vol.91 (6), p.1133-1140 [Periódico revisado por pares]EnglandTexto completo disponível |
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Material Type: Artigo
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1,2,4-thiadiazol-5(4H)-ones: a new class of selective inhibitors of Trypanosoma cruzi triosephosphate isomerase. Study of the mechanism of inhibitionAlvarez, Guzmán ; Aguirre-López, Beatriz ; Cabrera, Nallely ; Marins, Eliã B. ; Tinoco, Luzineide ; Batthyány, Carlos Ignacio ; de Gómez-Puyou, Marieta Tuena ; Puyou, Armando Gómez ; Pérez-Montfort, Ruy ; Cerecetto, Hugo ; González, MercedesJournal of enzyme inhibition and medicinal chemistry, 2013-10, Vol.28 (5), p.981-989 [Periódico revisado por pares]England: Informa HealthcareTexto completo disponível |
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Material Type: Artigo
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1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsyKaproń, Barbara ; Czarnomysy, Robert ; Wysokiński, Mariusz ; Andrys, Rudolf ; Musilek, Kamil ; Angeli, Andrea ; Supuran, Claudiu T. ; Plech, TomaszJournal of enzyme inhibition and medicinal chemistry, 2020-01, Vol.35 (1), p.993-1002 [Periódico revisado por pares]England: Taylor & FrancisTexto completo disponível |