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Refinado por: assunto: Pharmacology & Pharmacy remover
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1
Alzheimer's Disease: A Review from the Pathophysiology to Diagnosis, New Perspectives for Pharmacological Treatment
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Alzheimer's Disease: A Review from the Pathophysiology to Diagnosis, New Perspectives for Pharmacological Treatment

Dos Santos Picanco, Leide Caroline ; Ozela, Priscilla F ; de Fatima de Brito Brito, Maiara ; Pinheiro, Abraao A ; Padilha, Elias C ; Braga, Francinaldo S ; de Paula da Silva, Carlos Henrique Tomich ; Dos Santos, Cleydson Breno Rodrigues ; Rosa, Joaquín M C ; da Silva Hage-Melim, Lorane Izabel

Current medicinal chemistry, 2018-01, Vol.25 (26), p.3141-3159 [Periódico revisado por pares]

United Arab Emirates: Bentham Science Publishers Ltd

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2
Parkinsons Disease: A Review from Pathophysiology to Treatment
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Artigo
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Parkinsons Disease: A Review from Pathophysiology to Treatment

Marino, Bianca L B ; de Souza, Lucilene R ; Sousa, Kessia P A ; Ferreira, Jaderson V ; Padilha, Elias C ; da Silva, Carlos H T P ; Taft, Carlton A ; Hage-Melim, Lorane I S

Mini reviews in medicinal chemistry, 2020-01, Vol.20 (9), p.754-767 [Periódico revisado por pares]

Netherlands: Bentham Science Publishers Ltd

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3
Preclinical Pharmacokinetics and In Vitro Properties of GS-441524, a Potential Oral Drug Candidate for COVID-19 Treatment
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Artigo
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Preclinical Pharmacokinetics and In Vitro Properties of GS-441524, a Potential Oral Drug Candidate for COVID-19 Treatment

Wang, Amy Q. ; Hagen, Natalie R. ; Padilha, Elias C. ; Yang, Mengbi ; Shah, Pranav ; Chen, Catherine Z. ; Huang, Wenwei ; Terse, Pramod ; Sanderson, Philip ; Zheng, Wei ; Xu, Xin

Frontiers in pharmacology, 2022-08, Vol.13 [Periódico revisado por pares]

Frontiers Media S.A

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4
Development and validation of PAMPA-BBB QSAR model to predict brain penetration potential of novel drug candidates
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Artigo
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Development and validation of PAMPA-BBB QSAR model to predict brain penetration potential of novel drug candidates

Kato, Rintaro ; Zeng, Wenyu ; Siramshetty, Vishal B ; Williams, Jordan ; Kabir, Md ; Hagen, Natalie ; Padilha, Elias C ; Wang, Amy Q ; Mathé, Ewy A ; Xu, Xin ; Shah, Pranav

Frontiers in pharmacology, 2023-12, Vol.14, p.1291246-1291246 [Periódico revisado por pares]

Switzerland: Frontiers Media S.A

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5
Use of physiological based pharmacokinetic modeling for cross-species prediction of pharmacokinetic and tissue distribution profiles of a novel niclosamide prodrug
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Artigo
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Use of physiological based pharmacokinetic modeling for cross-species prediction of pharmacokinetic and tissue distribution profiles of a novel niclosamide prodrug

Yang, Mengbi ; Wang, Amy Q ; Padilha, Elias C ; Shah, Pranav ; Hagen, Natalie R ; Ryu, China ; Shamim, Khalida ; Huang, Wenwei ; Xu, Xin

Frontiers in pharmacology, 2023-04, Vol.14, p.1099425-1099425 [Periódico revisado por pares]

Switzerland: Frontiers Media S.A

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6
In vitro and in vivo pharmacokinetic characterization, chiral conversion and PBPK scaling towards human PK simulation of S-MRI-1867, a drug candidate for Hermansky-Pudlak syndrome pulmonary fibrosis
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In vitro and in vivo pharmacokinetic characterization, chiral conversion and PBPK scaling towards human PK simulation of S-MRI-1867, a drug candidate for Hermansky-Pudlak syndrome pulmonary fibrosis

Padilha, Elias C. ; Yang, Mengbi ; Shah, Pranav ; Wang, Amy Q. ; Duan, Jianmin ; Park, Joshua K. ; Zawatsky, Charles N. ; Malicdan, May Christine V. ; Kunos, George ; Iyer, Malliga R. ; Gaucher, Geneviève ; Ravenelle, François ; Cinar, Resat ; Xu, Xin

Biomedicine & pharmacotherapy, 2023-12, Vol.168, p.115178-115178, Article 115178 [Periódico revisado por pares]

France: Elsevier Masson SAS

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7
The presence of doping agents in dietary supplements: A glimpse into the Brazilian situation
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The presence of doping agents in dietary supplements: A glimpse into the Brazilian situation

Torres, Clarisse L. ; Oliveira, Felipe A. G. ; Jooris, Luis Felipe ; Padilha, Monica C. ; Pereira, Henrique M. G.

Drug testing and analysis, 2024-01, Vol.16 (1), p.38-48 [Periódico revisado por pares]

England: Wiley Subscription Services, Inc

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8
Identification of Selective CYP3A7 and CYP3A4 Substrates and Inhibitors Using a High-Throughput Screening Platform
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Artigo
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Identification of Selective CYP3A7 and CYP3A4 Substrates and Inhibitors Using a High-Throughput Screening Platform

Kabir, Md ; Padilha, Elias C. ; Shah, Pranav ; Huang, Ruili ; Sakamuru, Srilatha ; Gonzalez, Eric ; Ye, Lin ; Hu, Xin ; Henderson, Mark J. ; Xia, Menghang ; Xu, Xin

Frontiers in pharmacology, 2022-07, Vol.13, p.899536-899536 [Periódico revisado por pares]

Frontiers Media S.A

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9
Application of in vitro Drug Metabolism Studies in Chemical Structure Optimization for the Treatment of Fibrodysplasia Ossificans Progressiva (FOP)
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Application of in vitro Drug Metabolism Studies in Chemical Structure Optimization for the Treatment of Fibrodysplasia Ossificans Progressiva (FOP)

Padilha, Elias C ; Wang, Jianyao ; Kerns, Ed ; Lee, Arthur ; Huang, Wenwei ; Jiang, Jian-Kang ; McKew, John ; Mutlib, Abdul ; Peccinini, Rosangela G ; Yu, Paul B ; Sanderson, Philip ; Xu, Xin

Frontiers in pharmacology, 2019-04, Vol.10, p.234-234 [Periódico revisado por pares]

Switzerland: Frontiers Media S.A

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10
Design, Synthesis, and Biological Evaluation of Quinazolin-4-one-Based Hydroxamic Acids as Dual PI3K/HDAC Inhibitors
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Artigo
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Design, Synthesis, and Biological Evaluation of Quinazolin-4-one-Based Hydroxamic Acids as Dual PI3K/HDAC Inhibitors

Thakur, Ashish ; Tawa, Gregory J ; Henderson, Mark J ; Danchik, Carina ; Liu, Suiyang ; Shah, Pranav ; Wang, Amy Q ; Dunn, Garrett ; Kabir, Md ; Padilha, Elias C ; Xu, Xin ; Simeonov, Anton ; Kharbanda, Surender ; Stone, Richard ; Grewal, Gurmit

Journal of medicinal chemistry, 2020-04, Vol.63 (8), p.4256-4292 [Periódico revisado por pares]

United States: American Chemical Society

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