Mitigating hERG Inhibition: Design of Orally Bioavailable CCR5 Antagonists as Potent Inhibitors of R5 HIV-1 Replication

Skerlj, Renato ; Bridger, Gary ; Zhou, Yuanxi ; Bourque, Elyse ; McEachern, Ernest ; Danthi, Sanjay ; Langille, Jonathan ; Harwig, Curtis ; Veale, Duane ; Carpenter, Bryon ; Ba, Tuya ; Bey, Michael ; Baird, Ian ; Wilson, Trevor ; Metz, Markus ; MacFarland, Ron ; Mosi, Renee ; Bodart, Veronique ; Wong, Rebecca ; Fricker, Simon ; Huskens, Dana ; Schols, Dominique

ACS medicinal chemistry letters, 2012-03, Vol.3 (3), p.216-221 [Periódico revisado por pares]

United States: American Chemical Society

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