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1
1-(1H-Indol-3-yl)ethanamine Derivatives as Potent Staphylococcus aureus NorA Efflux Pump Inhibitors
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1-(1H-Indol-3-yl)ethanamine Derivatives as Potent Staphylococcus aureus NorA Efflux Pump Inhibitors

Hequet, Arnaud ; Burchak, Olga N. ; Jeanty, Matthieu ; Guinchard, Xavier ; Le Pihive, Emmanuelle ; Maigre, Laure ; Bouhours, Pascale ; Schneider, Dominique ; Maurin, Max ; Paris, Jean-Marc ; Denis, Jean-Noël ; Jolivalt, Claude

ChemMedChem, 2014-07, Vol.9 (7), p.1534-1545 [Periódico revisado por pares]

Weinheim: WILEY-VCH Verlag

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2
1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector Anopheles arabiensis and In Silico Molecular Docking Study
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1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector Anopheles arabiensis and In Silico Molecular Docking Study

Venugopala, Katharigatta N ; Shinu, Pottathil ; Tratrat, Christophe ; Deb, Pran Kishore ; Gleiser, Raquel M ; Chandrashekharappa, Sandeep ; Chopra, Deepak ; Attimarad, Mahesh ; Nair, Anroop B ; Sreeharsha, Nagaraja ; Mahomoodally, Fawzi M ; Haroun, Michelyne ; Kandeel, Mahmoud ; Asdaq, Syed Mohammed Basheeruddin ; Mohanlall, Viresh ; Al-Shar'i, Nizar A ; Morsy, Mohamed A

Molecules (Basel, Switzerland), 2022-04, Vol.27 (9), p.2676 [Periódico revisado por pares]

Switzerland: MDPI AG

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3
1,2,4‐Triazole and benzimidazole fused dihydropyrimidine derivatives: Design, green synthesis, antibacterial, antitubercular, and antimalarial activities
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1,2,4‐Triazole and benzimidazole fused dihydropyrimidine derivatives: Design, green synthesis, antibacterial, antitubercular, and antimalarial activities

Mokariya, Jaydeep A. ; Rajani, Dhanji P. ; Patel, Manish P.

Archiv der Pharmazie (Weinheim), 2023-04, Vol.356 (4), p.e2200545-n/a [Periódico revisado por pares]

Germany: Wiley Subscription Services, Inc

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4
1,2,4‐trihydroxynaphthalene‐2‐O‐β‐D‐glucopyranoside delays amyloid‐β42 aggregation and reduces amyloid cytotoxicity
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Artigo
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1,2,4‐trihydroxynaphthalene‐2‐O‐β‐D‐glucopyranoside delays amyloid‐β42 aggregation and reduces amyloid cytotoxicity

Dhouafli, Zohra ; Leri, Manuela ; Bucciantini, Monica ; Stefani, Massimo ; Gadhoumi, Hamza ; Mahjoub, Borhane ; Ben Jannet, Hichem ; Guillard, Jérôme ; Ksouri, Riadh ; Saidani Tounsi, Moufida ; Soto, Claudio ; Hayouni, El Akrem

BioFactors (Oxford), 2018-05, Vol.44 (3), p.272-280 [Periódico revisado por pares]

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5
1,2,4-Trimethoxybenzene selectively inhibits NLRP3 inflammasome activation and attenuates experimental autoimmune encephalomyelitis
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1,2,4-Trimethoxybenzene selectively inhibits NLRP3 inflammasome activation and attenuates experimental autoimmune encephalomyelitis

Pan, Rui-Yuan ; Kong, Xiang-Xi ; Cheng, Yong ; Du, Lu ; Wang, Zhen-Chao ; Yuan, Chao ; Cheng, Jin-Bo ; Yuan, Zeng-Qiang ; Zhang, Hai-Yan ; Liao, Ya-Jin

