[18F](R)-5-chloro-1-(1-cyclopropyl-2-methoxyethyl)-3-(4-(2-fluoroethoxy)-2,5-dimethyl phenylamino)pyrazin-2(1H)-one: Introduction of N3-phenylpyrazinones as potential CRF-R1 PET imaging agents

Deskus, Jeffrey A. ; Dischino, Douglas D. ; Mattson, Ronald J. ; Ditta, Jonathan L. ; Parker, Michael F. ; Denhart, Derek J. ; Zuev, Dmitry ; Huang, Hong ; Hartz, Richard A. ; Ahuja, Vijay T. ; Wong, Henry ; Mattson, Gail K. ; Molski, Thaddeus F. ; Grace, James E. ; Zueva, Larisa ; Nielsen, Julia M. ; Dulac, Heidi ; Li, Yu-Wen ; Guaraldi, Mary ; Azure, Michael ; Onthank, David ; Hayes, Megan ; Wexler, Eric ; McDonald, Jennifer ; Lodge, Nicholas J. ; Bronson, Joanne J. ; Macor, John E.

Bioorganic & medicinal chemistry letters, 2012-11, Vol.22 (21), p.6651-6655 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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