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4-{(2R)-[3-Aminopropionylamido]-3-(2,4-dichlorophenyl)propionyl}-1-{2-[(2-thienyl)ethylaminomethyl]phenyl}piperazine as a Potent and Selective Melanocortin-4 Receptor AntagonistDesign, Synthesis, and Characterization

Chen ; Pontillo, Joseph ; Fleck, Beth A ; Gao, Yinghong ; Wen, Jenny ; Tran, Joe A ; Tucci, Fabio C ; Marinkovic, Dragan ; Foster, Alan C ; Saunders, John

Journal of medicinal chemistry, 2004-12, Vol.47 (27), p.6821-6830 [Periódico revisado por pares]

Washington, DC: American Chemical Society

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