Acta pharmacologica Sinica, 2021-11, Vol.42 (11), p.1769-1779 [Periódico revisado por pares]

United States: Nature Publishing Group

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6
1,2,4,5-Tetrazine-tethered probes for fluorogenically imaging superoxide in live cells with ultrahigh specificity
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1,2,4,5-Tetrazine-tethered probes for fluorogenically imaging superoxide in live cells with ultrahigh specificity

Jiang, Xuefeng ; Li, Min ; Wang, Yule ; Wang, Chao ; Wang, Yingchao ; Shen, Tianruo ; Shen, Lili ; Liu, Xiaogang ; Wang, Yi ; Li, Xin

Nature communications, 2023-03, Vol.14 (1), p.1401-1401, Article 1401 [Periódico revisado por pares]

England: Nature Publishing Group

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7
[1,2,4]Triazolo[1,5-a]pyrimidine derivative (Mol-5) is a new NS5-RdRp inhibitor of DENV2 proliferation and DENV2-induced inflammation
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Artigo
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[1,2,4]Triazolo[1,5-a]pyrimidine derivative (Mol-5) is a new NS5-RdRp inhibitor of DENV2 proliferation and DENV2-induced inflammation

Wan, Yi-Hong ; Wu, Wen-Yu ; Guo, Song-Xin ; He, Shi-Jun ; Tang, Xiao-Dong ; Wu, Xiao-Yun ; Nandakumar, Kutty Selva ; Zou, Min ; Li, Lin ; Chen, Xiao-Guang ; Liu, Shu-Wen ; Yao, Xin-Gang

Acta pharmacologica Sinica, 2020-05, Vol.41 (5), p.706-718 [Periódico revisado por pares]

United States: Nature Publishing Group

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8
1,25-Dihydroxvitamin D3 attenuates the damage of human immortalised keratinocytes caused by Ultraviolet-B
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1,25-Dihydroxvitamin D3 attenuates the damage of human immortalised keratinocytes caused by Ultraviolet-B

Wang, Pingwei ; Liu, Dongge ; Cui, Jiajing ; Yan, Shuqi ; Liang, Yujun ; Chen, Qianqian ; Liu, Yanping ; Ren, Shuping ; Chen, Peng

Cutaneous and ocular toxicology, 2023-04, Vol.42 (2), p.74-81 [Periódico revisado por pares]

England: Taylor & Francis

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9
1,25‐Dihydroxyvitamin D3 attenuates platelet aggregation potentiated by SARS‐CoV‐2 spike protein via inhibiting integrin αIIbβ3 outside‐in signaling
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1,25‐Dihydroxyvitamin D3 attenuates platelet aggregation potentiated by SARS‐CoV‐2 spike protein via inhibiting integrin αIIbβ3 outside‐in signaling

Wang, Ruijie ; Tian, Zezhong ; Wang, Caixia ; Zhang, Bingying ; Zhu, Meiyan ; Yang, Yan

Cell biochemistry and function, 2024-06, Vol.42 (4), p.e4039-n/a [Periódico revisado por pares]

England: Wiley Subscription Services, Inc

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10
1,25‐dihydroxyvitamin D3‐induced dendritic cells suppress experimental autoimmune encephalomyelitis by increasing proportions of the regulatory lymphocytes and reducing T helper type 1 and type 17 cells
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1,25‐dihydroxyvitamin D3‐induced dendritic cells suppress experimental autoimmune encephalomyelitis by increasing proportions of the regulatory lymphocytes and reducing T helper type 1 and type 17 cells

Xie, Zhongxiang ; Chen, Jingtao ; Zheng, Chao ; Wu, Jing ; Cheng, Yun ; Zhu, Shan ; Lin, Chenhong ; Cao, Qingqing ; Zhu, Jie ; Jin, Tao

Immunology, 2017-11, Vol.152 (3), p.414-424 [Periódico revisado por pares]

Oxford: Wiley Subscription Services, Inc

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