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Material Type: Artigo
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2-aminobenzimidazoles for leishmaniasis: From initial hit discovery to in vivo profilingFerreira, Rafael Augusto Alves ; Junior, Celso de Oliveira Rezende ; Martinez, Pablo David Grigol ; Koovits, Paul John ; Soares, Bruna Miranda ; Ferreira, Leonardo L G ; Michelan-Duarte, Simone ; Chelucci, Rafael Consolin ; Andricopulo, Adriano D ; Galuppo, Mariana K ; Uliana, Silvia R B ; Matheeussen, An ; Caljon, Guy ; Maes, Louis ; Campbell, Simon ; Kratz, Jadel M ; Mowbray, Charles E ; Dias, Luiz Carlos Croft, Simon L.PLoS neglected tropical diseases, 2021-02, Vol.15 (2), p.e0009196 [Periódico revisado por pares]United States: Public Library of ScienceTexto completo disponível |
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Material Type: Artigo
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AI is a viable alternative to high throughput screening: a 318-target studyBernard, Denzil ; Morrison, Adrian ; Ng, Ho Leung ; Ahmed, Mostafa ; Anthis, Nicholas J. ; PrasadPrasad, Srimukh Veccham Krishna ; Shek, Stefani ; Lee, Andreia H. ; DeHaan, Nicholas ; Abramyan, Tigran M. ; Ghosh, Agnidipta ; Statsyuk, Alexander V. ; Caflisch, Amedeo ; Matheeussen, An ; Battistoni, Andrea ; Chini, Andrea ; Ilari, Andrea ; Foote, Andrea Talbot ; Samantha, Ariela ; ElSheikh, Assmaa ; Edelman, Benjamin L. ; Morten, Brianna C. ; Lempicki, Camille ; Chapman, Carly J. ; Partch, Carrie L. ; Huang, Chang ; Hu, Di ; Ortiz, Diana ; Dirksen, Dorian ; Lama, Eleonora ; Christensen, Emily M. ; Trakhtenberg, Ephraim F. ; Kroon, Erna Geessien ; Yu, Fang ; van den Akker, Focco ; Vizeacoumar, Franco J. ; Vizeacoumar, Frederick S. ; Mayer, Gaétan ; Girolimetti, Giulia ; Dahal, Gopal ; Bowman, Gregory R. ; Akk, Gustav ; Jafar-Nejad, Hamed ; Jung, Hoyoung ; Fan, Hua-Ying ; Arozarena, Imanol ; Ferreira, Jacob ; Siqueira-Neto, Jair L. ; Evans, Jay D. ; Wang, Jianghai ; So, Jonathan ; Gruber, Joshua J. ; Lasarte, Juan José ; Lescar, Julien ; Bogomolovas, Julijus ; Sistla, Jyothi C. ; Hopkins, Kevin M. ; Mostert, Konrad J. ; Rohde, Kyle H. ; Pusztai, Lajos ; Cowen, Leah E. ; Su, Leila ; Wert-Lamas, Leon ; Puchades-Carrasco, Leonor ; Zhuo, Ling ; Valli, Marilia ; Tye, Mark A. ; Wilson, Mark A. ; Alteen, Matthew G. ; Rizzi, Menico ; Paige, Mikell ; Matovic, Nick ; Horstmann, Nicola ; Khalaf, Noureddine Ben ; Sobrado, Pablo ; Chuong, Patrick ; Wu, Pengpeng ; Agogo-Mawuli, Percy ; Toogood, Peter ; von Hundelshausen, Philipp ; Lee, Pil H. ; Balaña-Fouce, Rafael ; Singh, Rakesh K. ; Tiwari, Rakesh Kumar ; Austin, Richard C. ; Bradley, Robert K. ; Reguera, Rosa Maria ; Uribe, Ruben Vazquez ; Gorgoglione, Ruggiero ; Geden, Sandra E. ; Chauhan, Shefali ; Shyng, Show-Ling ; Xu, Sophia Q. ; Gustincich, Stefano ; Marx, Steven O. ; Banerji, Versha ; Robinson, Victoria L. ; Gunasekharan, Vignesh ; Van Hung Le, Vuong ; Wu, XiaoyangScientific reports, 2024-04, Vol.14 (1), p.7526-16, Article 7526 [Periódico revisado por pares]England: Nature Publishing GroupTexto completo disponível |
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Material Type: Artigo
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Antifungal compounds from Streptomyces associated with attine ants also inhibit Leishmania donovaniOrtega, Humberto E ; Ferreira, Leonardo L G ; Melo, Weilan G P ; Oliveira, Ana Ligia L ; Ramos Alvarenga, René F ; Lopes, Norberto P ; Bugni, Tim S ; Andricopulo, Adriano D ; Pupo, Mônica T Fischer, KatjaPLoS neglected tropical diseases, 2019-08, Vol.13 (8), p.e0007643-e0007643 [Periódico revisado por pares]United States: Public Library of ScienceTexto completo disponível |
