Identification of a novel series of BET family bromodomain inhibitors: Binding mode and profile of I-BET151 (GSK1210151A)

Seal, Jonathan ; Lamotte, Yann ; Donche, Frédéric ; Bouillot, Anne ; Mirguet, Olivier ; Gellibert, Françoise ; Nicodeme, Edwige ; Krysa, Gael ; Kirilovsky, Jorge ; Beinke, Soren ; McCleary, Scott ; Rioja, Inma ; Bamborough, Paul ; Chung, Chun-Wa ; Gordon, Laurie ; Lewis, Toni ; Walker, Ann L. ; Cutler, Leanne ; Lugo, David ; Wilson, David M. ; Witherington, Jason ; Lee, Kevin ; Prinjha, Rab K.

Bioorganic & medicinal chemistry letters, 2012-04, Vol.22 (8), p.2968-2972 [Periódico revisado por pares]

Amsterdam: Elsevier Ltd

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