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1 |
Material Type: Artigo
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A pharmacophore-based virtual screening approach for the discovery of Trypanosoma cruzi GAPDH inhibitorsMaluf, Fernando V ; Andricopulo, Adriano D ; Oliva, Glaucius ; Guido, Rafael VcFuture medicinal chemistry, 2013-11, Vol.5 (17), p.2019-2035 [Periódico revisado por pares]EnglandTexto completo disponível |
2 |
Material Type: Artigo
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Benzimidazole inhibitors of the major cysteine protease of Trypanosoma bruceiPereira, Glaécia An ; Santos, Lucianna H ; Wang, Steven C ; Martins, Luan C ; Villela, Filipe S ; Liao, Weiting ; Dessoy, Marco A ; Dias, Luiz C ; Andricopulo, Adriano D ; Costa, Mariana Af ; Nagem, Ronaldo Ap ; Caffrey, Conor R ; Liedl, Klaus R ; Caffarena, Ernesto R ; Ferreira, Rafaela SFuture medicinal chemistry, 2019-07, Vol.11 (13), p.1537-1551 [Periódico revisado por pares]England: Newlands PressTexto completo disponível |
3 |
Material Type: Artigo
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Diaminomaleonitrile derivatives as new potential antichagasic compounds: a study of structure–activity relationshipsde Oliveira, Aldo S ; S Mello, Lucas Dos ; H Ogihara, Camila ; H Döring, Thiago ; L Palomino-Salcedo, David ; Michelan-Duarte, Simone ; Lg Ferreira, Leonardo ; M Souza, Julia ; Dávila-Rodríguez, María José ; Cruz Júnior, José W da ; R Dockal, Edward ; D Andricopulo, AdrianoFuture medicinal chemistry, 2021-12, Vol.13 (24), p.2167-2183 [Periódico revisado por pares]England: Newlands Press LtdTexto completo disponível |
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Material Type: Artigo
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Empowering neglected tropical disease drug discovery with translational medicinal chemistryFerreira, Leonardo Lg ; Andricopulo, Adriano DFuture medicinal chemistry, 2023-06, Vol.15 (12), p.1015-1017 [Periódico revisado por pares]England: Newlands Press LtdTexto completo disponível |
5 |
Material Type: Artigo
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From chemoinformatics to deep learning: an open road to drug discoveryFerreira, Leonardo LG ; Andricopulo, Adriano DFuture medicinal chemistry, 2019-03, Vol.11 (5), p.371-374 [Periódico revisado por pares]England: Future Science LtdTexto completo disponível |
6 |
Material Type: Artigo
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Inhibitors of Trypanosoma brucei trypanothione reductase: comparative molecular field analysis modeling and structural basis for selective inhibitionFerreira, Leonardo G ; Andricopulo, Adriano DFuture medicinal chemistry, 2013-10, Vol.5 (15), p.1753-1762 [Periódico revisado por pares]EnglandTexto completo disponível |
7 |
Material Type: Artigo
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Molecular modeling and structure-activity relationships for a series of benzimidazole derivatives as cruzain inhibitorsPauli, Ivani ; Ferreira, Leonardo G ; de Souza, Mariana L ; Oliva, Glaucius ; Ferreira, Rafaela S ; Dessoy, Marco A ; Slafer, Brian W ; Dias, Luiz C ; Andricopulo, Adriano DFuture medicinal chemistry, 2017-05, Vol.9 (7), p.641-657 [Periódico revisado por pares]England: Future Science LtdTexto completo disponível |
8 |
Material Type: Artigo
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Novel trypanocidal thiophen-chalcone cruzain inhibitors: structure- and ligand-based studiesde Oliveira, Aldo S ; Valli, Marilia ; Ferreira, Leonardo Lg ; Souza, Julia M ; Krogh, Renata ; Meier, Lidiane ; Abreu, Heitor R ; Voltolini, Bruna G ; Llanes, Luana C ; Nunes, Ricardo J ; Braga, Antonio L ; Andricopulo, Adriano DFuture medicinal chemistry, 2022-06, Vol.14 (11), p.795-808 [Periódico revisado por pares]England: Newlands Press LtdTexto completo disponível |
9 |
Material Type: Artigo
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Quantitative structure-activity relationships for a series of selective estrogen receptor-beta modulatorsSalum, L. B. ; Polikarpov, I. ; Andricopulo, A. D.SAR and QSAR in environmental research, 2007-10, Vol.18 (7-8), p.711-727 [Periódico revisado por pares]England: Taylor & Francis GroupTexto completo disponível |
10 |
Material Type: Artigo
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Structure-activity relationships for a class of selective inhibitors of the major cysteine protease from Trypanosoma cruziGuido, Rafael V. C. ; Trossini, Gustavo H. G. ; Castilho, Marcelo S. ; Oliva, Glaucius ; Ferreira, Elizabeth I. ; Andricopulo, Adriano D.Journal of enzyme inhibition and medicinal chemistry, 2008-01, Vol.23 (6), p.964-973 [Periódico revisado por pares]England: Informa UK LtdTexto completo disponível |