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Material Type: Artigo
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Antimicrobial Activity of an Fmoc-Plantaricin 149 Derivative Peptide against Multidrug-Resistant BacteriaRighetto, Gabriela Marinho ; Lopes, José Luiz de Souza ; Bispo, Paulo José Martins ; André, Camille ; Souza, Julia Medeiros ; Andricopulo, Adriano Defini ; Beltramini, Leila Maria ; Camargo, Ilana Lopes Baratella da CunhaAntibiotics (Basel), 2023-02, Vol.12 (2), p.391 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
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Material Type: Artigo
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Antioxidant Activity, Molecular Docking, Quantum Studies and In Vivo Antinociceptive Activity of Sulfonamides Derived From Carvacrolde Oliveira, Aldo S. ; Llanes, Luana C. ; Nunes, Ricardo J. ; Nucci-Martins, Catharina ; de Souza, Anacleto S. ; Palomino-Salcedo, David L. ; Dávila-Rodríguez, María J. ; Ferreira, Leonardo L. G. ; Santos, Adair R. S. ; Andricopulo, Adriano D.Frontiers in pharmacology, 2021-11, Vol.12, p.788850-788850 [Periódico revisado por pares]Frontiers Media S.ATexto completo disponível |
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Material Type: Artigo
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Antiplasmodial and trypanocidal activity of violacein and deoxyviolacein produced from synthetic operonsBilsland, Elizabeth ; Tavella, Tatyana A ; Krogh, Renata ; Stokes, Jamie E ; Roberts, Annabelle ; Ajioka, James ; Spring, David R ; Andricopulo, Adriano D ; Costa, Fabio T M ; Oliver, Stephen GBMC biotechnology, 2018-04, Vol.18 (1), p.22-22, Article 22 [Periódico revisado por pares]England: BioMed Central LtdTexto completo disponível |
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Material Type: Artigo
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Chemoinformatics Strategies for Leishmaniasis Drug DiscoveryFerreira, Leonardo L G ; Andricopulo, Adriano DFrontiers in pharmacology, 2018-11, Vol.9, p.1278-1278 [Periódico revisado por pares]Switzerland: Frontiers Research FoundationTexto completo disponível |
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Material Type: Artigo
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Chemoinformatics Studies on a Series of Imidazoles as Cruzain InhibitorsMedeiros, Alex R ; Ferreira, Leonardo L G ; de Souza, Mariana L ; de Oliveira Rezende Junior, Celso ; Espinoza-Chávez, Rocío Marisol ; Dias, Luiz Carlos ; Andricopulo, Adriano DBiomolecules (Basel, Switzerland), 2021-04, Vol.11 (4), p.579 [Periódico revisado por pares]Switzerland: MDPI AGTexto completo disponível |
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Material Type: Artigo
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Dimeric interactions and complex formation using direct coevolutionary couplingsdos Santos, Ricardo N ; Morcos, Faruck ; Jana, Biman ; Andricopulo, Adriano D ; Onuchic, José NScientific reports, 2015-09, Vol.5 (1), p.13652-13652, Article 13652 [Periódico revisado por pares]England: Nature Publishing GroupTexto completo disponível |
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Material Type: Artigo
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Discovery of a Series of Acridinones as Mechanism-Based Tubulin Assembly Inhibitors with Anticancer ActivityMagalhaes, Luma G ; Marques, Fernando B ; da Fonseca, Marina B ; Rogério, Kamilla R ; Graebin, Cedric S ; Andricopulo, Adriano D Lebedeva, Irina VPloS one, 2016-08, Vol.11 (8), p.e0160842-e0160842 [Periódico revisado por pares]United States: Public Library of ScienceTexto completo disponível |