Result Number | Material Type | Add to My Shelf Action | Record Details and Options |
---|---|---|---|
1 |
Material Type: Artigo
|
![]() |
Evaluating anticancer activity of emodin by enhancing antioxidant activities and affecting PKC/ADAMTS4 pathway in thioacetamide-induced hepatocellular carcinoma in ratsHassan, Hanan M. ; Hamdan, Ahmed M. ; Alattar, Abdullah ; Alshaman, Reem ; Bahattab, Omar ; Al-Gayyar, Mohammed M. H.Redox report : communications in free radical research, 2024-12, Vol.29 (1), p.2365590 [Periódico revisado por pares]Taylor & FrancisTexto completo disponível |
2 |
Material Type: Artigo
|
![]() |
Development of a multi-targeted chemotherapeutic approach based on G-quadruplex stabilisation and carbonic anhydrase inhibitionNocentini, Alessio ; Di Porzio, Anna ; Bonardi, Alessandro ; Bazzicalupi, Carla ; Petreni, Andrea ; Biver, Tarita ; Bua, Silvia ; Marzano, Simona ; Amato, Jussara ; Pagano, Bruno ; Iaccarino, Nunzia ; De Tito, Stefano ; Amente, Stefano ; Supuran, Claudiu T. ; Randazzo, Antonio ; Gratteri, PaolaJournal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2366236 [Periódico revisado por pares]Taylor & FrancisTexto completo disponível |
3 |
Material Type: Artigo
|
![]() |
Watermelon: setup and validation of an in silico fragment-based approachDi Stefano, Miriana ; Galati, Salvatore ; Piazza, Lisa ; Gado, Francesca ; Granchi, Carlotta ; Macchia, Marco ; Giordano, Antonio ; Tuccinardi, Tiziano ; Poli, GiulioJournal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2356179 [Periódico revisado por pares]Taylor & FrancisTexto completo disponível |
4 |
Material Type: Artigo
|
![]() |
Effects of thymoquinone and the curcumin analog EF-24 on the activity of the enzyme paraoxonase-1 in human glioblastoma cells U87MGSimsek, Ender ; Sunguroglu, Asuman ; Kilic, Ahmet ; Özgültekin, Nurbanu ; Ozensoy Guler, O.Journal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2339901 [Periódico revisado por pares]Taylor & FrancisTexto completo disponível |
5 |
Material Type: Artigo
|
![]() |
Cloning, expression, and purification of an α-carbonic anhydrase from Toxoplasma gondii to unveil its kinetic parameters and anion inhibition profileDe Luca, Viviana ; Giovannuzzi, Simone ; Capasso, Clemente ; Supuran, Claudiu T.Journal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2346523-2346523 [Periódico revisado por pares]Taylor & FrancisTexto completo disponível |
6 |
Material Type: Artigo
|
![]() |
Exploring of N-phthalimide-linked 1,2,3-triazole analogues with promising anti-SARS-CoV-2 activity: synthesis, biological screening, and molecular modelling studiesAljuhani, Ateyatallah ; Alsehli, Mosa ; Seleem, Mohamed A. ; Alraqa, Shaya Y. ; Ahmed, Hany E. A. ; Rezki, Nadjet ; Aouad, Mohamed R.Journal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2351861-2351861 [Periódico revisado por pares]Taylor & FrancisTexto completo disponível |
7 |
Material Type: Artigo
|
![]() |
Click estradiol dimers with novel aromatic bridging units: synthesis and anticancer evaluationŘehulka, Jiří ; Jurášek, Michal ; Dráber, Pavel ; Ivanová, Aleksandra ; Gurská, Soňa ; Ječmeňová, Kateřina ; Mokshyna, Olena ; Hajdúch, Marián ; Polishchuk, Pavel ; Drašar, Pavel B. ; Džubák, PetrJournal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2367139 [Periódico revisado por pares]Taylor & Francis GroupTexto completo disponível |
8 |
Material Type: Artigo
|
![]() |
New natural protein tyrosine phosphatase 1B inhibitors from Gynostemma pentaphyllumWang, Xianting ; Deng, Yidan ; Wang, Jianmei ; Qin, Lin ; Du, Yimei ; Zhang, Qianru ; Wu, Di ; Wu, Xingdong ; Xie, Jian ; He, Yuqi ; Tan, DaopengJournal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2360063 [Periódico revisado por pares]Taylor & FrancisTexto completo disponível |
9 |
Material Type: Artigo
|
![]() |
Identification of novel PD-1/PD-L1 small molecule inhibitors: virtual screening, synthesis and in vitro characterisationWu, Tingting ; Cheng, Hu ; Sima, Lijie ; Wang, Zhongyuan ; Ouyang, Weiwei ; Wang, Jianta ; Hou, Yunlei ; Zhao, Dongsheng ; Liao, Weike ; Hu, ChujiaoJournal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2353711 [Periódico revisado por pares]Taylor & FrancisTexto completo disponível |
10 |
Material Type: Artigo
|
![]() |
Novel NO-TZDs and trimethoxychalcone-based DHPMs: design, synthesis, and biological evaluation as potential VEGFR-2 inhibitorsMahnashi, Mater H. ; Nahari, Mohammed ; Almasoudi, Hassan ; Alhasaniah, Abdulaziz ; Elgazwi, Sara ; Abou-Salim, Mahrous A.Journal of enzyme inhibition and medicinal chemistry, 2024-12, Vol.39 (1), p.2358934 [Periódico revisado por pares]Taylor & Francis GroupTexto completo disponível |